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3WMG
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BU of 3wmg by Molmil
Crystal structure of an inward-facing eukaryotic ABC multidrug transporter G277V/A278V/A279V mutant in complex with an cyclic peptide inhibitor, aCAP
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ATP-binding cassette, sub-family B, ...
著者Kodan, A, Yamaguchi, T, Nakatsu, T, Sakiyama, K, Hipolito, C.J, Fujioka, A, Hirokane, R, Ikeguchi, K, Watanabe, B, Hirtake, J, Kimura, Y, Suga, H, Ueda, K, Kato, H.
登録日2013-11-18
公開日2014-04-30
最終更新日2017-11-22
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural basis for gating mechanisms of a eukaryotic P-glycoprotein homolog.
Proc.Natl.Acad.Sci.USA, 111, 2014
3VVP
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BU of 3vvp by Molmil
Crystal structure of MATE in complex with Br-NRF
分子名称: 6-bromo-1-ethyl-4-oxo-7-(piperazin-1-yl)-1,4-dihydroquinoline-3-carboxylic acid, Putative uncharacterized protein
著者Tanaka, Y, Ishitani, R, Nureki, O.
登録日2012-07-27
公開日2013-04-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.91 Å)
主引用文献Structural basis for the drug extrusion mechanism by a MATE multidrug transporter.
Nature, 496, 2013
3VVR
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BU of 3vvr by Molmil
Crystal structure of MATE in complex with MaD5
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Putative uncharacterized protein, macrocyclic peptide
著者Tanaka, Y, Ishitani, R, Nureki, O.
登録日2012-07-27
公開日2013-04-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural basis for the drug extrusion mechanism by a MATE multidrug transporter.
Nature, 496, 2013
3VVS
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BU of 3vvs by Molmil
Crystal structure of MATE in complex with MaD3S
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Putative uncharacterized protein, macrocyclic peptide
著者Tanaka, Y, Ishitani, R, Nureki, O.
登録日2012-07-27
公開日2013-04-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural basis for the drug extrusion mechanism by a MATE multidrug transporter.
Nature, 496, 2013
3VVO
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BU of 3vvo by Molmil
Crystal structure of MATE in the bent conformation
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Putative uncharacterized protein
著者Tanaka, Y, Ishitani, R, Nureki, O.
登録日2012-07-27
公開日2013-04-03
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.504 Å)
主引用文献Structural basis for the drug extrusion mechanism by a MATE multidrug transporter.
Nature, 496, 2013
3VVN
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BU of 3vvn by Molmil
Crystal structure of MATE in the straight conformation
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Putative uncharacterized protein
著者Tanaka, Y, Ishitani, R, Nureki, O.
登録日2012-07-27
公開日2013-04-03
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.398 Å)
主引用文献Structural basis for the drug extrusion mechanism by a MATE multidrug transporter.
Nature, 496, 2013
3WBN
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BU of 3wbn by Molmil
Crystal structure of MATE in complex with MaL6
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, MaL6, Putative uncharacterized protein
著者Tanaka, Y, Ishitani, R, Nureki, O.
登録日2013-05-20
公開日2013-06-12
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Structural basis for the drug extrusion mechanism by a MATE multidrug transporter.
Nature, 496, 2013
3WME
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BU of 3wme by Molmil
Crystal structure of an inward-facing eukaryotic ABC multidrug transporter
分子名称: ATP-binding cassette, sub-family B, member 1, ...
著者Kodan, A, Yamaguchi, T, Nakatsu, T, Kato, H.
登録日2013-11-18
公開日2014-03-19
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.751 Å)
主引用文献Structural basis for gating mechanisms of a eukaryotic P-glycoprotein homolog.
Proc.Natl.Acad.Sci.USA, 111, 2014
3W4T
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BU of 3w4t by Molmil
Crystal structure of MATE P26A mutant
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Putative uncharacterized protein
著者Tanaka, Y, Ishitani, R, Nureki, O.
登録日2013-01-16
公開日2013-04-03
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.096 Å)
主引用文献Structural basis for the drug extrusion mechanism by a MATE multidrug transporter.
Nature, 496, 2013
3WMF
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BU of 3wmf by Molmil
Crystal structure of an inward-facing eukaryotic ABC multitrug transporter G277V/A278V/A279V mutant
分子名称: ATP-binding cassette, sub-family B, member 1, ...
著者Kodan, A, Yamaguchi, T, Nakatsu, T, Kato, H.
登録日2013-11-18
公開日2014-03-19
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural basis for gating mechanisms of a eukaryotic P-glycoprotein homolog.
Proc.Natl.Acad.Sci.USA, 111, 2014

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件を2024-09-04に公開中

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