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3PUP
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BU of 3pup by Molmil
Structure of Glycogen Synthase Kinase 3 beta (GSK3B) in complex with a ruthenium octasporine ligand (OS1)
分子名称: Glycogen synthase kinase-3 beta, Ruthenium octasporine
著者Filippakopoulos, P, Kraling, K, Essen, L.O, Meggers, E, Knapp, S.
登録日2010-12-06
公開日2010-12-22
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.99 Å)
主引用文献Structurally sophisticated octahedral metal complexes as highly selective protein kinase inhibitors.
J.Am.Chem.Soc., 133, 2011
4AS0
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BU of 4as0 by Molmil
Cyclometalated Phthalimides as Protein Kinase Inhibitors
分子名称: PHTALIMIDE-RUTHENIUM COMPLEX, SERINE/THREONINE-PROTEIN KINASE PIM-1
著者Blanck, S, Geisselbrecht, Y, Middel, S, Mietke, T, Harms, K, Essen, L.-O, Meggers, E.
登録日2012-04-27
公開日2012-10-03
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Bioactive Cyclometalated Phthalimides: Design, Synthesis and Kinase Inhibition.
Dalton Trans, 41, 2012
3WE8
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BU of 3we8 by Molmil
Pim-1 kinase in complex with Ruthenium-based inhibitor
分子名称: Cyclopentadienyl(carbon monoxide)(7-oxo-7,10-dihydro-1,8-phenanthrolin-10-yl-kappa~2~C~10~,N~1~)ruthenium, SULFATE ION, Serine/threonine-protein kinase pim-1
著者Waehler, K, Kraeling, K, Steuber, H, Meggers, E.
登録日2013-07-02
公開日2014-05-21
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.954 Å)
主引用文献Non-ATP-Mimetic Organometallic Protein Kinase Inhibitor
ChemistryOpen, 2, 2013

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件を2024-08-28に公開中

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