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7VKO
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BU of 7vko by Molmil
Crystal structure of TrkA kinase with repotrectinib
分子名称: Repotrectinib, SULFATE ION, Tyrosine-protein kinase receptor
著者Murray, B.W, Rogers, E, Zhai, D, Deng, W, Chen, X, Sprengeler, P.A, Zhang, X, Graber, A, Reich, S.H, Stopatschinskaja, S, Solomon, B, Besse, B, Drilon, A.
登録日2021-09-30
公開日2021-10-13
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Molecular Characteristics of Repotrectinib That Enable Potent Inhibition of TRK Fusion Proteins and Resistant Mutations.
Mol.Cancer Ther., 20, 2021
7VKM
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BU of 7vkm by Molmil
Crystal structure of TrkA (G595R) kinase domain
分子名称: Tyrosine-protein kinase receptor
著者Murray, B.W, Rogers, E, Zhai, D, Deng, W, Chen, X, Sprengeler, P.A, Zhang, X, Graber, A, Reich, S.H, Stopatschinskaja, S, Solomon, B, Besse, B, Drilon, A.
登録日2021-09-30
公開日2021-10-13
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Molecular Characteristics of Repotrectinib That Enable Potent Inhibition of TRK Fusion Proteins and Resistant Mutations.
Mol.Cancer Ther., 20, 2021
7VKN
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BU of 7vkn by Molmil
Crystal structure of TrkA (G595R) kinase with repotrectinib
分子名称: Repotrectinib, SULFATE ION, Tyrosine-protein kinase receptor
著者Murray, B.W, Rogers, E, Zhai, D, Deng, W, Chen, X, Sprengeler, P.A, Zhang, X, Graber, A, Reich, S.H, Stopatschinskaja, S, Solomon, B, Besse, B, Drilon, A.
登録日2021-09-30
公開日2021-10-13
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Molecular Characteristics of Repotrectinib That Enable Potent Inhibition of TRK Fusion Proteins and Resistant Mutations.
Mol.Cancer Ther., 20, 2021
8TKM
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BU of 8tkm by Molmil
Murine NF-kappaB p50 Rel Homology Region homodimer in complex with 17-mer kappaB DNA from human interleukin-6 (IL-6) promoter
分子名称: 17-mer kappaB DNA, Nuclear factor NF-kappa-B p50 subunit
著者Zhu, N, Mealka, M, Mitchel, S, Rogers, W.E, Huxford, T.
登録日2023-07-25
公開日2023-10-11
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献X-ray Crystallographic Study of Preferred Spacing by the NF-kappa B p50 Homodimer on kappa B DNA.
Biomolecules, 13, 2023
8TKN
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BU of 8tkn by Molmil
Murine NF-kappaB p50 Rel Homology Region homodimer in complex with 10-mer kappaB DNA from human Neutrophil Gelatinase-associated Lipocalin (NGAL) promoter
分子名称: DNA A, DNA B, Nuclear factor NF-kappa-B p50 subunit
著者Zhu, N, Mealka, M, Mitchel, S, Rogers, W.E, Huxford, T.
登録日2023-07-25
公開日2023-10-11
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献X-ray Crystallographic Study of Preferred Spacing by the NF-kappa B p50 Homodimer on kappa B DNA.
Biomolecules, 13, 2023
8TKL
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BU of 8tkl by Molmil
Murine NF-kappaB p50 Rel Homology Region homodimer in complex with a Test 16-mer kappaB-like DNA
分子名称: Nuclear factor NF-kappa-B p50 subunit, Test 17-mer kappaB-like DNA
著者Mitchel, S, Mealka, M, Rogers, W.E, Milani, C, Acuna, L.M, Huxford, T.
登録日2023-07-25
公開日2023-10-18
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献X-ray Crystallographic Study of Preferred Spacing by the NF-kappa B p50 Homodimer on kappa B DNA.
Biomolecules, 13, 2023

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件を2024-06-12に公開中

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