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5H3Q
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BU of 5h3q by Molmil
Crystal Structure of TrkA kinase with ligand
分子名称: 1-[(3S,4R)-4-[3,4-bis(fluoranyl)phenyl]-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(5-ethoxy-4-methyl-2-phenyl-pyrazol-3-yl)urea, 2,3-DIHYDROXY-1,4-DITHIOBUTANE, High affinity nerve growth factor receptor, ...
著者Noritaka, F.
登録日2016-10-26
公開日2017-02-22
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The juxtamembrane region of TrkA kinase is critical for inhibitor selectivity
Bioorg. Med. Chem. Lett., 27, 2017
6IQN
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BU of 6iqn by Molmil
Crystal structure of TrkA kinase with ligand
分子名称: 4-[[4-azanyl-3-(4-cyclohexylpiperazin-1-yl)-9,10-bis(oxidanylidene)anthracen-1-yl]amino]benzoic acid, High affinity nerve growth factor receptor
著者Noritaka, F.
登録日2018-11-08
公開日2020-01-22
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.54 Å)
主引用文献An isoform-selective inhibitor of tropomyosin receptor kinase A behaves as molecular glue.
Bioorg.Med.Chem.Lett., 30, 2020

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件を2024-07-31に公開中

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