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6M0T
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BU of 6m0t by Molmil
Crystal Structure of Lysyl-tRNA Synthetase from Plasmodium falciparum complexed with L-lysine and Cladosporin derivative (CL-2)
分子名称: (3R)-3-[(R)-[(2R,6S)-6-methyloxan-2-yl]-oxidanyl-methyl]-6,8-bis(oxidanyl)-3,4-dihydroisochromen-1-one, LYSINE, Lysine--tRNA ligase
著者Babbar, P, Sharma, A, Manickam, Y.
登録日2020-02-22
公開日2021-04-21
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.68 Å)
主引用文献Design, Synthesis, and Structural Analysis of Cladosporin-Based Inhibitors of Malaria Parasites.
Acs Infect Dis., 7, 2021
5YB2
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BU of 5yb2 by Molmil
Crystal structure of LP-11/N44
分子名称: Envelope glycoprotein, LP-11
著者Zhang, X, Wang, X, He, Y.
登録日2017-09-03
公開日2018-02-28
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Structural Insights into the Mechanisms of Action of Short-Peptide HIV-1 Fusion Inhibitors Targeting the Gp41 Pocket
Front Cell Infect Microbiol, 8, 2018
4WTD
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BU of 4wtd by Molmil
CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS AND DELTA8 BETA HAIRPIN LOOP DELETION IN COMPLEX WITH ADP, MN2+ AND SYMMETRICAL PRIMER TEMPLATE 5'-AUAAAUUU
分子名称: ADENOSINE-5'-DIPHOSPHATE, CHLORIDE ION, MANGANESE (II) ION, ...
著者Edwards, T.E, Fox III, D, Appleby, T.C.
登録日2014-10-29
公開日2015-02-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural basis for RNA replication by the hepatitis C virus polymerase.
Science, 347, 2015
4WTF
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BU of 4wtf by Molmil
CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS AND DELTA8 BETA HAIRPIN LOOP DELETION IN COMPLEX WITH GS-639475, MN2+ AND SYMMETRICAL PRIMER TEMPLATE 5'-CAAAAUUU
分子名称: 2'-C-methyluridine 5'-(trihydrogen diphosphate), CHLORIDE ION, MANGANESE (II) ION, ...
著者Edwards, T.E, Appleby, T.C, Mcgrath, M.E.
登録日2014-10-30
公開日2015-02-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Structural basis for RNA replication by the hepatitis C virus polymerase.
Science, 347, 2015
4WTJ
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BU of 4wtj by Molmil
CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS IN COMPLEX WITH RNA TEMPLATE 5'-AUCC, RNA PRIMER 5'-PGG, MN2+, AND ADP
分子名称: 1,2-ETHANEDIOL, 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ...
著者Edwards, T.E, Appleby, T.C.
登録日2014-10-30
公開日2015-02-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural basis for RNA replication by the hepatitis C virus polymerase.
Science, 347, 2015
4WTM
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BU of 4wtm by Molmil
CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS IN COMPLEX WITH RNA TEMPLATE 5'-UAGG, RNA PRIMER 5'-PCC, MN2+, AND UDP
分子名称: CHLORIDE ION, MANGANESE (II) ION, RNA PRIMER CC, ...
著者Edwards, T.E, Appleby, T.C, Fox III, D.
登録日2014-10-30
公開日2015-02-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structural basis for RNA replication by the hepatitis C virus polymerase.
Science, 347, 2015
7SBM
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BU of 7sbm by Molmil
Human glutaminase C (Y466W) with L-Gln, open conformation
分子名称: GLUTAMINE, Isoform 3 of Glutaminase kidney isoform, mitochondrial
著者Nguyen, T.-T.T, Cerione, R.A.
登録日2021-09-25
公開日2022-02-02
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献High-resolution structures of mitochondrial glutaminase C tetramers indicate conformational changes upon phosphate binding.
J.Biol.Chem., 298, 2022
4YG7
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BU of 4yg7 by Molmil
Structure of FL autorepression promoter complex
分子名称: Antitoxin HipB, DNA (50-MER), Serine/threonine-protein kinase HipA
著者Schumacher, M.A.
登録日2015-02-25
公開日2015-07-29
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.77 Å)
主引用文献HipBA-promoter structures reveal the basis of heritable multidrug tolerance.
