7T30
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7T2R
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5DIT
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![BU of 5dit by Molmil](/molmil-images/mine/5dit) | The Fk1 domain of FKBP51 in complex with the new synthetic ligand (1R)-3-(3,4-dimethoxyphenyl)-1-f3-[2-(morpholin-4-yl)ethoxy]phenylgpropyl(2S)-1-[(2S,3R)-2-cyclohexyl-3-hydroxybutanoyl]piperidine-2-carboxylate | 分子名称: | (1R)-3-(3,4-dimethoxyphenyl)-1-{3-[2-(morpholin-4-yl)ethoxy]phenyl}propyl (2S)-1-[(2S,3R)-2-cyclohexyl-3-hydroxybutanoyl]piperidine-2-carboxylate, Peptidyl-prolyl cis-trans isomerase FKBP5 | 著者 | Feng, X, Sippel, C, Bracher, A, Hausch, F. | 登録日 | 2015-09-01 | 公開日 | 2015-10-14 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structure-Affinity Relationship Analysis of Selective FKBP51 Ligands. J.Med.Chem., 58, 2015
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6SAF
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![BU of 6saf by Molmil](/molmil-images/mine/6saf) | The Fk1 domain of FKBP51 in complex with (S)-(R)-3-(3,4-dimethoxyphenyl)-1-(3-(2-morpholinoethoxy)phenyl)propyl 1-((1R,4aR,8aR)-4-oxodecahydronaphthalene-1-carbonyl)piperidine-2-carboxylate | 分子名称: | Peptidyl-prolyl cis-trans isomerase FKBP5, [(1~{R})-3-(3,4-dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2~{S})-1-[[(1~{R},4~{a}~{R},8~{a}~{R})-4-oxidanylidene-2,3,4~{a},5,6,7,8,8~{a}-octahydro-1~{H}-naphthalen-1-yl]carbonyl]piperidine-2-carboxylate | 著者 | Feng, X, Sippel, C, Knaup, F, Bracher, A, Staibano, S, Romano, M.F, Hausch, F. | 登録日 | 2019-07-16 | 公開日 | 2019-12-18 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | A Novel Decalin-Based Bicyclic Scaffold for FKBP51-Selective Ligands. J.Med.Chem., 63, 2020
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7MCA
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8DVF
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![BU of 8dvf by Molmil](/molmil-images/mine/8dvf) | T4 Bacteriophage primosome with single strand DNA, state 1 | 分子名称: | DNA (5'-D(P*GP*GP*CP*TP*G)-3'), DNA (5'-D(P*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*T)-3'), DNA primase, ... | 著者 | Feng, X, Li, H. | 登録日 | 2022-07-28 | 公開日 | 2023-06-14 | 最終更新日 | 2023-08-23 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Structural basis of the T4 bacteriophage primosome assembly and primer synthesis. Nat Commun, 14, 2023
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8DVI
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8DTP
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8DW6
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8DUE
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8DUO
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![BU of 8duo by Molmil](/molmil-images/mine/8duo) | DNA-free T4 Bacteriophage gp41 hexamer | 分子名称: | DnaB-like replicative helicase, MAGNESIUM ION, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER | 著者 | Feng, X, Li, H. | 登録日 | 2022-07-27 | 公開日 | 2023-06-14 | 最終更新日 | 2023-08-23 | 実験手法 | ELECTRON MICROSCOPY (5.7 Å) | 主引用文献 | Structural basis of the T4 bacteriophage primosome assembly and primer synthesis. Nat Commun, 14, 2023
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8DWJ
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7KOE
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![BU of 7koe by Molmil](/molmil-images/mine/7koe) | Electron bifurcating flavoprotein Fix/EtfABCX | 分子名称: | Electron transfer flavoprotein, alpha subunit, beta subunit, ... | 著者 | Feng, X, Li, H. | 登録日 | 2020-11-08 | 公開日 | 2021-01-20 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Cryoelectron microscopy structure and mechanism of the membrane-associated electron-bifurcating flavoprotein Fix/EtfABCX. Proc.Natl.Acad.Sci.USA, 118, 2021
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8G0Z
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8GAO
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4ONC
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![BU of 4onc by Molmil](/molmil-images/mine/4onc) | Crystal Structure of Mycobacterium Tuberculosis Decaprenyl Diphosphate Synthase in Complex with BPH-640 | 分子名称: | Decaprenyl diphosphate synthase, [hydroxy(1,1':3',1''-terphenyl-3-yl)methanediyl]bis(phosphonic acid) | 著者 | Feng, X, Chan, H.C, Ko, T.P. | 登録日 | 2014-01-28 | 公開日 | 2014-04-02 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | Structure and Inhibition of Tuberculosinol Synthase and Decaprenyl Diphosphate Synthase from Mycobacterium tuberculosis J.Am.Chem.Soc., 136, 2014
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7X9Q
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![BU of 7x9q by Molmil](/molmil-images/mine/7x9q) | Crystal structure of human STING complexed with compound BSP16 | 分子名称: | (2R)-4-(5,6-dimethoxy-1-benzoselenophen-2-yl)-2-ethyl-4-oxidanylidene-butanoic acid, Stimulator of interferon genes protein | 著者 | Pan, L, Guan, X, Feng, X, Li, Z, Bian, J. | 登録日 | 2022-03-15 | 公開日 | 2022-09-28 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Discovery of Selenium-Containing STING Agonists as Orally Available Antitumor Agents. J.Med.Chem., 65, 2022
