8KHD
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![BU of 8khd by Molmil](/molmil-images/mine/8khd) | The interface structure of Omicron RBD binding to 5817 Fab | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Heavy chain of 5817, Light chain of 5817, ... | 著者 | Cao, L, Wang, X. | 登録日 | 2023-08-21 | 公開日 | 2024-04-17 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Identification of a broad sarbecovirus neutralizing antibody targeting a conserved epitope on the receptor-binding domain. Cell Rep, 43, 2024
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8KHC
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![BU of 8khc by Molmil](/molmil-images/mine/8khc) | SARS-CoV-2 Omicron spike in complex with 5817 Fab | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Heavy chain of 5817 Fab, ... | 著者 | Cao, L, Wang, X. | 登録日 | 2023-08-21 | 公開日 | 2024-04-17 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Identification of a broad sarbecovirus neutralizing antibody targeting a conserved epitope on the receptor-binding domain. Cell Rep, 43, 2024
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8QNI
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8QNG
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8QNH
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![BU of 8qnh by Molmil](/molmil-images/mine/8qnh) | Crystal structure of the E3 ubiquitin ligase Cbl-b with an allosteric inhibitor (WO2020264398 Ex23) | 分子名称: | 2-{3-[(1s,3R)-3-methyl-1-(4-methyl-4H-1,2,4-triazol-3-yl)cyclobutyl]phenyl}-6-{[(3S)-3-methylpiperidin-1-yl]methyl}-4-(trifluoromethyl)-2,3-dihydro-1H-isoindol-1-one, E3 ubiquitin-protein ligase CBL-B, SODIUM ION, ... | 著者 | Schimpl, M. | 登録日 | 2023-09-26 | 公開日 | 2023-11-22 | 最終更新日 | 2024-01-03 | 実験手法 | X-RAY DIFFRACTION (2.001 Å) | 主引用文献 | Discovery of a Novel Benzodiazepine Series of Cbl-b Inhibitors for the Enhancement of Antitumor Immunity. Acs Med.Chem.Lett., 14, 2023
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8D5P
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![BU of 8d5p by Molmil](/molmil-images/mine/8d5p) | Mouse TCR TG6 | 分子名称: | TCR-alpha, TCR-beta | 著者 | Wang, Y, Dai, S. | 登録日 | 2022-06-05 | 公開日 | 2022-09-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Peptide Centric V beta Specific Germline Contacts Shape a Specialist T Cell Response. Front Immunol, 13, 2022
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8D5N
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![BU of 8d5n by Molmil](/molmil-images/mine/8d5n) | Crystal structure of Ld-HF10 | 分子名称: | 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, Beta-2-microglobulin, ... | 著者 | Wang, Y, Dai, S. | 登録日 | 2022-06-05 | 公開日 | 2022-09-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Peptide Centric V beta Specific Germline Contacts Shape a Specialist T Cell Response. Front Immunol, 13, 2022
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8D5Q
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![BU of 8d5q by Molmil](/molmil-images/mine/8d5q) | TCR TG6 in complex with Ld-HF10 | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Dense granule protein 6, HF10 peptide, ... | 著者 | Wang, Y, Dai, S. | 登録日 | 2022-06-05 | 公開日 | 2022-09-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.501 Å) | 主引用文献 | Peptide Centric V beta Specific Germline Contacts Shape a Specialist T Cell Response. Front Immunol, 13, 2022
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6INW
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![BU of 6inw by Molmil](/molmil-images/mine/6inw) | A Pericyclic Reaction enzyme | 分子名称: | O-methyltransferase lepI, S-ADENOSYLMETHIONINE | 著者 | Feng, Y, Chang, M, Wang, H, Liu, Z, Zhou, Y. | 登録日 | 2018-10-28 | 公開日 | 2019-07-03 | 実験手法 | X-RAY DIFFRACTION (1.798 Å) | 主引用文献 | Crystal structure of the multifunctional SAM-dependent enzyme LepI provides insights into its catalytic mechanism. Biochem.Biophys.Res.Commun., 515, 2019
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5MES
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![BU of 5mes by Molmil](/molmil-images/mine/5mes) | MCL1 FAB COMPLEX IN COMPLEX WITH COMPOUND 29 | 分子名称: | (5~{R},13~{S},17~{S})-5-[[4-chloranyl-3-(2-phenylethyl)phenyl]methyl]-13-[(4-chlorophenyl)methyl]-8-methyl-1,4,8,12,16-pentazatricyclo[15.8.1.0^{20,25}]hexacosa-20(25),21,23-triene-3,7,15,26-tetrone, Heavy Chain, Induced myeloid leukemia cell differentiation protein Mcl-1 homolog,Induced myeloid leukemia cell differentiation protein Mcl-1, ... | 著者 | Hargreaves, D. | 登録日 | 2016-11-16 | 公開日 | 2017-01-18 | 最終更新日 | 2017-03-08 | 実験手法 | X-RAY DIFFRACTION (2.24 Å) | 主引用文献 | Structure Based Design of Non-Natural Peptidic Macrocyclic Mcl-1 Inhibitors. ACS Med Chem Lett, 8, 2017
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7P13
