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7QYR
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BU of 7qyr by Molmil
Crystal structure of RimK from Pseudomonas aeruginosa PAO1
分子名称: ADENOSINE-5'-DIPHOSPHATE, Probable alpha-L-glutamate ligase, poly-glutamate
著者Thompson, C.M.A, Little, R.H, Stevenson, C.E.M, Lawson, D.M, Malone, J.G.
登録日2022-01-29
公開日2022-10-05
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural insights into the mechanism of adaptive ribosomal modification by Pseudomonas RimK.
Proteins, 91, 2023
7QYS
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BU of 7qys by Molmil
Crystal structure of RimK from Pseudomonas syringae DC3000
分子名称: ADENOSINE-5'-DIPHOSPHATE, Probable alpha-L-glutamate ligase
著者Thompson, C.M.A, Little, R.H, Stevenson, C.E.M, Lawson, D.M, Malone, J.G.
登録日2022-01-29
公開日2022-10-05
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural insights into the mechanism of adaptive ribosomal modification by Pseudomonas RimK.
Proteins, 91, 2023
3KBY
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BU of 3kby by Molmil
Crystal structure of hypothetical protein from Staphylococcus aureus
分子名称: 1,2-ETHANEDIOL, Putative uncharacterized protein
著者Lam, R, Thompson, C.M, Battaile, K.P, Romanov, V, Kisselman, G, Gordon, E, Pai, E.F, Chirgadze, N.Y.
登録日2009-10-20
公開日2010-10-20
最終更新日2017-11-01
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of hypothetical protein from Staphylococcus aureus
To be Published
3L5A
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BU of 3l5a by Molmil
Crystal structure of a probable NADH-dependent flavin oxidoreductase from Staphylococcus aureus
分子名称: NADH/flavin oxidoreductase/NADH oxidase, TRIETHYLENE GLYCOL
著者Lam, R, Gordon, R.D, Vodsedalek, J, Battaile, K.P, Grebemeskel, S, Lam, K, Romanov, V, Chan, T, Mihajlovic, V, Thompson, C.M, Guthrie, J, Pai, E.F, Chirgadze, N.Y.
登録日2009-12-21
公開日2010-12-22
最終更新日2018-01-24
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Crystal structure of a probable NADH-dependent flavin oxidoreductase from Staphylococcus aureus
To be Published
3KWL
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BU of 3kwl by Molmil
Crystal structure of a hypothetical protein from Helicobacter pylori
分子名称: uncharacterized protein
著者Lam, R, Thompson, C.M, Vodsedalek, J, Lam, K, Romanov, V, Battaile, K.P, Beletskaya, I, Gordon, E, Pai, E.F, Chirgadze, N.Y.
登録日2009-12-01
公開日2010-12-01
最終更新日2017-11-01
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Crystal structure of a hypothetical protein from Helicobacter pylori
To be Published
1M7Q
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BU of 1m7q by Molmil
Crystal structure of p38 MAP kinase in complex with a dihydroquinazolinone inhibitor
分子名称: 1-(2,6-DICHLOROPHENYL)-5-(2,4-DIFLUOROPHENYL)-7-PIPERAZIN-1-YL-3,4-DIHYDROQUINAZOLIN-2(1H)-ONE, Mitogen-activated protein kinase 14, SULFATE ION
著者Stelmach, J.E, Liu, L, Patel, S.B, Pivnichny, J.V, Scapin, G, Singh, S, Hop, C.E.C.A, Wang, Z, Cameron, P.M, Nichols, E.A, O'Keefe, S.J, O'Neill, E.A, Schmatz, D.M, Schwartz, C.D, Thompson, C.M, Zaller, D.M, Doherty, J.B.
登録日2002-07-22
公開日2002-12-11
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Design and synthesis of potent, orally bioavailable dihydroquinazolinone inhibitors of p38 MAP kinase.
Bioorg.Med.Chem.Lett., 13, 2003
1OVE
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BU of 1ove by Molmil
The structure of p38 alpha in complex with a dihydroquinolinone
分子名称: 1-(2,6-DICHLOROPHENYL)-5-(2,4-DIFLUOROPHENYL)-7-PIPERIDIN-4-YL-3,4-DIHYDROQUINOLIN-2(1H)-ONE, GLYCEROL, Mitogen-activated protein kinase 14
著者Fitzgerald, C.E, Patel, S.B, Becker, J.W, Cameron, P.M, Zaller, D, Pikounis, V.B, O'Keefe, S.J, Scapin, G.
登録日2003-03-26
公開日2003-09-02
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural basis for p38alpha MAP kinase quinazolinone and pyridol-pyrimidine inhibitor specificity
Nat.Struct.Biol., 10, 2003
1OUY
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BU of 1ouy by Molmil
The structure of p38 alpha in complex with a dihydropyrido-pyrimidine inhibitor
分子名称: 1-(2,6-DICHLOROPHENYL)-6-[(2,4-DIFLUOROPHENYL)SULFANYL]-7-(1,2,3,6-TETRAHYDRO-4-PYRIDINYL)-3,4-DIHYDROPYRIDO[3,2-D]PYRIMIDIN-2(1H)-ONE, Mitogen-activated protein kinase 14
著者Fitzgerald, C.E, Patel, S.B, Becker, J.W, Cameron, P.M, Zaller, D, Pikounis, V.B, O'Keefe, S.J, Scapin, G.
登録日2003-03-25
公開日2003-09-02
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural basis for p38alpha MAP kinase quinazolinone and pyridol-pyrimidine inhibitor specificity
Nat.Struct.Biol., 10, 2003
1A8T
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BU of 1a8t by Molmil
METALLO-BETA-LACTAMASE IN COMPLEX WITH L-159,061
分子名称: 2-BUTYL-6-HYDROXY-3-[2'-(1H-TETRAZOL-5-YL)-BIPHENYL-4-YLMETHYL]-3H-QUINAZOLIN-4-ONE, METALLO-BETA-LACTAMASE, ZINC ION
著者Fitzgerald, P.M.D, Toney, J.H, Grover, N, Vanderwall, D.
登録日1998-03-23
公開日1998-10-14
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Antibiotic sensitization using biphenyl tetrazoles as potent inhibitors of Bacteroides fragilis metallo-beta-lactamase.
Chem.Biol., 5, 1998
1A7T
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BU of 1a7t by Molmil
METALLO-BETA-LACTAMASE WITH MES
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, METALLO-BETA-LACTAMASE, SODIUM ION, ...
著者Fitzgerald, P.M.D, Wu, J.K, Toney, J.H.
登録日1998-03-17
公開日1998-06-17
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Unanticipated inhibition of the metallo-beta-lactamase from Bacteroides fragilis by 4-morpholineethanesulfonic acid (MES): a crystallographic study at 1.85-A resolution.
Biochemistry, 37, 1998
6THK
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BU of 6thk by Molmil
Structural mechanism of pyocin S5 import into Pseudomonas aeruginosa
分子名称: GLYCEROL, Pyocin S5, ZINC ION
著者Behrens, H.M, Kleanthous, C, Lowe, E.D.
登録日2019-11-20
公開日2020-03-04
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Pyocin S5 Import into Pseudomonas aeruginosa Reveals a Generic Mode of Bacteriocin Transport.
Mbio, 11, 2020

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件を2024-07-10に公開中

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