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8TQS
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BU of 8tqs by Molmil
Complex of human thrombin (S195A) bound to a bivalent inhibitor comprised of DNA Aptamer HD22 conjugated to Dabigatran with a linker.
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, DNA (30-MER), ...
著者Krishnaswamy, S, Kumar, S.
登録日2023-08-08
公開日2024-05-01
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.207 Å)
主引用文献Aptameric hirudins as selective and reversible EXosite-ACTive site (EXACT) inhibitors.
Nat Commun, 15, 2024
5VOF
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BU of 5vof by Molmil
DesGla-XaS195A Bound to Aptamer 11F7t and Rivaroxaban
分子名称: 5-chloro-N-({(5S)-2-oxo-3-[4-(3-oxomorpholin-4-yl)phenyl]-1,3-oxazolidin-5-yl}methyl)thiophene-2-carboxamide, CALCIUM ION, Coagulation factor X, ...
著者Krishnaswamy, S, Kumar, S.
登録日2017-05-02
公開日2018-06-13
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Combination of aptamer and drug for reversible anticoagulation in cardiopulmonary bypass.
Nat. Biotechnol., 36, 2018
4PTN
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BU of 4ptn by Molmil
Crystal Structure of YagE, a KDG aldolase protein in complex with Magnesium cation coordinated L-glyceraldehyde
分子名称: 1,2-ETHANEDIOL, GLYCEROL, L-glyceraldehyde, ...
著者Manoj Kumar, P, Baskar, V, Manicka, S, Krishnaswamy, S.
登録日2014-03-11
公開日2014-12-03
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Crystal structure of YagE, a putative DHDPS-like protein from Escherichia coli K12.
Proteins, 71, 2008
4U4M
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BU of 4u4m by Molmil
Crystal structure of 0.5M urea unfolded YagE, a KDG aldolase protein in complex with Pyruvate
分子名称: 1,2-ETHANEDIOL, PYRUVIC ACID, UREA, ...
著者Manoj Kumar, P, Bhaskar, V, Manicka, S, Krishnaswamy, S.
登録日2014-07-24
公開日2015-07-29
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3.09 Å)
主引用文献Crystal structure of 0.5M urea unfolded YagE, a KDG aldolase protein in complex with Pyruvate
To be published
4OE7
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BU of 4oe7 by Molmil
Crystal structure of YagE, a KDG aldolase protein, in complex with aldol condensed product of pyruvate and glyoxal
分子名称: (4R)-4-hydroxy-2,5-dioxopentanoic acid, (4S)-4-hydroxy-2,5-dioxopentanoic acid, 1,2-ETHANEDIOL, ...
著者Manoj Kumar, P, Baskar, V, Manicka, S, Krishnaswamy, S.
登録日2014-01-12
公開日2014-12-24
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Crystal structure of YagE, a KDG aldolase protein, in complex with aldol condensed product of pyruvate and glyoxal
To be Published
4ONV
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BU of 4onv by Molmil
Crystal structure of YagE, a KDG aldolase protein in complex with 2-Keto-3-deoxy gluconate
分子名称: 1,2-ETHANEDIOL, 2-KETO-3-DEOXYGLUCONATE, GLYCEROL, ...
著者Manoj Kumar, P, Bhaskar, V, Manicka, S, Krishnaswamy, S.
登録日2014-01-29
公開日2015-01-14
実験手法X-RAY DIFFRACTION (2.57 Å)
主引用文献Crystal structure of YagE, a KDG aldolase protein in complex with 2-Keto-3-deoxy gluconate
To be Published
2BPA
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BU of 2bpa by Molmil
ATOMIC STRUCTURE OF SINGLE-STRANDED DNA BACTERIOPHAGE PHIX174 AND ITS FUNCTIONAL IMPLICATIONS
分子名称: DNA (5'-D(*AP*AP*AP*AP*C)-3'), PROTEIN (SUBUNIT OF BACTERIOPHAGE PHIX174)
著者McKenna, R, Xia, D, Willingmann, P, Ilag, L.L, Krishnaswamy, S, Rossmann, M.G, Olson, N.H, Baker, T.S, Incardona, N.L.
登録日1991-12-03
公開日1991-12-03
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Atomic structure of single-stranded DNA bacteriophage phi X174 and its functional implications.
Nature, 355, 1992
3JTC
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BU of 3jtc by Molmil
Importance of Mg2+ in the Ca2+-Dependent Folding of the gamma-Carboxyglutamic Acid Domains of Vitamin K-Dependent clotting and anticlotting Proteins
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Endothelial protein C receptor, ...
著者Bajaj, S.P, Vadivel, K, Agah, S, Cascio, D, Krishnaswamy, S, Esmon, C, Padmanabhan, K.
登録日2009-09-11
公開日2011-04-06
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural and Functional Studies of gamma-Carboxyglutamic Acid Domains of Factor VIIa and Activated Protein C: Role of Magnesium at Physiological Calcium.
