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1IAJ
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CRYSTAL STRUCTURE OF THE ATYPICAL PROTEIN KINASE DOMAIN OF A TRP CA-CHANNEL, CHAK (APO)
分子名称: TRANSIENT RECEPTOR POTENTIAL-RELATED PROTEIN, ZINC ION
著者Yamaguchi, H, Matsushita, M, Nairn, A.C, Kuriyan, J.
登録日2001-03-22
公開日2001-06-06
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structure of the atypical protein kinase domain of a TRP channel with phosphotransferase activity.
Mol.Cell, 7, 2001
1IAH
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BU of 1iah by Molmil
CRYSTAL STRUCTURE OF THE ATYPICAL PROTEIN KINASE DOMAIN OF A TRP CA-CHANNEL, CHAK (ADP-MG COMPLEX)
分子名称: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Yamaguchi, H, Matsushita, M, Nairn, A.C, Kuriyan, J.
登録日2001-03-22
公開日2001-06-06
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structure of the atypical protein kinase domain of a TRP channel with phosphotransferase activity.
Mol.Cell, 7, 2001
1IA9
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CRYSTAL STRUCTURE OF THE ATYPICAL PROTEIN KINASE DOMAIN OF A TRP CA-CHANNEL, CHAK (AMPPNP COMPLEX)
分子名称: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, TRANSIENT RECEPTOR POTENTIAL-RELATED PROTEIN, ...
著者Yamaguchi, H, Matsushita, M, Nairn, A.C, Kuriyan, J.
登録日2001-03-22
公開日2001-06-06
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of the atypical protein kinase domain of a TRP channel with phosphotransferase activity.
Mol.Cell, 7, 2001
1HKX
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BU of 1hkx by Molmil
Crystal structure of calcium/calmodulin-dependent protein kinase
分子名称: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE TYPE II ALPHA CHAIN, CHLORIDE ION, ...
著者Hoelz, A, Nairn, A.C, Kuriyan, J.
登録日2003-03-12
公開日2003-06-02
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Crystal Structure of a Tetradecameric Assembly of the Association Domain of Ca2+/Calmodulin-Dependent Kinase II
Mol.Cell, 11, 2003
1FJM
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Protein serine/threonine phosphatase-1 (alpha isoform, type 1) complexed with microcystin-LR toxin
分子名称: BETA-MERCAPTOETHANOL, MANGANESE (II) ION, PROTEIN SERINE/THREONINE PHOSPHATASE-1 (ALPHA ISOFORM, ...
著者Goldberg, J, Nairn, A.C, Kuriyan, J.
登録日1995-12-17
公開日1996-06-20
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Three-dimensional structure of the catalytic subunit of protein serine/threonine phosphatase-1.
Nature, 376, 1995
1A06
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BU of 1a06 by Molmil
CALMODULIN-DEPENDENT PROTEIN KINASE FROM RAT
分子名称: CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE
著者Kuriyan, J, Goldberg, J.
登録日1997-12-09
公開日1998-04-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural basis for the autoinhibition of calcium/calmodulin-dependent protein kinase I.
Cell(Cambridge,Mass.), 84, 1996
2BDW
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BU of 2bdw by Molmil
Crystal Structure of the Auto-Inhibited Kinase Domain of Calcium/Calmodulin Activated Kinase II
分子名称: Hypothetical protein K11E8.1d
著者Rosenberg, O.S, Kuriyan, J.
登録日2005-10-20
公開日2005-12-13
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure of the Autoinhibited Kinase Domain of CaMKII and SAXS Analysis of the Holoenzyme
Cell(Cambridge,Mass.), 123, 2005
3EGG
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BU of 3egg by Molmil
Crystal structure of a complex between Protein Phosphatase 1 alpha (PP1) and the PP1 binding and PDZ domains of Spinophilin
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GLYCEROL, MANGANESE (II) ION, ...
著者Ragusa, M.J, Page, R, Peti, W.
登録日2008-09-10
公開日2010-03-23
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Spinophilin directs protein phosphatase 1 specificity by blocking substrate binding sites.
