3TDD
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![BU of 3tdd by Molmil](/molmil-images/mine/3tdd) | Crystal structure of yeast CP in complex with Belactosin C | 分子名称: | Proteasome component C1, Proteasome component C11, Proteasome component C5, ... | 著者 | Korotkov, V.S, Ludwig, A, Larionov, O.V, Lygin, A.V, Groll, M, de Meijere, A. | 登録日 | 2011-08-10 | 公開日 | 2011-10-12 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Synthesis and biological activity of optimized belactosin C congeners. Org.Biomol.Chem., 9, 2011
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6H23
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![BU of 6h23 by Molmil](/molmil-images/mine/6h23) | Crystal structure of the hClpP Y118A mutant with an activating small molecule | 分子名称: | 1,2-ETHANEDIOL, ATP-dependent Clp protease proteolytic subunit, mitochondrial, ... | 著者 | Kick, L.M, Sieber, S.A, Schneider, S. | 登録日 | 2018-07-13 | 公開日 | 2018-08-29 | 最終更新日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (3.089 Å) | 主引用文献 | Selective Activation of Human Caseinolytic Protease P (ClpP). Angew. Chem. Int. Ed. Engl., 57, 2018
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5DL1
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![BU of 5dl1 by Molmil](/molmil-images/mine/5dl1) | ClpP from Staphylococcus aureus in complex with AV145 | 分子名称: | 1-(propan-2-yl)-N-{[2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-pyrazolo[3,4-b]pyridine-5-carboxamide, ATP-dependent Clp protease proteolytic subunit | 著者 | Vielberg, M.-T, Groll, M. | 登録日 | 2015-09-04 | 公開日 | 2015-11-25 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Reversible Inhibitors Arrest ClpP in a Defined Conformational State that Can Be Revoked by ClpX Association. Angew.Chem.Int.Ed.Engl., 54, 2015
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4Z1L
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![BU of 4z1l by Molmil](/molmil-images/mine/4z1l) | Yeast 20S proteasome in complex with belactosin C derivative 3 | 分子名称: | (2S,3S)-2-{(1R)-2-[(3,5-dimethoxybenzyl)amino]-1-hydroxy-2-oxoethyl}-3-methylpentanoic acid, CHLORIDE ION, MAGNESIUM ION, ... | 著者 | Huber, E.M, Groll, M. | 登録日 | 2015-03-27 | 公開日 | 2015-05-27 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | A Minimal beta-Lactone Fragment for Selective beta 5c or beta 5i Proteasome Inhibitors. Angew.Chem.Int.Ed.Engl., 54, 2015
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