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1S1G
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BU of 1s1g by Molmil
Crystal Structure of Kv4.3 T1 Domain
分子名称: Potassium voltage-gated channel subfamily D member 3, ZINC ION
著者Scannevin, R.H, Wang, K.W, Jow, F, Megules, J, Kopsco, D.C, Edris, W, Carroll, K.C, Lu, Q, Xu, W.X, Xu, Z.B, Katz, A.H, Olland, S, Lin, L, Taylor, M, Stahl, M, Malakian, K, Somers, W, Mosyak, L, Bowlby, M.R, Chanda, P, Rhodes, K.J.
登録日2004-01-06
公開日2004-03-23
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Two N-terminal domains of Kv4 K(+) channels regulate binding to and modulation by KChIP1.
Neuron, 41, 2004
1S1E
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BU of 1s1e by Molmil
Crystal Structure of Kv Channel-interacting protein 1 (KChIP-1)
分子名称: CALCIUM ION, Kv channel interacting protein 1
著者Scannevin, R.H, Wang, K.-W, Jow, F, Megules, J, Kopsco, D.C, Edris, W, Carroll, K.C, Lu, Q, Xu, W.-X, Xu, Z.-B, Katz, A.H, Olland, S, Lin, L, Taylor, M, Stahl, M, Malakian, K, Somers, W, Mosyak, L, Bowlby, M.R, Chanda, P, Rhodes, K.J.
登録日2004-01-06
公開日2005-01-11
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Two N-terminal domains of Kv4 K(+) channels regulate binding to and modulation by KChIP1.
Neuron, 41, 2004
6AR4
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BU of 6ar4 by Molmil
Crystal structure of PICK1 in complex with the small molecule inhibitor 1o
分子名称: N-[4-(4-bromophenyl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carbonyl]-3-cyclopropyl-L-alanine, PRKCA-binding protein
著者Marcotte, D.
登録日2017-08-21
公開日2018-08-22
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Potent PDZ-Domain PICK1 Inhibitors that Modulate Amyloid Beta-Mediated Synaptic Dysfunction.
Sci Rep, 8, 2018
5UE3
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BU of 5ue3 by Molmil
proMMP-9desFnII
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CALCIUM ION, Matrix metalloproteinase-9, ...
著者Alexander, R.S, Spurlino, J, Milligan, C.
登録日2016-12-29
公開日2017-09-13
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.599 Å)
主引用文献Discovery of a highly selective chemical inhibitor of matrix metalloproteinase-9 (MMP-9) that allosterically inhibits zymogen activation.
J. Biol. Chem., 292, 2017
5UE4
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BU of 5ue4 by Molmil
proMMP-9desFnII complexed to JNJ0966 INHIBITOR
分子名称: CALCIUM ION, Matrix metalloproteinase-9, SULFATE ION, ...
著者Alexander, R.S, Spurlino, J, Milligan, C.
登録日2016-12-29
公開日2017-09-13
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Discovery of a highly selective chemical inhibitor of matrix metalloproteinase-9 (MMP-9) that allosterically inhibits zymogen activation.
J. Biol. Chem., 292, 2017

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件を2024-06-12に公開中

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