J.Mol.Biol., 425, 2013
4ZPU
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BU of 4zpu by Molmil
The structure of DLP12 endolysin exhibits likely active and inactive conformations.
分子名称: ACETATE ION, FORMIC ACID, Lysozyme RrrD
著者Kesavan, B, Arockiasamy, A, Krishnaswamy, S.
登録日2015-05-08
公開日2015-06-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The structure of DLP12 endolysin exhibits likely an active and inactive conformations.
To Be Published
239D
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BU of 239d by Molmil
POLYMORPHISM IN LEFT HANDED DNA: THE CRYSTAL STRUCTURE OF D(CCCGGG)2
分子名称: DNA (5'-D(*CP*CP*CP*GP*GP*G)-3')
著者Karthe, P, Krishnaswamy, S, Gautham, N.
登録日1995-11-02
公開日1996-11-08
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Polymorphism in Left Handed DNA: The Crystal Structure of d(CCCGGG)2
To be Published, 1996
4BXW
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BU of 4bxw by Molmil
Crystal Structure of the Prothrombinase Complex from the Venom of Pseudonaja Textilis
分子名称: COAGULATION FACTOR V, FACTOR XA, GLYCEROL, ...
著者Lechtenberg, B.C, Murray-Rust, T.A, Johnson, D.J.D, Adams, T.E, Krishnaswamy, S, Camire, R.M, Huntington, J.A.
登録日2013-07-16
公開日2013-07-31
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.71 Å)
主引用文献Crystal Structure of the Prothrombinase Complex from the Venom of Pseudonaja Textilis.
Blood, 122, 2013
4BXS
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BU of 4bxs by Molmil
Crystal Structure of the Prothrombinase Complex from the Venom of Pseudonaja Textilis
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Lechtenberg, B.C, Murray-Rust, T.A, Johnson, D.J.D, Adams, T.E, Krishnaswamy, S, Camire, R.M, Huntington, J.A.
登録日2013-07-15
公開日2013-07-31
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.32 Å)
主引用文献Crystal Structure of the Prothrombinase Complex from the Venom of Pseudonaja Textilis.
Blood, 122, 2013
3NEV
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BU of 3nev by Molmil
Crystal structure of YagE, a prophage protein from E. coli K12 in complex with KDGal
分子名称: 1,2-ETHANEDIOL, 3-DEOXY-D-LYXO-HEXONIC ACID, Uncharacterized protein yagE
著者Bhaskar, V, Kumar, P.M, Manicka, S, Krishnaswamy, S.
登録日2010-06-09
公開日2011-04-13
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献Identification of biochemical and putative biological role of a xenolog from Escherichia coli using structural analysis.
Proteins, 79, 2011
3N2X
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BU of 3n2x by Molmil
Crystal structure of YagE, a prophage protein belonging to the dihydrodipicolinic acid synthase family from E. coli K12 in complex with pyruvate
分子名称: 1,2-ETHANEDIOL, Uncharacterized protein yagE
著者Bhaskar, V, Kumar, P.M, Manicka, S, Krishnaswamy, S.
登録日2010-05-19
公開日2011-04-13
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Identification of biochemical and putative biological role of a xenolog from Escherichia coli using structural analysis.
Proteins, 79, 2011
8EPC
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BU of 8epc by Molmil
Crystal structure of human coagulation factor IXa (S195A), apo-form
分子名称: CALCIUM ION, Coagulation factor IXa heavy chain, Coagulation factor IXa light chain
著者Kolyadko, V.N, Krishnaswamy, S.
登録日2022-10-05
公開日2024-07-03
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Allosteric Control of Coagulation Factor IXa via Its Exosite II Regulates Blood Clotting
Proc.Natl.Acad.Sci.USA, 2024
8EPH
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BU of 8eph by Molmil
Crystal structure of human coagulation factor IXa (S195A), apo-form, DES-GLA
分子名称: CALCIUM ION, Coagulation factor IXa heavy chain, Coagulation factor IXa light chain, ...
著者Kolyadko, V.N, Krishnaswamy, S.
登録日2022-10-05
公開日2024-07-03
実験手法X-RAY DIFFRACTION (1.88 Å)
主引用文献Allosteric Control of Coagulation Factor IXa via Its Exosite II Regulates Blood Clotting
Proc.Natl.Acad.Sci.USA, 2024
8EPK
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BU of 8epk by Molmil
Complex of anticoagulant RNA aptamer and human coagulation factor IXa (S195A)
分子名称: CALCIUM ION, Coagulation factor IXa heavy chain, Coagulation factor IXa light chain, ...
著者Kolyadko, V.N, Krishnaswamy, S.
登録日2022-10-05
公開日2024-07-03
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Allosteric Control of Coagulation Factor IXa via Its Exosite II Regulates Blood Clotting
Proc.Natl.Acad.Sci.USA, 2024
3NSG
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BU of 3nsg by Molmil
Crystal Structure of OmpF, an Outer Membrane Protein from Salmonella typhi
分子名称: CITRATE ANION, GLYCEROL, L(+)-TARTARIC ACID, ...
