5Y5N
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5y5n by Molmil](/molmil-images/mine/5y5n) | Crystal structure of human Sirtuin 2 in complex with a selective inhibitor | 分子名称: | 2-[[3-(2-phenylethoxy)phenyl]amino]benzamide, NAD-dependent protein deacetylase sirtuin-2, ZINC ION | 著者 | Mellini, P, Itoh, Y, Tsumoto, H, Li, Y, Suzuki, M, Tokuda, N, Kakizawa, T, Miura, Y, Takeuchi, J, Lahtela-Kakkonen, M, Suzuki, T. | 登録日 | 2017-08-09 | 公開日 | 2017-09-06 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Potent mechanism-based sirtuin-2-selective inhibition by anin situ-generated occupant of the substrate-binding site, "selectivity pocket" and NAD+-binding site. Chem Sci, 8, 2017
|
|
4H8K
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4h8k by Molmil](/molmil-images/mine/4h8k) | Crystal structure of LC11-RNase H1 in complex with RNA/DNA hybrid | 分子名称: | DNA (5'-D(*GP*GP*AP*AP*TP*CP*AP*GP*GP*TP*GP*TP*CP*G)-3'), RNA (5'-R(*CP*GP*AP*CP*AP*CP*CP*UP*GP*AP*UP*UP*CP*C)-3'), Ribonuclease H | 著者 | Nguyen, T.N, You, D.J, Matsumoto, H, Kanaya, E, Kanaya, S. | 登録日 | 2012-09-23 | 公開日 | 2013-09-25 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure of metagenome-derived LC11-RNase H1 in complex with RNA/DNA hybrid J.Struct.Biol., 182, 2013
|
|
6KAL
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6kal by Molmil](/molmil-images/mine/6kal) | Crystal structure of FKRP in complex with Mg ion and CMP | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CYTIDINE-5'-MONOPHOSPHATE, Fukutin-related protein, ... | 著者 | Kuwabara, N. | 登録日 | 2019-06-23 | 公開日 | 2020-01-15 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal structures of fukutin-related protein (FKRP), a ribitol-phosphate transferase related to muscular dystrophy. Nat Commun, 11, 2020
|
|
6KAN
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6kan by Molmil](/molmil-images/mine/6kan) | Crystal structure of FKRP in complex with Ba ion | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, BARIUM ION, Fukutin-related protein, ... | 著者 | Kuwabara, N. | 登録日 | 2019-06-23 | 公開日 | 2020-01-15 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.251 Å) | 主引用文献 | Crystal structures of fukutin-related protein (FKRP), a ribitol-phosphate transferase related to muscular dystrophy. Nat Commun, 11, 2020
|
|
6L7U
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6l7u by Molmil](/molmil-images/mine/6l7u) | Crystal structure of FKRP in complex with Ba ion, Ba-SAD data | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, BARIUM ION, Fukutin-related protein, ... | 著者 | Kuwabara, N. | 登録日 | 2019-11-03 | 公開日 | 2020-01-15 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.24 Å) | 主引用文献 | Crystal structures of fukutin-related protein (FKRP), a ribitol-phosphate transferase related to muscular dystrophy. Nat Commun, 11, 2020
|
|
6L7T
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6l7t by Molmil](/molmil-images/mine/6l7t) | |
6L7S
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6l7s by Molmil](/molmil-images/mine/6l7s) | Crystal structure of FKRP in complex with Mg ion, Zinc peak data | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Fukutin-related protein, MAGNESIUM ION, ... | 著者 | Kuwabara, N. | 登録日 | 2019-11-03 | 公開日 | 2020-01-15 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.41 Å) | 主引用文献 | Crystal structures of fukutin-related protein (FKRP), a ribitol-phosphate transferase related to muscular dystrophy. Nat Commun, 11, 2020
|
|
6KAM
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6kam by Molmil](/molmil-images/mine/6kam) | Crystal structure of FKRP in complex with Ba ion, CDP-ribtol, and sugar acceptor | 分子名称: | 2-acetamido-2-deoxy-beta-D-galactopyranose-(1-3)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-alpha-D-mannopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, BARIUM ION, ... | 著者 | Kuwabara, N. | 登録日 | 2019-06-23 | 公開日 | 2020-01-15 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.46 Å) | 主引用文献 | Crystal structures of fukutin-related protein (FKRP), a ribitol-phosphate transferase related to muscular dystrophy. Nat Commun, 11, 2020
|
|
6KAK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6kak by Molmil](/molmil-images/mine/6kak) | Crystal structure of FKRP in complex with Mg ion | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Fukutin-related protein, MAGNESIUM ION, ... | 著者 | Kuwabara, N. | 登録日 | 2019-06-23 | 公開日 | 2020-01-15 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.056 Å) | 主引用文献 | Crystal structures of fukutin-related protein (FKRP), a ribitol-phosphate transferase related to muscular dystrophy. Nat Commun, 11, 2020
|
|
6KAJ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6kaj by Molmil](/molmil-images/mine/6kaj) | Crystal structure of FKRP in complex with Ba ion | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, BARIUM ION, CYTIDINE-5'-DIPHOSPHATE, ... | 著者 | Kuwabara, N. | 登録日 | 2019-06-23 | 公開日 | 2020-01-29 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.2249 Å) | 主引用文献 | Crystal structures of fukutin-related protein (FKRP), a ribitol-phosphate transferase related to muscular dystrophy. Nat Commun, 11, 2020
|
|
4X86
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4x86 by Molmil](/molmil-images/mine/4x86) | Crystal structure of BAG6-Ubl4a complex | 分子名称: | 3-[(3-CHOLAMIDOPROPYL)DIMETHYLAMMONIO]-1-PROPANESULFONATE, Large proline-rich protein BAG6, SULFATE ION, ... | 著者 | Kuwabara, N, Kato, R. | 登録日 | 2014-12-10 | 公開日 | 2015-02-25 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Structure of a BAG6 (Bcl-2-associated Athanogene 6)-Ubl4a (Ubiquitin-like Protein 4a) Complex Reveals a Novel Binding Interface That Functions in Tail-anchored Protein Biogenesis J.Biol.Chem., 290, 2015
|
|
3A2O
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3a2o by Molmil](/molmil-images/mine/3a2o) | Crystal Structure of HIV-1 Protease Complexed with KNI-1689 | 分子名称: | (4R)-3-[(2S,3S)-3-{[(4-amino-2,6-dimethylphenoxy)acetyl]amino}-2-hydroxy-4-phenylbutanoyl]-5,5-dimethyl-N-(2-methylprop -2-en-1-yl)-1,3-thiazolidine-4-carboxamide, GLYCEROL, PROTEASE | 著者 | Adachi, M, Tamada, T, Hidaka, K, Kimura, T, Kiso, Y, Kuroki, R. | 登録日 | 2009-05-26 | 公開日 | 2010-03-02 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (0.88 Å) | 主引用文献 | Small-sized human immunodeficiency virus type-1 protease inhibitors containing allophenylnorstatine to explore the S2' pocket. J.Med.Chem., 52, 2009
|
|