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4RO0
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BU of 4ro0 by Molmil
Crystal structure of MthK gating ring in a ligand-free form
分子名称: Calcium-gated potassium channel MthK
著者Dong, W, Guo, R, Chai, H, Chen, Z, Cui, H, Ren, Z, Li, Y, Ye, S.
登録日2014-10-27
公開日2015-10-28
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.18 Å)
主引用文献The principle of cooperative gating in a calcium-gated K+ channel
To be Published
1N1L
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BU of 1n1l by Molmil
CRYSTAL STRUCTURE OF HCV NS3 PROTEASE DOMAIN:NS4A PEPTIDE COMPLEX WITH COVALENTLY BOUND INHIBITOR (GW472467X)
分子名称: HCV NS3 SERINE PROTEASE, NS4A COFACTOR, ZINC ION, ...
著者Andrews, D.M, Chaignot, H, Coomber, B.A, Good, A.C, Hind, S.L, Jones, P.S, Mill, G, Robinson, J.E, Skarzynski, T, Slater, M.J, Somers, D.O.N.
登録日2002-10-18
公開日2003-10-21
最終更新日2021-10-27
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Pyrrolidine-5,5-trans-lactams. 2. The use of X-ray Crystal Structure Data in the Optimisation of P3 and P4 Substituents
Org.Lett., 4, 2002
1RTL
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CRYSTAL STRUCTURE OF HCV NS3 PROTEASE DOMAIN: NS4A PEPTIDE COMPLEX WITH COVALENTLY BOUND PYRROLIDINE-5,5-TRANSLACTAM INHIBITOR
分子名称: N-[(2R,3S)-1-((2S)-2-{[(CYCLOPENTYLAMINO)CARBONYL]AMINO}-3-METHYLBUTANOYL)-2-(1-FORMYL-1-CYCLOBUTYL)PYRROLIDINYL]CYCLOPROPANECARBOXAMIDE, NS3 protease/helicase, NS4A COFACTOR, ...
著者Skarzynski, T, Somers, D.O.N.
登録日2003-12-10
公開日2004-12-14
最終更新日2021-10-27
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Pyrrolidine-5,5-trans-lactams. 4. Incorporation of a P3/P4 urea leads to potent intracellular inhibitors of hepatitis C virus NS3/4A protease
Org.Lett., 5, 2003

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件を2024-09-04に公開中

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