Nature, 524, 2015
5YB4
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BU of 5yb4 by Molmil
Crystal structure of HP23LN36KR
分子名称: HP23L, N36KR
著者Zhang, X, Wang, X, He, Y.
登録日2017-09-03
公開日2018-02-28
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural Insights into the Mechanisms of Action of Short-Peptide HIV-1 Fusion Inhibitors Targeting the Gp41 Pocket
Front Cell Infect Microbiol, 8, 2018
8W8D
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BU of 8w8d by Molmil
Structural mechanism of inhibition of the Rho transcription termination factor by Rof
分子名称: Protein rof, Transcription termination factor Rho
著者Zhang, J, Wang, C.
登録日2023-09-01
公開日2024-05-01
実験手法ELECTRON MICROSCOPY (2.8 Å)
主引用文献A widely conserved protein Rof inhibits transcription termination factor Rho and promotes Salmonella virulence program.
Nat Commun, 15, 2024
5V5W
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BU of 5v5w by Molmil
Molecular Mechanism of MDGA1: Regulation of Neuroligin 2:Neurexin Trans-synaptic Bridges
分子名称: MAM domain-containing glycosylphosphatidylinositol anchor protein 1, SULFATE ION
著者Machius, M, Gangwar, S.P, Rudenko, G.
登録日2017-03-15
公開日2017-07-05
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.718 Å)
主引用文献Molecular Mechanism of MDGA1: Regulation of Neuroligin 2:Neurexin Trans-synaptic Bridges.
Neuron, 94, 2017
5V5V
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BU of 5v5v by Molmil
Complex of NLGN2 with MDGA1 Ig1-Ig2
分子名称: MAM domain-containing glycosylphosphatidylinositol anchor protein 1, Neuroligin-2
著者Gangwar, S.P, Machius, M, Rudenko, G.
登録日2017-03-15
公開日2017-07-05
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (4.11 Å)
主引用文献Molecular Mechanism of MDGA1: Regulation of Neuroligin 2:Neurexin Trans-synaptic Bridges.
Neuron, 94, 2017
4YG4
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BU of 4yg4 by Molmil
HipB-O1-O1* complex
分子名称: Antitoxin HipB, DNA (28-MER), DNA (5'-D(*AP*TP*AP*TP*CP*CP*CP*CP*TP*TP*AP*AP*GP*GP*GP*GP*AP*TP*AP*A)-3')
著者Schumacher, M.A.
登録日2015-02-25
公開日2015-07-29
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献HipBA-promoter structures reveal the basis of heritable multidrug tolerance.
Nature, 524, 2015
6N3I
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BU of 6n3i by Molmil
Crystal structure of a double Trp XylE mutants (G58W/L315W)
分子名称: D-xylose transporter
著者Jiang, X, Wu, J.P, Yan, N.
登録日2018-11-15
公開日2019-03-27
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.69 Å)
主引用文献Engineered XylE as a tool for mechanistic investigation and ligand discovery of the glucose transporters GLUTs.
Cell Discov, 5, 2019
4YFB
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BU of 4yfb by Molmil
Structure of N-acylhomoserine lactone acylase MacQ in complex with phenylacetic acid
分子名称: 2-PHENYLACETIC ACID, GLYCEROL, Protein related to penicillin acylase
著者Yasutake, Y, Kusada, H, Kimura, N.
登録日2015-02-25
公開日2016-03-02
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Bifunctional quorum-quenching and antibiotic-acylase MacQ forms a 170-kDa capsule-shaped molecule containing spacer polypeptides
Sci Rep, 7, 2017
2K9E
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BU of 2k9e by Molmil
NMR Solution Structure for ShK-192: A Potent KV1.3-Specific Immunosuppressive Polypeptide
分子名称: Kappa-stichotoxin-She3a
著者Galea, C.A.
登録日2008-10-09
公開日2009-01-20
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Engineering a stable and selective peptide blocker of the Kv1.3 channel in T lymphocytes
Mol.Pharmacol., 75, 2009
5VDR
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BU of 5vdr by Molmil
Human cyclic GMP-AMP synthase (cGAS) in complex with 3',3'-cdIMP
分子名称: 3',3'-cdIMP, Cyclic GMP-AMP synthase, ZINC ION
著者Byrnes, L.J, Hall, J.D.
登録日2017-04-03
公開日2017-09-27
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.042 Å)
主引用文献The catalytic mechanism of cyclic GMP-AMP synthase (cGAS) and implications for innate immunity and inhibition.
