5TIU
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![BU of 5tiu by Molmil](/molmil-images/mine/5tiu) | Crystal structure of SYK kinase domain with inhibitor | 分子名称: | 5-{[(2S)-2-aminopropyl]amino}-3-(1H-indol-2-yl)pyrazine-2-carboxamide, Tyrosine-protein kinase SYK | 著者 | Ellis, J.M, Altman, M.D, Cash, B, Haidle, A.M, Kubiak, R.L, Maddess, M.L, Yan, Y, Northrup, A.B. | 登録日 | 2016-10-03 | 公開日 | 2017-01-11 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.49 Å) | 主引用文献 | Carboxamide Spleen Tyrosine Kinase (Syk) Inhibitors: Leveraging Ground State Interactions To Accelerate Optimization. ACS Med Chem Lett, 7, 2016
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6VLM
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![BU of 6vlm by Molmil](/molmil-images/mine/6vlm) | |
6VLV
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![BU of 6vlv by Molmil](/molmil-images/mine/6vlv) | Factor XIa in complex with compound 11 | 分子名称: | 1-carbamimidamido-4-chloro-N-[(2R)-3-methyl-1-(morpholin-4-yl)-1-oxobutan-2-yl]isoquinoline-7-sulfonamide, CITRATE ANION, Coagulation factor XIa light chain | 著者 | Lesburg, C.A. | 登録日 | 2020-01-27 | 公開日 | 2020-05-06 | 最終更新日 | 2020-10-07 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | Augmenting Hit Identification by Virtual Screening Techniques in Small Molecule Drug Discovery. J.Chem.Inf.Model., 60, 2020
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6VLU
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![BU of 6vlu by Molmil](/molmil-images/mine/6vlu) | Factor XIa in complex with compound 7 | 分子名称: | CITRIC ACID, Coagulation factor XIa light chain, N-cyclohexyl-D-leucyl-N-[(1-aminoisoquinolin-6-yl)methyl]-4,4-difluoro-L-prolinamide | 著者 | Lesburg, C.A, Fradera, X. | 登録日 | 2020-01-27 | 公開日 | 2020-05-06 | 最終更新日 | 2020-10-07 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Augmenting Hit Identification by Virtual Screening Techniques in Small Molecule Drug Discovery. J.Chem.Inf.Model., 60, 2020
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