6MTU
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![BU of 6mtu by Molmil](/molmil-images/mine/6mtu) | Crystal structure of human Scribble PDZ1:pMCC complex | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, Colorectal mutant cancer protein, ... | 著者 | Caria, S, Stewart, B.Z, Humbert, P.O, Kvansakul, M. | 登録日 | 2018-10-22 | 公開日 | 2019-08-14 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.141 Å) | 主引用文献 | Structural analysis of phosphorylation-associated interactions of human MCC with Scribble PDZ domains. Febs J., 286, 2019
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6MTV
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![BU of 6mtv by Molmil](/molmil-images/mine/6mtv) | Crystal structure of human Scribble PDZ1:MCC complex | 分子名称: | Colorectal mutant cancer protein, DI(HYDROXYETHYL)ETHER, Protein scribble homolog, ... | 著者 | Caria, S, Stewart, B.Z, Humbert, P.O, Kvansakul, M. | 登録日 | 2018-10-22 | 公開日 | 2019-08-14 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.597 Å) | 主引用文献 | Structural analysis of phosphorylation-associated interactions of human MCC with Scribble PDZ domains. Febs J., 286, 2019
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5TWA
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![BU of 5twa by Molmil](/molmil-images/mine/5twa) | Crystal structure of Geodia cydonium BHP2 in complex with Lubomirskia baicalensis Bak-2 | 分子名称: | 1,2-ETHANEDIOL, 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, BAK-2 protein, ... | 著者 | Caria, S, Hinds, M.G, Kvansakul, M. | 登録日 | 2016-11-12 | 公開日 | 2017-01-25 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Structural insight into an evolutionarily ancient programmed cell death regulator - the crystal structure of marine sponge BHP2 bound to LB-Bak-2. Cell Death Dis, 8, 2017
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5WOU
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![BU of 5wou by Molmil](/molmil-images/mine/5wou) | |
7ZDD
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![BU of 7zdd by Molmil](/molmil-images/mine/7zdd) | Crystal structure of TRIM33 PHD-Bromodomain isoform B in complex with H3K10ac histone peptide. | 分子名称: | 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM33, Histone H3.X, ... | 著者 | Caria, S, Duclos, S, Crespillo, S, Errey, J, Barker, J.J. | 登録日 | 2022-03-29 | 公開日 | 2022-06-29 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.625 Å) | 主引用文献 | Identification of Histone Peptide Binding Specificity and Small-Molecule Ligands for the TRIM33 alpha and TRIM33 beta Bromodomains. Acs Chem.Biol., 17, 2022
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6MRY
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![BU of 6mry by Molmil](/molmil-images/mine/6mry) | NoD173 plant defensin | 分子名称: | 1,2-ETHANEDIOL, 5-amino-2,4,6-triiodobenzene-1,3-dicarboxylic acid, CHLORIDE ION, ... | 著者 | Caria, S, Kvansakul, M. | 登録日 | 2018-10-15 | 公開日 | 2019-04-24 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural and functional characterization of the membrane-permeabilizing activity ofNicotiana occidentalisdefensin NoD173 and protein engineering to enhance oncolysis. Faseb J., 33, 2019
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2VF7
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![BU of 2vf7 by Molmil](/molmil-images/mine/2vf7) | Crystal structure of UvrA2 from Deinococcus radiodurans | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, EXCINUCLEASE ABC, SUBUNIT A., ... | 著者 | Timmins, J, Gordon, E, Caria, S, Leonard, G, Kuo, M.S, Monchois, V, McSweeney, S. | 登録日 | 2007-10-31 | 公開日 | 2008-12-16 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural and mutational analyses of Deinococcus radiodurans UvrA2 provide insight into DNA binding and damage recognition by UvrAs. Structure, 17, 2009
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2VF8
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![BU of 2vf8 by Molmil](/molmil-images/mine/2vf8) | Crystal structure of UvrA2 from Deinococcus radiodurans | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, EXCINUCLEASE ABC SUBUNIT A, PHOSPHATE ION, ... | 著者 | Timmins, J, Gordon, E, Caria, S, Leonard, G, Kuo, M.S, Monchois, V, McSweeney, S. | 登録日 | 2007-10-31 | 公開日 | 2008-12-16 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural and Mutational Analyses of Deinococcus Radiodurans Uvra2 Provide Insight Into DNA Binding and Damage Recognition by Uvras. Structure, 17, 2009
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7S1L
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![BU of 7s1l by Molmil](/molmil-images/mine/7s1l) | Crystal structure of E.coli DsbA in complex with compound MIPS-0001896 (compound 72) | 分子名称: | COPPER (II) ION, Thiol:disulfide interchange protein DsbA, methyl cis-4-({[3-(thiophen-3-yl)benzyl]amino}methyl)cyclohexanecarboxylate | 著者 | Heras, B, Scanlon, M.J, Martin, J.L, Caria, S. | 登録日 | 2021-09-02 | 公開日 | 2023-02-08 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.623 Å) | 主引用文献 | Fluoromethylketone-fragment conjugates designed as covalent modifiers of EcDsbA are atypical substrates Chemrxiv, 2022
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7S1D
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![BU of 7s1d by Molmil](/molmil-images/mine/7s1d) | Crystal structure of E.coli DsbA in complex with compound MIPS-0001877 (compound 39) | 分子名称: | 1-[3-(thiophen-3-yl)benzyl]piperidin-2-one, COPPER (II) ION, Thiol:disulfide interchange protein DsbA | 著者 | Heras, B, Scanlon, M.J, Martin, J.L, Caria, S. | 登録日 | 2021-09-02 | 公開日 | 2023-02-08 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.59 Å) | 主引用文献 | Fluoromethylketone-fragment conjugates designed as covalent modifiers of EcDsbA are atypical substrates Chemrxiv, 2022