Protein Sci., 26, 2017
5VDP
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BU of 5vdp by Molmil
Human cyclic GMP-AMP synthase (cGAS) in complex with 2',3'-cGAMP
分子名称: Cyclic GMP-AMP synthase, SULFATE ION, ZINC ION, ...
著者Byrnes, L.J, Hall, J.D.
登録日2017-04-03
公開日2017-09-27
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The catalytic mechanism of cyclic GMP-AMP synthase (cGAS) and implications for innate immunity and inhibition.
Protein Sci., 26, 2017
4WT9
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BU of 4wt9 by Molmil
APO CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH E86Q E87Q S15G C223H V321I AND DELTA8 MUTATIONS
分子名称: 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CHLORIDE ION, ...
著者Edwards, T.E, Appleby, T.C.
登録日2014-10-29
公開日2015-02-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural basis for RNA replication by the hepatitis C virus polymerase.
Science, 347, 2015
4WTA
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BU of 4wta by Molmil
CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS AND DELTA8 BETA HAIRPIN LOOP DELETION IN COMPLEX WITH UDP, MN2+ AND SYMMETRICAL PRIMER TEMPLATE 5'-CAAAAUUU
分子名称: CHLORIDE ION, MANGANESE (II) ION, RNA PRIMER TEMPLATE CAAAAUUU, ...
著者Edwards, T.E, Appleby, T.C.
登録日2014-10-29
公開日2015-02-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structural basis for RNA replication by the hepatitis C virus polymerase.
Science, 347, 2015
4WTC
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BU of 4wtc by Molmil
CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS AND DELTA8 BETA HAIRPIN LOOP DELETION IN COMPLEX WITH CDP, MN2+ AND SYMMETRICAL PRIMER TEMPLATE 5'-AGAAAUUU
分子名称: CHLORIDE ION, CYTIDINE-5'-DIPHOSPHATE, MANGANESE (II) ION, ...
著者Edwards, T.E, Appleby, T.C.
登録日2014-10-29
公開日2015-02-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Structural basis for RNA replication by the hepatitis C virus polymerase.
Science, 347, 2015
4WTE
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BU of 4wte by Molmil
CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS AND DELTA8 BETA HAIRPIN LOOP DELETION IN COMPLEX WITH GDP, MN2+ AND SYMMETRICAL PRIMER TEMPLATE 5'-ACAAAUUU
分子名称: CHLORIDE ION, GUANOSINE-5'-DIPHOSPHATE, MANGANESE (II) ION, ...
著者Edwards, T.E, Appleby, T.C.
登録日2014-10-29
公開日2015-02-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural basis for RNA replication by the hepatitis C virus polymerase.
Science, 347, 2015
4WTG
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BU of 4wtg by Molmil
CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS AND DELTA8 BETA HAIRPIN LOOP DELETION IN COMPLEX WITH SOFOSBUVIR DIPHOSPHATE GS-607596, MN2+ AND SYMMETRICAL PRIMER TEMPLATE 5'-CAAAAUUU
分子名称: 2'-deoxy-2'-fluoro-2'-methyluridine 5'-(trihydrogen diphosphate), CHLORIDE ION, MANGANESE (II) ION, ...
著者Edwards, T.E, Appleby, T.C.
登録日2014-10-30
公開日2015-02-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural basis for RNA replication by the hepatitis C virus polymerase.
Science, 347, 2015
4WTI
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BU of 4wti by Molmil
CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS IN COMPLEX WITH RNA TEMPLATE 5'-ACGG, RNA PRIMER 5'-PCC, MN2+, AND GDP
分子名称: 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, GUANOSINE-5'-DIPHOSPHATE, ...
著者Edwards, T.E, Appleby, T.C.
登録日2014-10-30
公開日2015-02-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structural basis for RNA replication by the hepatitis C virus polymerase.
Science, 347, 2015
4WTK
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BU of 4wtk by Molmil
CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS IN COMPLEX WITH RNA TEMPLATE 5'-AGCC, RNA PRIMER 5'-PGG, MN2+, AND CDP
分子名称: 1,2-ETHANEDIOL, 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ...
著者Edwards, T.E, Appleby, T.C.
登録日2014-10-30
公開日2015-02-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural basis for RNA replication by the hepatitis C virus polymerase.
Science, 347, 2015

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