Nat.Struct.Mol.Biol., 17, 2010
3EGH
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Crystal structure of a complex between Protein Phosphatase 1 alpha (PP1), the PP1 binding and PDZ domains of Spinophilin and the small natural molecular toxin Nodularin-R
分子名称: GLYCEROL, MANGANESE (II) ION, Serine/threonine-protein phosphatase PP1-alpha catalytic subunit, ...
著者Ragusa, M.J, Page, R, Peti, W.
登録日2008-09-10
公開日2010-03-23
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Spinophilin directs protein phosphatase 1 specificity by blocking substrate binding sites.
Nat.Struct.Mol.Biol., 17, 2010
2FN5
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BU of 2fn5 by Molmil
NMR Structure of the Neurabin PDZ domain (502-594)
分子名称: Neurabin-1
著者Dancheck, B, Peti, W.
登録日2006-01-10
公開日2007-01-09
最終更新日2024-05-08
実験手法SOLUTION NMR
主引用文献Structural basis for spinophilin-neurabin receptor interaction.
Biochemistry, 46, 2007
2G5M
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Spinophilin PDZ domain
分子名称: Neurabin-2
著者Kelker, M.S, Peti, W.
登録日2006-02-23
公開日2007-01-09
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Structural basis for spinophilin-neurabin receptor interaction.
Biochemistry, 46, 2007
2GLE
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BU of 2gle by Molmil
Solution structure of neurabin SAM domain
分子名称: Neurabin-1
著者Ju, T, Hudak, J, Peti, W.
登録日2006-04-04
公開日2007-03-13
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Structural characterization of the neurabin SAM domain
TO BE PUBLISHED
2F86
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BU of 2f86 by Molmil
The Association Domain of C. elegans CaMKII
分子名称: Hypothetical protein K11E8.1d
著者Rosenberg, O.S, Kuriyan, J.
登録日2005-12-01
公開日2006-02-07
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.64 Å)
主引用文献Oligomerization states of the association domain and the holoenyzme of Ca2+/CaM kinase II.
Febs J., 273, 2006
4MOV
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BU of 4mov by Molmil
1.45 A Resolution Crystal Structure of Protein Phosphatase 1
分子名称: CHLORIDE ION, MANGANESE (II) ION, PHOSPHATE ION, ...
著者Choy, M.S, Peti, W, Page, R.
登録日2013-09-12
公開日2014-03-26
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.4503 Å)
主引用文献Understanding the antagonism of retinoblastoma protein dephosphorylation by PNUTS provides insights into the PP1 regulatory code.
Proc.Natl.Acad.Sci.USA, 111, 2014
4MOY
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BU of 4moy by Molmil
Structure of a second nuclear PP1 Holoenzyme, crystal form 1
分子名称: CHLORIDE ION, GLYCEROL, MANGANESE (II) ION, ...
著者Choy, M.S, Hieke, M, Peti, W, Page, R.
登録日2013-09-12
公開日2014-03-26
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.1953 Å)
主引用文献Understanding the antagonism of retinoblastoma protein dephosphorylation by PNUTS provides insights into the PP1 regulatory code.
Proc.Natl.Acad.Sci.USA, 111, 2014
4MP0
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BU of 4mp0 by Molmil
Structure of a second nuclear PP1 Holoenzyme, crystal form 2
分子名称: GLYCEROL, MANGANESE (II) ION, PHOSPHATE ION, ...
著者Choy, M.S, Hieke, M, Peti, W, Page, R.
登録日2013-09-12
公開日2014-03-26
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.1003 Å)
主引用文献Understanding the antagonism of retinoblastoma protein dephosphorylation by PNUTS provides insights into the PP1 regulatory code.
Proc.Natl.Acad.Sci.USA, 111, 2014
3HVQ
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BU of 3hvq by Molmil
Crystal structure of a complex between Protein Phosphatase 1 alpha (PP1) and the PP1 binding and PDZ domains of Neurabin
分子名称: GLYCEROL, MANGANESE (II) ION, Neurabin-1, ...
著者Critton, D.A, Ragusa, M.J, Page, R, Peti, W.
登録日2009-06-16
公開日2010-03-23
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Spinophilin directs protein phosphatase 1 specificity by blocking substrate binding sites.
