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5WIV
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BU of 5wiv by Molmil
Structure of the sodium-bound human D4 Dopamine receptor in complex with Nemonapride
分子名称: D(4) dopamine receptor, soluble cytochrome b562 chimera, DI(HYDROXYETHYL)ETHER, ...
著者Wacker, D, Wang, S, Levit, A, Che, T, Betz, R.M, McCorvy, J.D, Venkatakrishnan, A.J, Huang, X.-P, Dror, R.O, Shoichet, B.K, Roth, B.L.
登録日2017-07-20
公開日2017-10-18
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.143 Å)
主引用文献D4 dopamine receptor high-resolution structures enable the discovery of selective agonists.
Science, 358, 2017
5WIU
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BU of 5wiu by Molmil
Structure of the human D4 Dopamine receptor in complex with Nemonapride
分子名称: D(4) dopamine receptor, soluble cytochrome b562 chimera, DI(HYDROXYETHYL)ETHER, ...
著者Wacker, D, Wang, S, Levit, A, Che, T, Betz, R.M, McCorvy, J.D, Venkatakrishnan, A.J, Huang, X.-P, Dror, R.O, Shoichet, B.K, Roth, B.L.
登録日2017-07-20
公開日2017-10-18
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.962 Å)
主引用文献D4 dopamine receptor high-resolution structures enable the discovery of selective agonists.
Science, 358, 2017
5TVN
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BU of 5tvn by Molmil
Crystal structure of the LSD-bound 5-HT2B receptor
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, (8alpha)-N,N-diethyl-6-methyl-9,10-didehydroergoline-8-carboxamide, CHOLESTEROL, ...
著者Wacker, D, Wang, S, McCorvy, J.D, Betz, R.M, Venkatakrishnan, A.J, Levit, A, Lansu, K, Schools, Z.L, Che, T, Nichols, D.E, Shoichet, B.K, Dror, R.O, Roth, B.L.
登録日2016-11-09
公開日2017-02-01
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal Structure of an LSD-Bound Human Serotonin Receptor.
Cell, 168, 2017
6DK0
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BU of 6dk0 by Molmil
Human sigma-1 receptor bound to NE-100
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, GLYCEROL, N-{2-[4-methoxy-3-(2-phenylethoxy)phenyl]ethyl}-N-propylpropan-1-amine, ...
著者Schmidt, H.R, Kruse, A.C.
登録日2018-05-28
公開日2018-10-17
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural basis for sigma1receptor ligand recognition.
Nat. Struct. Mol. Biol., 25, 2018
6DJZ
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BU of 6djz by Molmil
Human sigma-1 receptor bound to haloperidol
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 4-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-1-(4-fluorophenyl)butan-1-one, GLYCEROL, ...
著者Schmidt, H.R, Kruse, A.C.
登録日2018-05-28
公開日2018-10-17
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.084 Å)
主引用文献Structural basis for sigma1receptor ligand recognition.
Nat. Struct. Mol. Biol., 25, 2018
6DK1
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BU of 6dk1 by Molmil
Human sigma-1 receptor bound to (+)-pentazocine
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, (2S,6S,11S)-6,11-dimethyl-3-(3-methylbut-2-en-1-yl)-1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocin-8-ol, GLYCEROL, ...
著者Schmidt, H.R, Kruse, A.C.
登録日2018-05-28
公開日2018-10-17
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.12 Å)
主引用文献Structural basis for sigma1receptor ligand recognition.
Nat. Struct. Mol. Biol., 25, 2018

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件を2024-07-17に公開中

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