8C54
| Cryo-EM structure of NADH bound SLA dehydrogenase RlGabD from Rhizobium leguminosarum bv. trifolii SRD1565 | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, Succinate semialdehyde dehydrogenase | 著者 | Sharma, M, Meek, R.W, Armstrong, Z, Blaza, J.N, Alhifthi, A, Li, J, Goddard-Borger, E.D, Williams, S.J, Davies, G.J. | 登録日 | 2023-01-06 | 公開日 | 2023-09-20 | 最終更新日 | 2024-04-10 | 実験手法 | ELECTRON MICROSCOPY (2.52 Å) | 主引用文献 | Molecular basis of sulfolactate synthesis by sulfolactaldehyde dehydrogenase from Rhizobium leguminosarum. Chem Sci, 14, 2023
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8VB1
| Crystal structure of HIV-1 protease with GS-9770 | 分子名称: | (2S)-2-{(3M)-4-chloro-3-[1-(difluoromethyl)-1H-1,2,4-triazol-5-yl]phenyl}-2-[(2E,4R)-4-[4-(2-cyclopropyl-2H-1,2,3-triazol-4-yl)phenyl]-2-imino-5-oxo-4-(3,3,3-trifluoro-2,2-dimethylpropyl)imidazolidin-1-yl]ethyl [1-(difluoromethyl)cyclopropyl]carbamate, HIV-1 protease | 著者 | Lansdon, E.B. | 登録日 | 2023-12-11 | 公開日 | 2024-03-06 | 最終更新日 | 2024-04-17 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Preclinical characterization of a non-peptidomimetic HIV protease inhibitor with improved metabolic stability. Antimicrob.Agents Chemother., 68, 2024
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8DA2
| Acinetobacter baumannii L,D-transpeptidase | 分子名称: | L,D-transpeptidase family protein | 著者 | Toth, M, Stewart, N.K, Smith, C.A, Vakulenko, S.B. | 登録日 | 2022-06-12 | 公開日 | 2022-09-14 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | The l,d-Transpeptidase Ldt Ab from Acinetobacter baumannii Is Poorly Inhibited by Carbapenems and Has a Unique Structural Architecture. Acs Infect Dis., 8, 2022
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4XZZ
| Structure of Helicobacter pylori Csd6 in the ligand-free state | 分子名称: | Conserved hypothetical secreted protein, GLYCEROL | 著者 | Kim, H.S, Im, H.N, Yoon, H.J, Suh, S.W. | 登録日 | 2015-02-05 | 公開日 | 2015-09-02 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | The Cell Shape-determining Csd6 Protein from Helicobacter pylori Constitutes a New Family of l,d-Carboxypeptidase J.Biol.Chem., 290, 2015
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4Y4V
| Structure of Helicobacter pylori Csd6 in the D-Ala-bound state | 分子名称: | Conserved hypothetical secreted protein, D-ALANINE, GLYCEROL | 著者 | Kim, H.S, Im, H.N, Yoon, H.J, Suh, S.W. | 登録日 | 2015-02-11 | 公開日 | 2015-09-02 | 最終更新日 | 2022-03-23 | 実験手法 | X-RAY DIFFRACTION (2.04 Å) | 主引用文献 | The Cell Shape-determining Csd6 Protein from Helicobacter pylori Constitutes a New Family of l,d-Carboxypeptidase J.Biol.Chem., 290, 2015
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7JMT
| Crystal structure of schistosome BCL-2 bound to ABT-737 | 分子名称: | 4-{4-[(4'-CHLOROBIPHENYL-2-YL)METHYL]PIPERAZIN-1-YL}-N-{[4-({(1R)-3-(DIMETHYLAMINO)-1-[(PHENYLTHIO)METHYL]PROPYL}AMINO)-3-NITROPHENYL]SULFONYL}BENZAMIDE, BCL-2 protein | 著者 | Smith, N.A, Smith, B.J, Lee, E.F, Colman, P.M, Fairlie, W.D. | 登録日 | 2020-08-02 | 公開日 | 2021-02-17 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Optimization of Benzothiazole and Thiazole Hydrazones as Inhibitors of Schistosome BCL-2. Acs Infect Dis., 7, 2021
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7PJ4
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7PJ6
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7PJ5
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7PL2
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7PL5
