8A1A
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![BU of 8a1a by Molmil](/molmil-images/mine/8a1a) | Structure of a leucinostatin derivative determined by host lattice display : L1F11V1 construct | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one, ... | 著者 | Mittl, P.R.E. | 登録日 | 2022-06-01 | 公開日 | 2022-12-07 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structure of a hydrophobic leucinostatin derivative determined by host lattice display. Acta Crystallogr D Struct Biol, 78, 2022
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8A19
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![BU of 8a19 by Molmil](/molmil-images/mine/8a19) | Structure of a leucinostatin derivative determined by host lattice display : L1E4V1 construct | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one, ... | 著者 | Mittl, P.R.E. | 登録日 | 2022-06-01 | 公開日 | 2022-12-07 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.358 Å) | 主引用文献 | Structure of a hydrophobic leucinostatin derivative determined by host lattice display. Acta Crystallogr D Struct Biol, 78, 2022
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7BHE
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![BU of 7bhe by Molmil](/molmil-images/mine/7bhe) | DARPin_D5/Her3 domain 4 complex, monoclinic crystals | 分子名称: | ACETATE ION, DARPin_D5, GLYCEROL, ... | 著者 | Mittl, P.R.E, Radom, F, Pluckthun, A. | 登録日 | 2021-01-11 | 公開日 | 2021-11-24 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.297 Å) | 主引用文献 | Crystal structures of HER3 extracellular domain 4 in complex with the designed ankyrin-repeat protein D5. Acta Crystallogr.,Sect.F, 77, 2021
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7BHF
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![BU of 7bhf by Molmil](/molmil-images/mine/7bhf) | DARPin_D5/Her3 domain 4 complex, orthorhombic crystals | 分子名称: | ACETATE ION, DARPin_D5, Isoform 4 of Receptor tyrosine-protein kinase erbB-3 | 著者 | Mittl, P.R.E, Radom, F, Pluckthun, A. | 登録日 | 2021-01-11 | 公開日 | 2021-11-24 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.997 Å) | 主引用文献 | Crystal structures of HER3 extracellular domain 4 in complex with the designed ankyrin-repeat protein D5. Acta Crystallogr.,Sect.F, 77, 2021
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1GET
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![BU of 1get by Molmil](/molmil-images/mine/1get) | |
1GES
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![BU of 1ges by Molmil](/molmil-images/mine/1ges) | |
1GEU
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![BU of 1geu by Molmil](/molmil-images/mine/1geu) | |
2DKO
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![BU of 2dko by Molmil](/molmil-images/mine/2dko) | Extended substrate recognition in caspase-3 revealed by high resolution X-ray structure analysis | 分子名称: | Caspase-3, PHQ-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE | 著者 | Mittl, P.R.E, Ganesan, R, Jelakovic, S, Grutter, M.G. | 登録日 | 2006-04-12 | 公開日 | 2006-07-04 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.06 Å) | 主引用文献 | Extended Substrate Recognition in Caspase-3 Revealed by High Resolution X-ray Structure Analysis J.Mol.Biol., 359, 2006
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1AIE
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![BU of 1aie by Molmil](/molmil-images/mine/1aie) | |
5OD1
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![BU of 5od1 by Molmil](/molmil-images/mine/5od1) | Structure of the engineered metalloesterase MID1sc10 complexed with a phosphonate transition state analogue | 分子名称: | GLYCEROL, MID1sc10, ZINC ION, ... | 著者 | Mittl, P.R.E, Studer, S, Hansen, D.A, Hilvert, D. | 登録日 | 2017-07-04 | 公開日 | 2018-12-12 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.34 Å) | 主引用文献 | Evolution of a highly active and enantiospecific metalloenzyme from short peptides. Science, 362, 2018
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8QBC