著者Balasubramaniam, D, Arockiasamy, A, Sharma, A, Krishnaswamy, S.
登録日2010-07-01
公開日2011-07-13
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.79 Å)
主引用文献Asymmetric pore occupancy in crystal structure of OmpF porin from Salmonella typhi
J.Struct.Biol., 178, 2012
2RMU
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BU of 2rmu by Molmil
THREE-DIMENSIONAL STRUCTURES OF DRUG-RESISTANT MUTANTS OF HUMAN RHINOVIRUS 14
分子名称: HUMAN RHINOVIRUS 14 COAT PROTEIN (SUBUNIT VP1), HUMAN RHINOVIRUS 14 COAT PROTEIN (SUBUNIT VP2), HUMAN RHINOVIRUS 14 COAT PROTEIN (SUBUNIT VP3), ...
著者Badger, J, Krishnaswamy, S, Kremer, M.J, Oliveira, M.A, Rossmann, M.G, Heinz, B.A, Rueckert, R.R, Dutko, F.J, Mckinlay, M.A.
登録日1988-10-03
公開日1990-01-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Three-dimensional structures of drug-resistant mutants of human rhinovirus 14.
J.Mol.Biol., 207, 1989
2J4U
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BU of 2j4u by Molmil
E.coli OmpC - camel Lactoferrin complex
分子名称: LACTOTRANSFERRIN, OUTER MEMBRANE PROTEIN C PRECURSOR
著者Baalaji, S, Acharya, R.K, Singh, T.P, Krishnaswamy, S.
登録日2006-09-06
公開日2007-02-13
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.99 Å)
主引用文献Crystal Structure of the Membrane Protein Ompc Complex with Antibacterial Lactoferrin
To be Published
1RMU
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BU of 1rmu by Molmil
THREE-DIMENSIONAL STRUCTURES OF DRUG-RESISTANT MUTANTS OF HUMAN RHINOVIRUS 14
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, HUMAN RHINOVIRUS 14 COAT PROTEIN (SUBUNIT VP1), HUMAN RHINOVIRUS 14 COAT PROTEIN (SUBUNIT VP2), ...
著者Badger, J, Krishnaswamy, S, Kremer, M.J, Oliveira, M.A, Rossmann, M.G, Heinz, B.A, Rueckert, R.R, Dutko, F.J, Mckinlay, M.A.
登録日1988-10-03
公開日1990-01-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Three-dimensional structures of drug-resistant mutants of human rhinovirus 14.
J.Mol.Biol., 207, 1989
2V9D
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BU of 2v9d by Molmil
Crystal Structure of YagE, a prophage protein belonging to the dihydrodipicolinic acid synthase family from E. coli K12
分子名称: YAGE
著者Manicka, S, Peleg, Y, Unger, T, Albeck, S, Dym, O, Greenblatt, H.M, Bourenkov, G, Lamzin, V, Krishnaswamy, S, Sussman, J.L.
登録日2007-08-23
公開日2008-03-04
最終更新日2019-11-06
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Crystal Structure of Yage, a Putative Dhdps Like Protein from Escherichia Coli K12.
Proteins: Struct., Funct., Bioinf., 71, 2008
4KR8
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BU of 4kr8 by Molmil
Salmonella typhi OmpF complex with Daunomycin
分子名称: DAUNOMYCIN, Outer membrane protein F
著者Madhuranayaki, T, Balasubramaniam, D, Krishnaswamy, S.
登録日2013-05-16
公開日2014-05-28
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Salmonella typhi OmpF complex with Daunomycin
To be published
2V8Z
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BU of 2v8z by Molmil
Crystal Structure of YagE, a prophage protein belonging to the dihydrodipicolinic acid synthase family from E. coli K12
分子名称: YAGE
著者Manicka, S, Peleg, Y, Unger, T, Albeck, S, Dym, O, Greenblatt, H.M, Bourenkov, G, Lamzin, V, Krishnaswamy, S, Sussman, J.L.
登録日2007-08-16
公開日2008-03-04
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal Structure of Yage, a Putative Dhdps Like Protein from Escherichia Coli K12.
Proteins: Struct., Funct., Bioinf., 71, 2008
4KRA
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BU of 4kra by Molmil
Salmonella typhi OmpF complex with Ciprofloxacin
分子名称: 1-CYCLOPROPYL-6-FLUORO-4-OXO-7-PIPERAZIN-1-YL-1,4-DIHYDROQUINOLINE-3-CARBOXYLIC ACID, Outer membrane protein F
著者Madhuranayaki, T, Balasubramaniam, D, Krishnaswamy, S.
登録日2013-05-16
公開日2014-05-28
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (3.32 Å)
主引用文献Salmonella typhi OmpF complex with Ciprofloxacin
To be published

 

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