7OMD
| Crystal structure of azacoelenterazine-bound Renilla reniformis luciferase variant RLuc8-D162A | 分子名称: | 6-(4-hydroxyphenyl)-2-[(4-hydroxyphenyl)methyl]-8-(phenylmethyl)-[1,2,4]triazolo[4,3-a]pyrazin-3-one, CHLORIDE ION, Coelenterazine h 2-monooxygenase, ... | 著者 | Schenkmayerova, A, Janin, Y.L, Marek, M. | 登録日 | 2021-05-21 | 公開日 | 2022-06-01 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.601 Å) | 主引用文献 | Catalytic mechanism for Renilla-type luciferases Nat Catal, 2023
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7QXR
| Azacoelenterazine-bound Renilla-type luciferase (AncFT) | 分子名称: | 3-(4-hydroxyphenyl)-8-[(4-hydroxyphenyl)methyl]-5-(phenylmethyl)-1$l^{4},4,7,8-tetrazabicyclo[4.3.0]nona-1(6),2,4-trien-9-one, Fragment transplantation onto a hyperstable ancestor of haloalkane dehalogenases and Renilla luciferase (Anc-FT) | 著者 | Marek, M, Schenkmayerova, A, Janin, Y.L. | 登録日 | 2022-01-27 | 公開日 | 2022-12-07 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.052 Å) | 主引用文献 | Catalytic mechanism for Renilla-type luciferases Nat Catal, 2023
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8QQY
| Crystal structure of human Ephrin type-A receptor 2 (EPHA2) Kinase domain in complex with JG165 | 分子名称: | 1,2-ETHANEDIOL, 6-(4-fluoranyl-3-methoxy-phenyl)-13$l^{6}-thia-2,4,8,12,19-pentazatricyclo[12.3.1.1^{3,7}]nonadeca-1(18),3,5,7(19),14,16-hexaene 13,13-dioxide, Ephrin type-A receptor 2 | 著者 | Zhubi, R, Gerninghaus, J, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC) | 登録日 | 2023-10-06 | 公開日 | 2023-11-22 | 最終更新日 | 2024-07-31 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | IPP/CNRS-A017: A chemical probe for human dihydroorotate dehydrogenase (hDHODH) Curr Res Chem Biol, 2, 2022
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8BO9
| NanoLuc-D9R/H57A/K89R mutant complexed with azacoelenterazine bound in intra-barrel catalytic site | 分子名称: | 3-(4-hydroxyphenyl)-8-[(4-hydroxyphenyl)methyl]-5-(phenylmethyl)-1$l^{4},4,7,8-tetrazabicyclo[4.3.0]nona-1(6),2,4-trien-9-one, Non structural polyprotein | 著者 | Marek, M, Janin, L.Y. | 登録日 | 2022-11-15 | 公開日 | 2023-09-27 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Illuminating the mechanism and allosteric behavior of NanoLuc luciferase. Nat Commun, 14, 2023
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7OME
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8AQH
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8AQ6
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8AQI
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7OMO
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7OMR
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7QXQ
| Coelenteramide-bound Renilla-type luciferase (AncFT) | 分子名称: | Fragment transplantation onto hyperstable ancestor of haloalkane dehalogenases and Renilla luciferase (Anc-FT), N-[3-BENZYL-5-(4-HYDROXYPHENYL)PYRAZIN-2-YL]-2-(4-HYDROXYPHENYL)ACETAMIDE | 著者 | Marek, M, Schenkmayerova, A. | 登録日 | 2022-01-27 | 公開日 | 2022-12-07 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.251 Å) | 主引用文献 | Catalytic mechanism for Renilla-type luciferases Nat Catal, 2023
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