Nat.Struct.Mol.Biol., 17, 2010
1LCM
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BU of 1lcm by Molmil
NMR minimized average structure of microcystin-LR
分子名称: microcystin LR
著者Trogen, G, Zdunek, J.
登録日1995-12-30
公開日1996-12-07
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Conformational studies of microcystin-LR using NMR spectroscopy and molecular dynamics calculations.
Biochemistry, 35, 1996
5OVR
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BU of 5ovr by Molmil
X-Ray Characterization of Striatal-Enriched Protein Tyrosine Phosphatase Inhibitors
分子名称: Tyrosine-protein phosphatase non-receptor type 5, [(~{S})-[4-[3-[(~{R})-(3,4-dichlorophenyl)-oxidanyl-methyl]phenyl]phenyl]-oxidanyl-methyl]phosphonic acid
著者Kack, H, Wissler, L.
登録日2017-08-29
公開日2017-11-22
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献X-ray Characterization and Structure-Based Optimization of Striatal-Enriched Protein Tyrosine Phosphatase Inhibitors.
J. Med. Chem., 60, 2017
5OVX
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X-Ray Characterization of Striatal-Enriched Protein Tyrosine Phosphatase Inhibitors
分子名称: Tyrosine-protein phosphatase non-receptor type 5, [(~{S})-[4-[3-[(~{S})-(3,4-dichlorophenyl)-oxidanyl-methyl]phenyl]phenyl]-oxidanyl-methyl]phosphonic acid
著者Kack, H, Wissler, L.
登録日2017-08-30
公開日2017-11-22
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献X-ray Characterization and Structure-Based Optimization of Striatal-Enriched Protein Tyrosine Phosphatase Inhibitors.
J. Med. Chem., 60, 2017
5OW1
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BU of 5ow1 by Molmil
X-Ray Characterization of Striatal-Enriched Protein Tyrosine Phosphatase Inhibitors
分子名称: Tyrosine-protein phosphatase non-receptor type 5, [[3-(3-cyclohexyl-2-oxidanyl-phenyl)phenyl]-bis(fluoranyl)methyl]phosphonic acid
著者Kack, H, Wissler, L.
登録日2017-08-30
公開日2017-11-22
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献X-ray Characterization and Structure-Based Optimization of Striatal-Enriched Protein Tyrosine Phosphatase Inhibitors.
J. Med. Chem., 60, 2017
1CDK
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CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT (E.C.2.7.1.37) (PROTEIN KINASE A) COMPLEXED WITH PROTEIN KINASE INHIBITOR PEPTIDE FRAGMENT 5-24 (PKI(5-24) ISOELECTRIC VARIANT CA) AND MN2+ ADENYLYL IMIDODIPHOSPHATE (MNAMP-PNP) AT PH 5.6 AND 7C AND 4C
分子名称: CAMP-DEPENDENT PROTEIN KINASE, MANGANESE (II) ION, MYRISTIC ACID, ...
著者Bossemeyer, D, Engh, R.A, Kinzel, V, Ponstingl, H, Huber, R.
登録日1994-07-04
公開日1995-10-15
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Phosphotransferase and substrate binding mechanism of the cAMP-dependent protein kinase catalytic subunit from porcine heart as deduced from the 2.0 A structure of the complex with Mn2+ adenylyl imidodiphosphate and inhibitor peptide PKI(5-24).
EMBO J., 12, 1993
1EVB
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NMR structure of cyanobacterial toxin, phosphatase-1/-2A inhibitor
分子名称: MICROCYSTIN-LR
著者Bagu, J.R, Sykes, B.D.
登録日1996-02-14
公開日1996-11-08
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Comparison of the solution structures of microcystin-LR and motuporin.
Nat.Struct.Biol., 2, 1995
1EVA
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NMR structure of cyanobacterial toxin, phosphatase-1/-2A inhibitor
分子名称: MICROCYSTIN-LR
著者Bagu, J.R, Sykes, B.D.
登録日1996-02-14
公開日1996-11-08
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Comparison of the solution structures of microcystin-LR and motuporin.
Nat.Struct.Biol., 2, 1995

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