1VJY
| Crystal Structure of a Naphthyridine Inhibitor of Human TGF-beta Type I Receptor | 分子名称: | 2-[5-(6-METHYLPYRIDIN-2-YL)-2,3-DIHYDRO-1H-PYRAZOL-4-YL]-1,5-NAPHTHYRIDINE, TGF-beta receptor type I | 著者 | Gellibert, F, Woolven, J, Fouchet, M.-H, Mathews, N, Goodland, H, Lovegrove, V, Laroze, A, Nguyen, V.-L, Sautet, S, Wang, R, Janson, C, Smith, W, Krysa, G, Boullay, V, de Gouville, A.-C, Huet, S, Hartley, D. | 登録日 | 2004-04-07 | 公開日 | 2004-08-31 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Identification of 1,5-Naphthyridine Derivatives as a Novel Series of Potent and Selective TGF-beta Type I Receptor Inhibitors. J.Med.Chem., 47, 2004
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1XLY
| X-RAY STRUCTURE OF THE RNA-BINDING PROTEIN SHE2p | 分子名称: | SHE2p | 著者 | Niessing, D, Huettelmaier, S, Zenklusen, D, Singer, R.H, Burley, S.K. | 登録日 | 2004-09-30 | 公開日 | 2004-11-16 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | She2p is a novel RNA binding protein with a basic helical hairpin motif Cell(Cambridge,Mass.), 119, 2004
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6FY5
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3GXL
| ALK-5 kinase complex with GW857175 | 分子名称: | N-1H-indazol-5-yl-2-(6-methylpyridin-2-yl)quinazolin-4-amine, TGF-beta receptor type-1 | 著者 | Smith, W, Janson, C. | 登録日 | 2009-04-02 | 公開日 | 2009-04-21 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Design of novel quinazoline derivatives and related analogues as potent and selective ALK5 inhibitors Bioorg.Med.Chem.Lett., 19, 2009
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3HMM
| Structure of Alk5 + GW855857 | 分子名称: | 2-(6-methylpyridin-2-yl)-N-pyridin-4-ylquinazolin-4-amine, TGF-beta receptor type-1 | 著者 | Smith, W, Janson, C. | 登録日 | 2009-05-29 | 公開日 | 2009-06-23 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Design of novel quinazoline derivatives and related analogues as potent and selective ALK5 inhibitors Bioorg.Med.Chem.Lett., 19, 2009
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3DY6
| PPARdelta complexed with an anthranilic acid partial agonist | 分子名称: | 2-({[3-(3,4-dihydroisoquinolin-2(1H)-ylsulfonyl)phenyl]carbonyl}amino)benzoic acid, IODIDE ION, Peroxisome proliferator-activated receptor delta | 著者 | Lambert, M.L, Xu, R, Shearer, B.G, Wilson, T.M. | 登録日 | 2008-07-25 | 公開日 | 2008-10-07 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Discovery of a novel class of PPARdelta partial agonists Bioorg.Med.Chem.Lett., 18, 2008
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6G04
| NMR Solution Structure of Yeast TSR2(1-152) in Complex with S26A(100-119) | 分子名称: | 40S ribosomal protein S26-A, Pre-rRNA-processing protein TSR2 | 著者 | Michel, E, Schuetz, S, Damberger, F.F, Allain, F.H.-T, Panse, V.G. | 登録日 | 2018-03-16 | 公開日 | 2018-09-19 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Molecular basis for disassembly of an importin:ribosomal protein complex by the escortin Tsr2. Nat Commun, 9, 2018
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6G03
| NMR Solution Structure of yeast TSR2(1-152) | 分子名称: | Pre-rRNA-processing protein TSR2 | 著者 | Michel, E, Schuetz, S, Damberger, F.F, Allain, F.H.-T, Panse, V.G. | 登録日 | 2018-03-16 | 公開日 | 2018-09-19 | 最終更新日 | 2024-06-19 | 実験手法 | SOLUTION NMR | 主引用文献 | Molecular basis for disassembly of an importin:ribosomal protein complex by the escortin Tsr2. Nat Commun, 9, 2018
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2OB0
| Human MAK3 homolog in complex with Acetyl-CoA | 分子名称: | ACETYL COENZYME *A, Human MAK3 homolog | 著者 | Walker, J.R, Schuetz, S, Antoshenko, T, Wu, H, Bernstein, G, Loppnau, P, Weigelt, J, Sundstrom, M, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Plotnikov, A.N, Structural Genomics Consortium (SGC) | 登録日 | 2006-12-18 | 公開日 | 2006-12-26 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure of Human MAK3 homolog To be Published
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