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![BU of 8qbc by Molmil](/molmil-images/mine/8qbc) | Reactive amide intermediate in sperm whale myoglobin mutant H64V V68A | 分子名称: | ACETATE ION, Myoglobin, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Tinzl, M, Mittl, P.R.E, Hilvert, D. | 登録日 | 2023-08-24 | 公開日 | 2023-12-13 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.23 Å) | 主引用文献 | Myoglobin-Catalyzed Azide Reduction Proceeds via an Anionic Metal Amide Intermediate. J.Am.Chem.Soc., 146, 2024
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8QBA
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![BU of 8qba by Molmil](/molmil-images/mine/8qba) | Sperm whale myoblogin mutant H64V V68A in complex with glycine ethyl ester | 分子名称: | ACETATE ION, Myoglobin, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Tinzl, M, Mittl, P.R.E, Hilvert, D. | 登録日 | 2023-08-24 | 公開日 | 2023-12-13 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.39 Å) | 主引用文献 | Myoglobin-Catalyzed Azide Reduction Proceeds via an Anionic Metal Amide Intermediate. J.Am.Chem.Soc., 146, 2024
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2CJX
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![BU of 2cjx by Molmil](/molmil-images/mine/2cjx) | Extended substrate recognition in caspase-3 revealed by high resolution X-ray structure analysis | 分子名称: | CASPASE-3, PHQ-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE | 著者 | Ganesan, R, Mittl, P.R.E, Jelakovic, S, Grutter, M.G. | 登録日 | 2006-04-09 | 公開日 | 2006-06-27 | 最終更新日 | 2017-06-28 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Extended Substrate Recognition in Caspase-3 Revealed by High Resolution X-Ray Structure Analysis J.Mol.Biol., 359, 2006
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2CJY
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![BU of 2cjy by Molmil](/molmil-images/mine/2cjy) | Extended substrate recognition in caspase-3 revealed by high resolution X-ray structure analysis | 分子名称: | CASPASE-3, PHQ-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE | 著者 | Ganesan, R, Mittl, P.R.E, Jelakovic, S, Grutter, M.G. | 登録日 | 2006-04-09 | 公開日 | 2006-06-27 | 最終更新日 | 2017-06-28 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Extended Substrate Recognition in Caspase-3 Revealed by High Resolution X-Ray Structure Analysis J.Mol.Biol., 359, 2006
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7QNP
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![BU of 7qnp by Molmil](/molmil-images/mine/7qnp) | Designed Armadillo repeat protein N(A4)M4C(AII) co-crystallized with hen egg white lysozyme | 分子名称: | 1,2-ETHANEDIOL, 1,4-DIETHYLENE DIOXIDE, Designed Armadillo Repeat Protein N(A4)M4C(AII), ... | 著者 | Michel, E, Mittl, P.R.E, Plueckthun, A. | 登録日 | 2021-12-21 | 公開日 | 2022-06-08 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.586 Å) | 主引用文献 | Improved Repeat Protein Stability by Combined Consensus and Computational Protein Design. Biochemistry, 62, 2023
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5OD9
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![BU of 5od9 by Molmil](/molmil-images/mine/5od9) | Structure of the engineered metalloesterase MID1sc9 | 分子名称: | (2~{S})-2-phenylpropanoic acid, 1,2-ETHANEDIOL, CHLORIDE ION, ... | 著者 | Studer, S, Mittl, P.R.E, Hilvert, D. | 登録日 | 2017-07-05 | 公開日 | 2018-12-12 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.13 Å) | 主引用文献 | Evolution of a highly active and enantiospecific metalloenzyme from short peptides. Science, 362, 2018
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6QEP
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![BU of 6qep by Molmil](/molmil-images/mine/6qep) | EngBF DARPin Fusion 4b H14 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, MANGANESE (II) ION, ... | 著者 | Ernst, P, Pluckthun, A, Mittl, P.R.E. | 登録日 | 2019-01-08 | 公開日 | 2019-11-06 | 最終更新日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural analysis of biological targets by host:guest crystal lattice engineering. Sci Rep, 9, 2019
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6QFO
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![BU of 6qfo by Molmil](/molmil-images/mine/6qfo) | EngBF DARPin Fusion 9b 3G124 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, MANGANESE (II) ION, ... | 著者 | Ernst, P, Pluckthun, A, Mittl, P.R.E. | 登録日 | 2019-01-10 | 公開日 | 2019-11-06 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural analysis of biological targets by host:guest crystal lattice engineering. Sci Rep, 9, 2019
