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1XMK
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BU of 1xmk by Molmil
The Crystal structure of the Zb domain from the RNA editing enzyme ADAR1
分子名称: CADMIUM ION, CHLORIDE ION, Double-stranded RNA-specific adenosine deaminase, ...
著者Athanasiadis, A, Placido, D, Maas, S, Brown II, B.A, Lowenhaupt, K, Rich, A.
登録日2004-10-03
公開日2005-08-02
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (0.97 Å)
主引用文献The Crystal Structure of the Z[beta] Domain of the RNA-editing Enzyme ADAR1 Reveals Distinct Conserved Surfaces Among Z-domains.
J.Mol.Biol., 351, 2005
8RIJ
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BU of 8rij by Molmil
Discovery of the first orally bioavailable ADAMTS7 inhibitor BAY-9835
分子名称: CALCIUM ION, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ...
著者Schafer, M, Meibom, D, Wasnaire, P, Beyer, K, Broehl, A, Cancho-Grande, Y, Elowe, N, Henninger, K, Johannes, S, Jungmann, N, Krainz, T, Lindner, N, Maassen, S, MacDonald, B, Menshykau, D, Mittendorf, J, Sanchez, G, Stefan, E, Torge, A, Xing, Y, Zubov, D.
登録日2023-12-18
公開日2024-02-21
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献BAY-9835: Discovery of the First Orally Bioavailable ADAMTS7 Inhibitor.
J.Med.Chem., 67, 2024
8BPY
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BU of 8bpy by Molmil
X-RAY STRUCTURE OF PDE9A IN COMPLEX WITH Inhibitor 13A
分子名称: (8~{S})-6-[2-(2,3-dihydroindol-1-yl)-2-oxidanylidene-ethyl]-4-(4-methylphenyl)-2-oxidanylidene-8-propyl-1,5,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile, High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A, MAGNESIUM ION, ...
著者Steuber, H.
登録日2022-11-18
公開日2022-12-28
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献BAY-7081: A Potent, Selective, and Orally Bioavailable Cyanopyridone-Based PDE9A Inhibitor.
J.Med.Chem., 65, 2022

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件を2024-07-17に公開中

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