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7AQT
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BU of 7aqt by Molmil
NMR2 structure of BRD4-BD2 in complex with iBET-762
分子名称: 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide, Bromodomain-containing protein 4
著者Orts, J, Torres, F, Milbradt, A.G, Walser, R.
登録日2020-10-23
公開日2022-03-02
最終更新日2024-06-19
実験手法SOLUTION NMR
主引用文献NMR Molecular Replacement Provides New Insights into Binding Modes to Bromodomains of BRD4 and TRIM24.
J.Med.Chem., 65, 2022
7B9X
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BU of 7b9x by Molmil
NMR2 structure of TRIM24-BD in complex with a precursor of IACS-9571
分子名称: N-{6-[3-(4-Aminobutoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl}-3,4-dimethoxybenzene-1-sulfonamide, Transcription intermediary factor 1-alpha
著者Orts, J, Torres, F, Milbradt, A.G, Walser, R.
登録日2020-12-14
公開日2022-01-12
最終更新日2024-06-19
実験手法SOLUTION NMR
主引用文献NMR Molecular Replacement Provides New Insights into Binding Modes to Bromodomains of BRD4 and TRIM24.
J.Med.Chem., 65, 2022
8CA0
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BU of 8ca0 by Molmil
Macrophage inhibitory factor (MIF) in complex with small molecule PAV174
分子名称: 1-ethyl-9-methyl-3,7-dipyrrolidin-1-yl-phenothiazine, Macrophage migration inhibitory factor
著者Mueller, A, Torres, F, Roland, R, Korth, C.
登録日2023-01-24
公開日2024-02-07
実験手法SOLUTION NMR
主引用文献Oxidized MIF is a drug target at the molecular intersection between immune activation and tau cellular pathology
To Be Published
8OVI
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BU of 8ovi by Molmil
BRICHOS monomer
分子名称: Pulmonary surfactant-associated protein C (Fragment)
著者Ghosh, D, Torres, F, Guentert, P, Riek, R.
登録日2023-04-26
公開日2024-06-26
実験手法SOLUTION NMR
主引用文献The inhibitory action of the chaperone BRICHOS against the alpha-Synuclein secondary nucleation pathway at near-atomic resolution
To Be Published
8OX2
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BU of 8ox2 by Molmil
BRICHOS trimer
分子名称: Pulmonary surfactant-associated protein C
著者Ghosh, D, Torres, F, Guentert, P, Riek, R.
登録日2023-04-30
公開日2024-06-26
実験手法SOLUTION NMR
主引用文献The inhibitory action of the chaperone BRICHOS against the alpha-Synuclein secondary nucleation pathway at near-atomic resolution
To Be Published
1OCU
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BU of 1ocu by Molmil
Crystal structure of the yeast PX-domain protein Grd19p (sorting nexin 3) complexed to phosphatidylinosytol-3-phosphate.
分子名称: 2-(BUTANOYLOXY)-1-{[(HYDROXY{[2,3,4,6-TETRAHYDROXY-5-(PHOSPHONOOXY)CYCLOHEXYL]OXY}PHOSPHORYL)OXY]METHYL}ETHYL BUTANOATE, SORTING NEXIN
著者Zhou, C.Z, Li de La Sierra-Gallay, I, Cheruel, S, Collinet, B, Minard, P, Blondeau, K, Henkes, G, Aufrere, R, Leulliot, N, Graille, M, Sorel, I, Savarin, P, de la Torre, F, Poupon, A, Janin, J, van Tilbeurgh, H.
登録日2003-02-10
公開日2003-12-12
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of the yeast Phox homology (PX) domain protein Grd19p complexed to phosphatidylinositol-3-phosphate.
J. Biol. Chem., 278, 2003
1OCS
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BU of 1ocs by Molmil
Crystal structure of the yeast PX-doamin protein Grd19p (sorting nexin3) complexed to phosphatidylinosytol-3-phosphate.
分子名称: GLYCEROL, SORTING NEXIN GRD19
著者Zhou, C.Z, Li De La Sierra-Gallay, I, Cheruel, S, Collinet, B, Minard, P, Blondeau, K, Henkes, G, Aufrere, R, Leulliot, N, Graille, M, Sorel, I, Savarin, P, De La Torre, F, Poupon, A, Janin, J, Van Tilbeurgh, H.
登録日2003-02-10
公開日2003-12-12
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献Crystal Structure of the Yeast Phox Homology (Px) Protein Grd19P (Sorting Nexin 3) Complexed to Phosphatidylinositol-3-Phosphate
J.Biol.Chem., 278, 2003

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件を2024-07-03に公開中

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