6GJV
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6GK9
| Inhibited structure of IMPDH from Pseudomonas aeruginosa | 分子名称: | (5~{S})-7-azanyl-5-(4-chlorophenyl)-2,4-bis(oxidanylidene)-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile, Inosine-5'-monophosphate dehydrogenase, SULFATE ION | 著者 | Labesse, G, Alexandre, T, Haouz, A, Munier-Lehmann, H. | 登録日 | 2018-05-18 | 公開日 | 2019-02-27 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.54 Å) | 主引用文献 | First-in-class allosteric inhibitors of bacterial IMPDHs. Eur J Med Chem, 167, 2019
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5AHL
| Apo-form of the DeltaCBS mutant of IMPDH from Pseudomonas aeruginosa | 分子名称: | INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE, SODIUM ION | 著者 | Labesse, G, Alexandre, T, Gelin, M, Haouz, A, Munier-Lehmann, H. | 登録日 | 2015-02-06 | 公開日 | 2015-07-15 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.951 Å) | 主引用文献 | Crystallographic Studies of Two Variants of Pseudomonas Aeruginosa Impdh with Impaired Allosteric Regulation Acta Crystallogr.,Sect.D, 71, 2015
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5AHM
| IMP-bound form of the DeltaCBS mutant of IMPDH from Pseudomonas aeruginosa | 分子名称: | INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE, INOSINIC ACID, PHOSPHATE ION | 著者 | Labesse, G, Alexandre, T, Gelin, M, Haouz, A, Munier-Lehmann, H. | 登録日 | 2015-02-06 | 公開日 | 2015-07-15 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Crystallographic Studies of Two Variants of Pseudomonas Aeruginosa Impdh with Impaired Allosteric Regulation Acta Crystallogr.,Sect.D, 71, 2015
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5AHN
| IMP-bound form of the D199N mutant of IMPDH from Pseudomonas aeruginosa | 分子名称: | INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE, INOSINIC ACID, MAGNESIUM ION | 著者 | Labesse, G, Alexandre, T, Gelin, M, Haouz, A, Munier-Lehmann, H. | 登録日 | 2015-02-06 | 公開日 | 2015-07-15 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.652 Å) | 主引用文献 | Crystallographic Studies of Two Variants of Pseudomonas Aeruginosa Impdh with Impaired Allosteric Regulation Acta Crystallogr.,Sect.D, 71, 2015
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4DQW
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7QEM
| bacterial IMPDH chimera | 分子名称: | INOSINIC ACID, Inosine-5'-monophosphate dehydrogenase | 著者 | Labesse, G, Gelin, M, Gedeon, A, Haouz, A, Munier-Lehmann, H. | 登録日 | 2021-12-03 | 公開日 | 2023-06-14 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (3.09 Å) | 主引用文献 | Insight into the role of the Bateman domain at the molecular and physiological levels through engineered IMP dehydrogenases. Protein Sci., 32, 2023
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