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6QEV
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![BU of 6qev by Molmil](/molmil-images/mine/6qev) | EngBF DARPin Fusion 4b B6 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, MANGANESE (II) ION, PEGA domain-containing protein,PEGA domain-containing protein,EngBF DARPin fusion B6 complex, ... | 著者 | Ernst, P, Pluckthun, A, Mittl, P.R.E. | 登録日 | 2019-01-08 | 公開日 | 2019-11-06 | 最終更新日 | 2020-04-22 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structural analysis of biological targets by host:guest crystal lattice engineering. Sci Rep, 9, 2019
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6QFK
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![BU of 6qfk by Molmil](/molmil-images/mine/6qfk) | EngBF DARPin Fusion 4b G10 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ... | 著者 | Ernst, P, Pluckthun, A, Mittl, P.R.E. | 登録日 | 2019-01-10 | 公開日 | 2019-11-06 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural analysis of biological targets by host:guest crystal lattice engineering. Sci Rep, 9, 2019
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6SA7
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![BU of 6sa7 by Molmil](/molmil-images/mine/6sa7) | DARPin-Armadillo fusion C8long83 | 分子名称: | DARPin-Armadillo fusion C8long83 | 著者 | Ernst, P, Honegger, A, van der Valk, F, Ewald, C, Mittl, P.R.E, Plucktun, A. | 登録日 | 2019-07-16 | 公開日 | 2019-11-20 | 最終更新日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (3.3 Å) | 主引用文献 | Rigid fusions of designed helical repeat binding proteins efficiently protect a binding surface from crystal contacts. Sci Rep, 9, 2019
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6SA8
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![BU of 6sa8 by Molmil](/molmil-images/mine/6sa8) | ring-like DARPin-Armadillo fusion H83_D01 | 分子名称: | 1,2-ETHANEDIOL, LYS-ARG-LYS-ARG-LYS-ARG-LYS-ARG-LYS-ARG, ring-like DARPin-Armadillo fusion H83_D01 | 著者 | Ernst, P, Honegger, A, van der Valk, F, Ewald, C, Mittl, P.R.E, Plucktun, A. | 登録日 | 2019-07-16 | 公開日 | 2019-11-20 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Rigid fusions of designed helical repeat binding proteins efficiently protect a binding surface from crystal contacts. Sci Rep, 9, 2019
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6SH9
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![BU of 6sh9 by Molmil](/molmil-images/mine/6sh9) | EngBF DARPin Fusion 4b D12 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Endo-alpha-N-acetylgalactosaminidase,DARPin 4b D12, ... | 著者 | Ernst, P, Pluckthun, A, Mittl, P.R.E. | 登録日 | 2019-08-06 | 公開日 | 2019-11-06 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural analysis of biological targets by host:guest crystal lattice engineering. Sci Rep, 9, 2019
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6SA6
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![BU of 6sa6 by Molmil](/molmil-images/mine/6sa6) | DARPin-Armadillo fusion A5 | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, DARPin-Armadillo fusion A5 | 著者 | Ernst, P, Honegger, A, van der Valk, F, Ewald, C, Mittl, P.R.E, Pluckthun, A. | 登録日 | 2019-07-16 | 公開日 | 2019-11-20 | 最終更新日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Rigid fusions of designed helical repeat binding proteins efficiently protect a binding surface from crystal contacts. Sci Rep, 9, 2019
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4BS0
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![BU of 4bs0 by Molmil](/molmil-images/mine/4bs0) | Crystal Structure of Kemp Eliminase HG3.17 E47N,N300D Complexed with Transition State Analog 6-Nitrobenzotriazole | 分子名称: | 6-NITROBENZOTRIAZOLE, KEMP ELIMINASE HG3.17, SULFATE ION | 著者 | Blomberg, R, Kries, H, Pinkas, D.M, Mittl, P.R.E, Gruetter, M.G, Privett, H.K, Mayo, S, Hilvert, D. | 登録日 | 2013-06-06 | 公開日 | 2013-10-16 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.09 Å) | 主引用文献 | Precision is Essential for Efficient Catalysis in an Evolved Kemp Eliminase Nature, 503, 2013
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