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BU of 3p9j by Molmil

Aurora A kinase domain with phthalazinone pyrazole inhibitor
分子名称:	4-[(5-methyl-1H-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2H)-one, Serine/threonine-protein kinase 6
著者	Kairies, N.A, Oliveira, T, Engh, R.A.
登録日	2010-10-17
公開日	2011-03-23
最終更新日	2024-02-21
実験手法	X-RAY DIFFRACTION (2.8 Å)
主引用文献	Phthalazinone pyrazoles as potent, selective, and orally bioavailable inhibitors of aurora-a kinase. J.Med.Chem., 54, 2011

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BU of 1yoj by Molmil

Crystal structure of Src kinase domain
分子名称:	proto-oncogene tyrosine-protein kinase SRC
著者	Breitenlechner, C.B, Kairies, N.A, Honold, K, Scheiblich, S, Koll, H, Greiter, E, Koch, S, Schaefer, W, Huber, R, Engh, R.A.
登録日	2005-01-27
公開日	2006-01-27
最終更新日	2024-04-03
実験手法	X-RAY DIFFRACTION (1.95 Å)
主引用文献	Crystal structures of active SRC kinase domain complexes J.Mol.Biol., 353, 2005

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BU of 1yol by Molmil

Crystal structure of Src kinase domain in complex with CGP77675
分子名称:	1-{4-[4-AMINO-5-(3-METHOXYPHENYL)-7H-PYRROLO[2,3-D]PYRIMIDIN-7-YL]BENZYL}PIPERIDIN-4-OL, Proto-oncogene tyrosine-protein kinase Src
著者	Breitenlechner, C.B, Kairies, N.A, Honold, K, Scheiblich, S, Koll, H, Greiter, E, Koch, S, Schaefer, W, Huber, R, Engh, R.A.
登録日	2005-01-27
公開日	2006-01-27
最終更新日	2023-10-25
実験手法	X-RAY DIFFRACTION (2.3 Å)
主引用文献	Crystal structures of active SRC kinase domain complexes J.Mol.Biol., 353, 2005

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BU of 1yom by Molmil

Crystal structure of Src kinase domain in complex with Purvalanol A
分子名称:	2-({6-[(3-CHLOROPHENYL)AMINO]-9-ISOPROPYL-9H-PURIN-2-YL}AMINO)-3-METHYLBUTAN-1-OL, Proto-oncogene tyrosine-protein kinase Src
著者	Breitenlechner, C.B, Kairies, N.A, Honold, K, Scheiblich, S, Koll, H, Greiter, E, Koch, S, Schaefer, W, Huber, R, Engh, R.A.
登録日	2005-01-27
公開日	2006-01-27
最終更新日	2024-05-29
実験手法	X-RAY DIFFRACTION (2.9 Å)
主引用文献	Crystal structures of active SRC kinase domain complexes J.Mol.Biol., 353, 2005

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BU of 3w16 by Molmil

Structure of Aurora kinase A complexed to pyrazole-aminoquinoline inhibitor III
分子名称:	4-[(5-methyl-1H-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2H)-one, Aurora kinase A
著者	Oliveira, T.M, Kairies, N.A, Engh, R.A.
登録日	2012-11-07
公開日	2014-02-05
最終更新日	2024-03-20
実験手法	X-RAY DIFFRACTION (2.8 Å)
主引用文献	Flexibility and multiple conformations of the activation and glycine rich loops of Aurora A accompanying inhibitor binding To be Published

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BU of 3w10 by Molmil

Aurora kinase A complexed to pyrazole aminoquinoline I
分子名称:	1-(3-methoxyphenyl)-N-(5-methyl-1H-pyrazol-3-yl)isoquinolin-3-amine, Aurora kinase A
著者	Oliveira, T.M, Kairies, N.A, Engh, R.A.
登録日	2012-11-06
公開日	2014-02-05
実験手法	X-RAY DIFFRACTION (2.7 Å)
主引用文献	Flexibility and multiple conformations of the activation and glycine rich loops of Aurora A accompanying inhibitor binding To be Published

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BU of 3w18 by Molmil

Structure of Aurora kinase A complexed to benzoimidazole-indazole inhibitor XIII
分子名称:	2-{3-[3-(1H-benzimidazol-2-yl)-1H-indazol-6-yl]-1H-pyrazol-5-yl}-N-(3-fluorophenyl)acetamide, Aurora kinase A
著者	Oliveira, T.M, Kairies, N.A, Engh, R.A.
登録日	2012-11-09
公開日	2014-02-05
最終更新日	2024-03-20
実験手法	X-RAY DIFFRACTION (2.5 Å)
主引用文献	Flexibility and multiple conformations of the activation and glycine rich loops of Aurora A accompanying inhibitor binding To be Published

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BU of 3w2c by Molmil

Structure of Aurora kinase A complexed to benzoimidazole-indazole inhibitor XV
分子名称:	2-{4-[3-(1H-benzimidazol-2-yl)-1H-indazol-6-yl]-1H-pyrazol-1-yl}-N-(3-methylbutyl)acetamide, Aurora kinase A
著者	Oliveira, T.M, Kairies, N.A, Engh, R.A.
登録日	2012-11-28
公開日	2014-02-05
最終更新日	2024-03-20
実験手法	X-RAY DIFFRACTION (2.45 Å)
主引用文献	Flexibility and multiple conformations of the activation and glycine rich loops of aurora A accompanying inhibitor binding To be Published

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件を2024-09-04に公開中

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