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4AN1
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BU of 4an1 by Molmil
PROLYL OLIGOPEPTIDASE FROM PORCINE BRAIN WITH A COVALENTLY BOUND INHIBITOR IC-4
分子名称: (2S)-N-benzyl-2-({(2S)-2-[(1R)-1,2-dihydroxyethyl]pyrrolidin-1-yl}carbonyl)pyrrolidine-1-carboxamide, GLYCEROL, PROLYL ENDOPEPTIDASE
著者Kaszuba, K, Rog, T, Danne, R, Canning, P, Fulop, V, Juhasz, T, Szeltner, Z, St-Pierre, J.F, Garcia-Horsman, A, Mannisto, P.T, Karttunen, M, Hokkanen, J, Bunker, A.
登録日2012-03-14
公開日2012-05-16
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Molecular Dynamics, Crystallography and Mutagenesis Studies on the Substrate Gating Mechanism of Prolyl Oligopeptidase.
Biochimie, 94, 2012
4AN0
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BU of 4an0 by Molmil
PROLYL OLIGOPEPTIDASE FROM PORCINE BRAIN WITH A COVALENTLY BOUND INHIBITOR IC-3
分子名称: (2S)-1-[1-(4-phenylbutanoyl)-L-prolyl]pyrrolidine-2-carbonitrile, GLYCEROL, PROLYL ENDOPEPTIDASE
著者Kaszuba, K, Rog, T, Danne, R, Canning, P, Fulop, V, Juhasz, T, Szeltner, Z, St-Pierre, J.F, Garcia-Horsman, A, Mannisto, P.T, Karttunen, M, Hokkanen, J, Bunker, A.
登録日2012-03-14
公開日2012-05-16
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Molecular dynamics, crystallography and mutagenesis studies on the substrate gating mechanism of prolyl oligopeptidase.
Biochimie, 94, 2012
4AMY
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BU of 4amy by Molmil
PROLYL OLIGOPEPTIDASE FROM PORCINE BRAIN WITH A COVALENTLY BOUND INHIBITOR IC-1
分子名称: 1-[(2R,5S)-2-tert-butyl-5-({(2S)-2-[(1R)-1,2-dihydroxyethyl]pyrrolidin-1-yl}carbonyl)pyrrolidin-1-yl]-4-phenylbutan-1-one, GLYCEROL, PROLYL ENDOPEPTIDASE
著者Kaszuba, K, Rog, T, Danne, R, Canning, P, Fulop, V, Juhasz, T, Szeltner, Z, St-Pierre, J.F, Garcia-Horsman, A, Mannisto, P.T, Karttunen, M, Hokkanen, J, Bunker, A.
登録日2012-03-14
公開日2012-05-16
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Molecular Dynamics, Crystallography and Mutagenesis Studies on the Substrate Gating Mechanism of Prolyl Oligopeptidase.
Biochimie, 94, 2012
4AMZ
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BU of 4amz by Molmil
PROLYL OLIGOPEPTIDASE FROM PORCINE BRAIN WITH A COVALENTLY BOUND INHIBITOR IC-2
分子名称: (5R)-N-benzyl-5-({(2S)-2-[(1R)-1,2-dihydroxyethyl]pyrrolidin-1-yl}carbonyl)cyclopent-1-ene-1-carboxamide, GLYCEROL, PROLYL ENDOPEPTIDASE
著者Kaszuba, K, Rog, T, Danne, R, Canning, P, Fulop, V, Juhasz, T, Szeltner, Z, St-Pierre, J.F, Garcia-Horsman, A, Mannisto, P.T, Karttunen, M, Hokkanen, J, Bunker, A.
登録日2012-03-14
公開日2012-05-16
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Molecular Dynamics, Crystallography and Mutagenesis Studies on the Substrate Gating Mechanism of Prolyl Oligopeptidase.
Biochimie, 94, 2012
6QV0
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BU of 6qv0 by Molmil
Structure of ATP-bound outward-facing TM287/288 in complex with sybody Sb_TM35
分子名称: ABC transporter, ATP-binding protein, ADENOSINE-5'-TRIPHOSPHATE, ...
著者Hutter, C.A.J, Huerlimann, L.M, Zimmermann, I, Egloff, P, Seeger, M.A.
登録日2019-03-01
公開日2019-05-29
最終更新日2019-06-05
実験手法X-RAY DIFFRACTION (3.12 Å)
主引用文献The extracellular gate shapes the energy profile of an ABC exporter.
Nat Commun, 10, 2019
6QV2
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BU of 6qv2 by Molmil
Structure of ATPgS-bound outward-facing TM287/288 in complex with nanobody Nb_TM#2
分子名称: ABC transporter, ATP-binding protein, MAGNESIUM ION, ...
著者Hutter, C.A.J, Huerlimann, L.M, Zimmermann, I, Egloff, P, Seeger, M.A.
登録日2019-03-01
公開日2019-05-29
最終更新日2019-06-05
実験手法X-RAY DIFFRACTION (4.23 Å)
主引用文献The extracellular gate shapes the energy profile of an ABC exporter.
Nat Commun, 10, 2019
6QV1
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BU of 6qv1 by Molmil
Structure of ATPgS-bound outward-facing TM287/288 in complex with nanobody Nb_TM1
分子名称: ABC transporter, ATP-binding protein, MAGNESIUM ION, ...
著者Hutter, C.A.J, Huerlimann, L.M, Zimmermann, I, Egloff, P, Seeger, M.A.
登録日2019-03-01
公開日2019-05-29
最終更新日2019-06-05
実験手法X-RAY DIFFRACTION (3.48 Å)
主引用文献The extracellular gate shapes the energy profile of an ABC exporter.
Nat Commun, 10, 2019
6QUZ
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BU of 6quz by Molmil
Structure of ATPgS-bound outward-facing TM287/288 in complex with sybody Sb_TM35
分子名称: ABC transporter, ATP-binding protein, MAGNESIUM ION, ...
著者Hutter, C.A.J, Huerlimann, L.M, Zimmermann, I, Egloff, P, Seeger, M.A.
登録日2019-03-01
公開日2019-05-29
最終更新日2019-06-05
実験手法X-RAY DIFFRACTION (3.21 Å)
主引用文献The extracellular gate shapes the energy profile of an ABC exporter.
Nat Commun, 10, 2019

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件を2024-09-04に公開中

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