| Crystal structure of choline-binding module (R1-R9) of LytB from Streptococcus pneumoniae | 分子名称: | CHOLINE ION, Putative endo-beta-N-acetylglucosaminidase, TRIETHYLENE GLYCOL, ... | 著者 | Molina, R, Martinez Caballero, S, Hermoso, J.A. | 登録日 | 2021-08-28 | 公開日 | 2022-09-07 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.99 Å) | 主引用文献 | Molecular basis of the final step of cell division in Streptococcus pneumoniae. Cell Rep, 42, 2023
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7PJ3
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7PL3
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7POD
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5MMH
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6E2M
| ASK1 kinase domain complex with inhibitor | 分子名称: | Mitogen-activated protein kinase kinase kinase 5, N-[3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamide | 著者 | Lansdon, E.B. | 登録日 | 2018-07-11 | 公開日 | 2018-09-19 | 最終更新日 | 2018-10-17 | 実験手法 | X-RAY DIFFRACTION (2.253 Å) | 主引用文献 | ASK1 contributes to fibrosis and dysfunction in models of kidney disease. J. Clin. Invest., 128, 2018
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6E2N
| ASK1 kinase domain complex with inhibitor | 分子名称: | Mitogen-activated protein kinase kinase kinase 5, N-[3-(4-cyclopropyl-4H-1,2,4-triazol-3-yl)phenyl][3,4'-bipyridine]-2'-carboxamide | 著者 | Lansdon, E.B. | 登録日 | 2018-07-11 | 公開日 | 2018-09-19 | 最終更新日 | 2018-10-17 | 実験手法 | X-RAY DIFFRACTION (2.098 Å) | 主引用文献 | ASK1 contributes to fibrosis and dysfunction in models of kidney disease. J. Clin. Invest., 128, 2018
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6E2O
| ASK1 kinase domain complex with inhibitor | 分子名称: | 4-(4-cyclopropyl-1H-imidazol-1-yl)-N-[3-(4-cyclopropyl-4H-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamide, Mitogen-activated protein kinase kinase kinase 5 | 著者 | Lansdon, E.B. | 登録日 | 2018-07-11 | 公開日 | 2018-09-19 | 最終更新日 | 2018-10-17 | 実験手法 | X-RAY DIFFRACTION (2.389 Å) | 主引用文献 | ASK1 contributes to fibrosis and dysfunction in models of kidney disease. J. Clin. Invest., 128, 2018
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6R5N
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6R5O
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6R5R
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6R5I
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5OAU
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5OJ1
| Penicillin Binding Protein 2x (PBP2x) from S.pneumoniae in complex with Oxacillin and a tetrasaccharide | 分子名称: | (2R,4S)-5,5-dimethyl-2-[(1R)-1-{[(5-methyl-3-phenyl-1,2-oxazol-4-yl)carbonyl]amino}-2-oxoethyl]-1,3-thiazolidine-4-carb oxylic acid, Penicillin-binding protein 2X, SODIUM ION | 著者 | Bernardo-Garcia, N, Hermoso, J.A. | 登録日 | 2017-07-20 | 公開日 | 2018-05-30 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | Allostery, Recognition of Nascent Peptidoglycan, and Cross-linking of the Cell Wall by the Essential Penicillin-Binding Protein 2x of Streptococcus pneumoniae. ACS Chem. Biol., 13, 2018
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6Z3C
| High resolution structure of RgNanOx | 分子名称: | CITRATE ANION, Gfo/Idh/MocA family oxidoreductase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE | 著者 | Naismith, J.H, Lee, M.O. | 登録日 | 2020-05-19 | 公開日 | 2020-06-03 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Uncovering a novel molecular mechanism for scavenging sialic acids in bacteria. J.Biol.Chem., 295, 2020
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