7CNL
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![BU of 7cnl by Molmil](/molmil-images/mine/7cnl) | Crystal structure of TEAD3 in complex with VT105 | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, N-[(1S)-1-pyridin-2-ylethyl]-8-[4-(trifluoromethyl)phenyl]quinoline-3-carboxamide, ... | 著者 | Tang, T.T, Konradi, A.W. | 登録日 | 2020-08-01 | 公開日 | 2021-04-28 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Small Molecule Inhibitors of TEAD Auto-palmitoylation Selectively Inhibit Proliferation and Tumor Growth of NF2 -deficient Mesothelioma. Mol.Cancer Ther., 20, 2021
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8PQO
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![BU of 8pqo by Molmil](/molmil-images/mine/8pqo) | PITP in complex with the inhibitor VT01545 | 分子名称: | (2~{R})-2-azanyl-3-[(2~{S},3~{R})-2-methyl-5-oxidanylidene-pyrrolidin-3-yl]sulfanyl-propanal, (2~{R})-3-methyl-2-(methylamino)butanoic acid, (2~{R})-4-methyl-2-(methylamino)pentanamide, ... | 著者 | Boura, E, Eisenreichova, A. | 登録日 | 2023-07-11 | 公開日 | 2024-05-08 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Non-vesicular phosphatidylinositol transfer plays critical roles in defining organelle lipid composition. Embo J., 43, 2024
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