6UH5
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![BU of 6uh5 by Molmil](/molmil-images/mine/6uh5) | Structural basis of COMPASS eCM recognition of the H2Bub nucleosome | 分子名称: | Bre2, DNA (146-MER), H3 N-terminus, ... | 著者 | Hsu, P.L, Shi, H, Zheng, N. | 登録日 | 2019-09-26 | 公開日 | 2019-11-20 | 最終更新日 | 2019-12-18 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Structural Basis of H2B Ubiquitination-Dependent H3K4 Methylation by COMPASS. Mol.Cell, 76, 2019
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6UGM
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![BU of 6ugm by Molmil](/molmil-images/mine/6ugm) | Structural basis of COMPASS eCM recognition of an unmodified nucleosome | 分子名称: | Bre2, DNA (146-MER), H3 N-terminus, ... | 著者 | Hsu, P.L, Shi, H, Zheng, N. | 登録日 | 2019-09-26 | 公開日 | 2019-11-20 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Structural Basis of H2B Ubiquitination-Dependent H3K4 Methylation by COMPASS. Mol.Cell, 76, 2019
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6CHG
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![BU of 6chg by Molmil](/molmil-images/mine/6chg) | Crystal structure of the yeast COMPASS catalytic module | 分子名称: | H3, Histone-lysine N-methyltransferase, H3 lysine-4 specific, ... | 著者 | Hsu, P.L, Li, H, Zheng, N. | 登録日 | 2018-02-22 | 公開日 | 2018-08-22 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.985 Å) | 主引用文献 | Crystal Structure of the COMPASS H3K4 Methyltransferase Catalytic Module. Cell, 174, 2018
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4M3O
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![BU of 4m3o by Molmil](/molmil-images/mine/4m3o) | Crystal structure of K.lactis Rtr1 NTD | 分子名称: | KLLA0F12672p, ZINC ION | 著者 | Hsu, P.L, Yang, W, Zheng, N, Varani, G. | 登録日 | 2013-08-06 | 公開日 | 2014-07-16 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Rtr1 Is a Dual Specificity Phosphatase That Dephosphorylates Tyr1 and Ser5 on the RNA Polymerase II CTD. J.Mol.Biol., 426, 2014
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8T51
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![BU of 8t51 by Molmil](/molmil-images/mine/8t51) | |
8VW5
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![BU of 8vw5 by Molmil](/molmil-images/mine/8vw5) | Crystal structure of Cbl-b TKB bound to compound 2 | 分子名称: | CALCIUM ION, E3 ubiquitin-protein ligase CBL-B, MAGNESIUM ION, ... | 著者 | Yu, C, Murray, J, Hsu, P.L. | 登録日 | 2024-01-31 | 公開日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | Optimization of a Novel DEL Hit That Binds in the Cbl-b SH2 Domain and Blocks Substrate Binding. Acs Med.Chem.Lett., 15, 2024
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8VW4
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![BU of 8vw4 by Molmil](/molmil-images/mine/8vw4) | Crystal structure of Cbl-b TKB bound to compound 26 | 分子名称: | (7-methoxy-2-{2-[(1S,3S,4S)-3-(3-methoxy-2-methyl-5-nitrophenyl)-1-methyl-5-oxo-1,5-dihydroimidazo[1,5-a]pyridin-2(3H)-yl]-2-oxoethoxy}quinolin-8-yl)acetic acid, DI(HYDROXYETHYL)ETHER, E3 ubiquitin-protein ligase CBL-B, ... | 著者 | Yu, C, Murray, J, Hsu, P.L. | 登録日 | 2024-01-31 | 公開日 | 2024-07-03 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Optimization of a Novel DEL Hit That Binds in the Cbl-b SH2 Domain and Blocks Substrate Binding. Acs Med.Chem.Lett., 15, 2024
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6EEY
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![BU of 6eey by Molmil](/molmil-images/mine/6eey) | |
6B3X
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![BU of 6b3x by Molmil](/molmil-images/mine/6b3x) | Crystal structure of CstF-50 in complex with CstF-77 | 分子名称: | Cleavage stimulation factor subunit 1, Cleavage stimulation factor subunit 3 | 著者 | Yang, W, Hsu, P, Yang, F, Song, J.E, Varani, G. | 登録日 | 2017-09-25 | 公開日 | 2017-11-29 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Reconstitution of the CstF complex unveils a regulatory role for CstF-50 in recognition of 3'-end processing signals. Nucleic Acids Res., 46, 2018
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6OF7
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![BU of 6of7 by Molmil](/molmil-images/mine/6of7) | Crystal structure of the CRY1-PER2 complex | 分子名称: | Cryptochrome-1, Period circadian protein homolog 2 | 著者 | Michael, A.K, Fribourgh, J.L, Tripathi, S.M, Partch, C.L. | 登録日 | 2019-03-28 | 公開日 | 2020-03-04 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (3.11 Å) | 主引用文献 | Dynamics at the serine loop underlie differential affinity of cryptochromes for CLOCK:BMAL1 to control circadian timing. Elife, 9, 2020
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7SZR
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![BU of 7szr by Molmil](/molmil-images/mine/7szr) | NIK bound to inhibitor G02792917 | 分子名称: | 1-(3-{[(1R,4R,5S)-4-hydroxy-2-methyl-3-oxo-2-azabicyclo[3.1.0]hexan-4-yl]ethynyl}phenyl)-1H-pyrazolo[3,4-b]pyridine-3-carboxamide, Mitogen-activated protein kinase kinase kinase 14, SULFATE ION | 著者 | Liau, N.P.D, Hymowitz, S.G. | 登録日 | 2021-11-29 | 公開日 | 2023-06-07 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Filling a nick in NIK: Extending the half-life of a NIK inhibitor through structure-based drug design. Bioorg.Med.Chem.Lett., 89, 2023
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