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7S1F
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![BU of 7s1f by Molmil](/molmil-images/mine/7s1f) | Crystal structure of E.coli DsbA in complex with compound MIPS-0001886 (compound 38) | 分子名称: | 1-[(3-thiophen-3-ylphenyl)methyl]-3~{H}-pyrrol-2-one, COPPER (II) ION, GLYCEROL, ... | 著者 | Heras, B, Scanlon, M.J, Martin, J.L, Caria, S. | 登録日 | 2021-09-02 | 公開日 | 2023-02-08 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | Fluoromethylketone-fragment conjugates designed as covalent modifiers of EcDsbA are atypical substrates Chemrxiv, 2022
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4WF5
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![BU of 4wf5 by Molmil](/molmil-images/mine/4wf5) | Crystal structure of E.Coli DsbA soaked with compound 4 | 分子名称: | 1,2-ETHANEDIOL, 4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-5-carboxylic acid, COPPER (II) ION, ... | 著者 | Adams, L.A, Sharma, P, Mohanty, B, Ilyichova, O.V, Mulcair, M.D, Williams, M.L, Gleeson, E.C, Totsika, M, Doak, B.C, Caria, S, Rimmer, K, Shouldice, S.R, Vazirani, M, Headey, S.J, Plumb, B.R, Martin, J.L, Heras, B, Simpson, J.S, Scanlon, M.J. | 登録日 | 2014-09-12 | 公開日 | 2015-01-21 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Application of Fragment-Based Screening to the Design of Inhibitors of Escherichia coli DsbA. Angew.Chem.Int.Ed.Engl., 54, 2015
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4WEY
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![BU of 4wey by Molmil](/molmil-images/mine/4wey) | Crystal structure of E.Coli DsbA in complex with compound 17 | 分子名称: | 1,2-ETHANEDIOL, N-({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}carbonyl)-L-serine, Thiol:disulfide interchange protein | 著者 | Adams, L.A, Sharma, P, Mohanty, B, Ilyichova, O.V, Mulcair, M.D, Williams, M.L, Gleeson, E.C, Totsika, M, Doak, B.C, Caria, S, Rimmer, K, Shouldice, S.R, Vazirani, M, Headey, S.J, Plumb, B.R, Martin, J.L, Heras, B, Simpson, J.S, Scanlon, M.J. | 登録日 | 2014-09-11 | 公開日 | 2015-01-21 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Application of Fragment-Based Screening to the Design of Inhibitors of Escherichia coli DsbA. Angew.Chem.Int.Ed.Engl., 54, 2015
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4WF4
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![BU of 4wf4 by Molmil](/molmil-images/mine/4wf4) | Crystal structure of E.Coli DsbA co-crystallised in complex with compound 4 | 分子名称: | 1,2-ETHANEDIOL, 4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-5-carboxylic acid, Thiol:disulfide interchange protein | 著者 | Adams, L.A, Sharma, P, Mohanty, B, Ilyichova, O.V, Mulcair, M.D, Williams, M.L, Gleeson, E.C, Totsika, M, Doak, B.C, Caria, S, Rimmer, K, Shouldice, S.R, Vazirani, M, Headey, S.J, Plumb, B.R, Martin, J.L, Heras, B, Simpson, J.S, Scanlon, M.J. | 登録日 | 2014-09-12 | 公開日 | 2015-01-21 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Application of Fragment-Based Screening to the Design of Inhibitors of Escherichia coli DsbA. Angew.Chem.Int.Ed.Engl., 54, 2015
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6MS1
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![BU of 6ms1 by Molmil](/molmil-images/mine/6ms1) | Crystal structure of the human Scribble PDZ1 domain bound to the PDZ-binding motif of APC | 分子名称: | 1,2-ETHANEDIOL, APC C-terminus peptide, Protein scribble homolog | 著者 | How, J.Y, Kvansakul, M, Caria, S, Humbert, P.O. | 登録日 | 2018-10-16 | 公開日 | 2019-02-06 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Crystal structure of the human Scribble PDZ1 domain bound to the PDZ-binding motif of APC. FEBS Lett., 593, 2019
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5UA4
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![BU of 5ua4 by Molmil](/molmil-images/mine/5ua4) | |
5UA5
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![BU of 5ua5 by Molmil](/molmil-images/mine/5ua5) | |
6FBX
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![BU of 6fbx by Molmil](/molmil-images/mine/6fbx) | |
7S1C
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![BU of 7s1c by Molmil](/molmil-images/mine/7s1c) | Crystal structure of E.coli DsbA in complex with compound MIPS-0001897 (compound 1) | 分子名称: | COPPER (II) ION, Thiol:disulfide interchange protein DsbA, ~{N}-methyl-1-(3-thiophen-3-ylphenyl)methanamine | 著者 | Heras, B, Scanlon, M.J, Martin, J.L, Sharma, P. | 登録日 | 2021-09-02 | 公開日 | 2023-02-08 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.949 Å) | 主引用文献 | Fluoromethylketone-fragment conjugates designed as covalent modifiers of EcDsbA are atypical substrates Chemrxiv, 2022
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6H1N
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![BU of 6h1n by Molmil](/molmil-images/mine/6h1n) | |
8B82
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![BU of 8b82 by Molmil](/molmil-images/mine/8b82) | |
8B87
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![BU of 8b87 by Molmil](/molmil-images/mine/8b87) | |
8B8O
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![BU of 8b8o by Molmil](/molmil-images/mine/8b8o) | |
8B9T
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![BU of 8b9t by Molmil](/molmil-images/mine/8b9t) | |
8BJ0
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![BU of 8bj0 by Molmil](/molmil-images/mine/8bj0) | |