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7X9P
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![BU of 7x9p by Molmil](/molmil-images/mine/7x9p) | Crystal structure of human STING complexed with compound BSP17 | 分子名称: | 4-[6-methoxy-5-[3-[[6-methoxy-2-(4-oxidanyl-4-oxidanylidene-butanoyl)-1-benzoselenophen-5-yl]oxy]propoxy]-1-benzoselenophen-2-yl]-4-oxidanylidene-butanoic acid, Stimulator of interferon genes protein | 著者 | Pan, L, Guan, X, Feng, X, Li, Z, Bian, J. | 登録日 | 2022-03-15 | 公開日 | 2023-03-22 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Discovery of Selenium-containing STING agonists as orally available anti tumor agents To be published
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5DIV
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![BU of 5div by Molmil](/molmil-images/mine/5div) | The Fk1 domain of FKBP51 in complex with the new synthetic ligand (S)-N-(1-carbamoylcyclopentyl)-1-((S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl)piperidine-2-carboxamide | 分子名称: | (2S)-N-(1-carbamoylcyclopentyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide, Peptidyl-prolyl cis-trans isomerase FKBP5 | 著者 | Gaali, S, Feng, X, Sippel, C, Bracher, A, Hausch, F. | 登録日 | 2015-09-01 | 公開日 | 2016-03-23 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Rapid, Structure-Based Exploration of Pipecolic Acid Amides as Novel Selective Antagonists of the FK506-Binding Protein 51. J.Med.Chem., 59, 2016
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4Z2Z
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3W01
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![BU of 3w01 by Molmil](/molmil-images/mine/3w01) | Crystal structure of PcrB complexed with PEG from Staphylococcus aureus subsp. aureus Mu3 | 分子名称: | Heptaprenylglyceryl phosphate synthase, TRIETHYLENE GLYCOL | 著者 | Ren, F, Feng, X, Ko, T.P, Huang, C.H, Hu, Y, Chan, H.C, Liu, Y.L, Wang, K, Chen, C.C, Pang, X, He, M, Li, Y, Oldfield, E, Guo, R.T. | 登録日 | 2012-10-17 | 公開日 | 2012-12-26 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | Insights into TIM-barrel prenyl transferase mechanisms: crystal structures of PcrB from Bacillus subtilis and Staphylococcus aureus Chembiochem, 14, 2013
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3VZZ
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![BU of 3vzz by Molmil](/molmil-images/mine/3vzz) | Crystal structure of PcrB complexed with FsPP from bacillus subtilis subap. subtilis str. 168 | 分子名称: | CHLORIDE ION, Heptaprenylglyceryl phosphate synthase, MAGNESIUM ION, ... | 著者 | Ren, F, Feng, X, Ko, T.P, Huang, C.H, Hu, Y, Chan, H.C, Liu, Y.L, Wang, K, Chen, C.C, Pang, X, He, M, Li, Y, Oldfield, E, Guo, R.T. | 登録日 | 2012-10-17 | 公開日 | 2012-12-26 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.04 Å) | 主引用文献 | Insights into TIM-barrel prenyl transferase mechanisms: crystal structures of PcrB from Bacillus subtilis and Staphylococcus aureus Chembiochem, 14, 2013
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3VZX
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![BU of 3vzx by Molmil](/molmil-images/mine/3vzx) | Crystal structure of PcrB from bacillus subtilis subap. subtilis str. 168 | 分子名称: | CHLORIDE ION, Heptaprenylglyceryl phosphate synthase, MAGNESIUM ION | 著者 | Ren, F, Feng, X, Ko, T.P, Huang, C.H, Hu, Y, Chan, H.C, Liu, Y.L, Wang, K, Chen, C.C, Pang, X, He, M, Li, Y, Oldfield, E, Guo, R.T. | 登録日 | 2012-10-17 | 公開日 | 2012-12-26 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | Insights into TIM-barrel prenyl transferase mechanisms: crystal structures of PcrB from Bacillus subtilis and Staphylococcus aureus Chembiochem, 14, 2013
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3VZY
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![BU of 3vzy by Molmil](/molmil-images/mine/3vzy) | Crystal structure of PcrB complexed with G1P from bacillus subtilis subap. subtilis str. 168 | 分子名称: | CHLORIDE ION, Heptaprenylglyceryl phosphate synthase, MAGNESIUM ION, ... | 著者 | Ren, F, Feng, X, Ko, T.P, Huang, C.H, Hu, Y, Chan, H.C, Liu, Y.L, Wang, K, Chen, C.C, Pang, X, He, M, Li, Y, Oldfield, E, Guo, R.T. | 登録日 | 2012-10-17 | 公開日 | 2012-12-26 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | Insights into TIM-barrel prenyl transferase mechanisms: crystal structures of PcrB from Bacillus subtilis and Staphylococcus aureus Chembiochem, 14, 2013
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3W02
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![BU of 3w02 by Molmil](/molmil-images/mine/3w02) | Crystal structure of PcrB complexed with SO4 from Staphylococcus aureus subsp. aureus Mu3 | 分子名称: | Heptaprenylglyceryl phosphate synthase, SULFATE ION | 著者 | Ren, F, Feng, X, Ko, T.P, Huang, C.H, Hu, Y, Chan, H.C, Liu, Y.L, Wang, K, Chen, C.C, Pang, X, He, M, Li, Y, Oldfield, E, Guo, R.T. | 登録日 | 2012-10-17 | 公開日 | 2012-12-26 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.98 Å) | 主引用文献 | Insights into TIM-barrel prenyl transferase mechanisms: crystal structures of PcrB from Bacillus subtilis and Staphylococcus aureus Chembiochem, 14, 2013
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