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![BU of 7p13 by Molmil](/molmil-images/mine/7p13) | 2.29 A Mycobacterium tuberculosis EspB. | 分子名称: | ESX-1 secretion-associated protein EspB | 著者 | Gijsbers, A, Zhang, Y, Vinciauskaite, V, Siroy, A, Gao, Y, Tria, G, Mathew, A, Sanchez-Puig, N, Lopez-Iglesias, C, Peters, P.J, Ravelli, R.B.G. | 登録日 | 2021-07-01 | 公開日 | 2021-08-18 | 最終更新日 | 2021-10-13 | 実験手法 | ELECTRON MICROSCOPY (2.29 Å) | 主引用文献 | Priming mycobacterial ESX-secreted protein B to form a channel-like structure. Curr Res Struct Biol, 3, 2021
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8DD5
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![BU of 8dd5 by Molmil](/molmil-images/mine/8dd5) | Crystal structure of KAT6A in complex with inhibitor CTx-648 (PF-9363) | 分子名称: | 2,6-dimethoxy-N-{4-methoxy-6-[(1H-pyrazol-1-yl)methyl]-1,2-benzoxazol-3-yl}benzene-1-sulfonamide, Histone acetyltransferase KAT6A, ZINC ION | 著者 | Greasley, S.E, Johnson, E, Brodsky, O. | 登録日 | 2022-06-17 | 公開日 | 2023-07-05 | 実験手法 | X-RAY DIFFRACTION (2.58 Å) | 主引用文献 | Targeting KAT6A/KAT6B dependencies in breast cancer with a novel selective, orally bioavailable KAT6 inhibitor, CTx-648/PF-9363 To Be Published
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4RGQ
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![BU of 4rgq by Molmil](/molmil-images/mine/4rgq) | Crystal structure of the Methanocaldococcus jannaschii G1PDH with NADPH and DHAP | 分子名称: | 1,2-ETHANEDIOL, 1,3-DIHYDROXYACETONEPHOSPHATE, Glycerol-1-phosphate dehydrogenase, ... | 著者 | Carbone, V, Ronimus, R.S, Schofield, L.R, Sutherland-Smith, A.J. | 登録日 | 2014-09-30 | 公開日 | 2015-07-22 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.23 Å) | 主引用文献 | Structure and Evolution of the Archaeal Lipid Synthesis Enzyme sn-Glycerol-1-phosphate Dehydrogenase. J.Biol.Chem., 290, 2015
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4RGV
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![BU of 4rgv by Molmil](/molmil-images/mine/4rgv) | Crystal structure of the Methanocaldococcus jannaschii G1PDH | 分子名称: | Glycerol-1-phosphate dehydrogenase, MAGNESIUM ION, ZINC ION | 著者 | Carbone, V, Ronimus, R.S, Schofield, L.R, Sutherland-Smith, A.J. | 登録日 | 2014-09-30 | 公開日 | 2015-07-22 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Structure and Evolution of the Archaeal Lipid Synthesis Enzyme sn-Glycerol-1-phosphate Dehydrogenase. J.Biol.Chem., 290, 2015
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4RFL
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![BU of 4rfl by Molmil](/molmil-images/mine/4rfl) | Crystal structure of G1PDH with NADPH from Methanocaldococcus jannaschii | 分子名称: | 1,2-ETHANEDIOL, Glycerol-1-phosphate dehydrogenase [NAD(P)+], NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... | 著者 | Carbone, V, Ronimus, R.S, Schofield, L.R, Sutherland-Smith, A.J. | 登録日 | 2014-09-26 | 公開日 | 2015-07-22 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structure and Evolution of the Archaeal Lipid Synthesis Enzyme sn-Glycerol-1-phosphate Dehydrogenase. J.Biol.Chem., 290, 2015
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7Y77
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![BU of 7y77 by Molmil](/molmil-images/mine/7y77) | Crystal structure of rice NAL1 | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Protein NARROW LEAF 1 | 著者 | Yan, J.J, Guan, Z.Y, Yin, P, Xiong, L.Z. | 登録日 | 2022-06-21 | 公開日 | 2023-07-12 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Serine protease NAL1 exerts pleiotropic functions through degradation of TOPLESS-related corepressor in rice. Nat.Plants, 9, 2023
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1RHU
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![BU of 1rhu by Molmil](/molmil-images/mine/1rhu) | CRYSTAL STRUCTURE OF THE COMPLEX OF CASPASE-3 WITH A 5,6,7 TRICYCLIC PEPTIDOMIMETIC INHIBITOR | 分子名称: | (3S)-3-[({(2S)-5-[(N-ACETYL-L-ALPHA-ASPARTYL)AMINO]-4-OXO-1,2,4,5,6,7-HEXAHYDROAZEPINO[3,2,1-HI]INDOL-2-YL}CARBONYL)AMINO]-5-(BENZYLSULFANYL)-4-OXOPENTANOIC ACID, Caspase-3 | 著者 | Becker, J.W, Rotonda, J, Soisson, S.M. | 登録日 | 2003-11-14 | 公開日 | 2004-05-11 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.51 Å) | 主引用文献 | Reducing the Peptidyl Features of Caspase-3 Inhibitors: A Structural Analysis. J.Med.Chem., 47, 2004
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1RE1
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4ZQA
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![BU of 4zqa by Molmil](/molmil-images/mine/4zqa) | |
1RHQ
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8D1G
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![BU of 8d1g by Molmil](/molmil-images/mine/8d1g) | hBest2 Ca2+-bound open state | 分子名称: | 1,2-DIMYRISTOYL-RAC-GLYCERO-3-PHOSPHOCHOLINE, 2-[2-[(1~{S},2~{S},4~{S},5'~{R},6~{R},7~{S},8~{R},9~{S},12~{S},13~{R},16~{S})-5',7,9,13-tetramethylspiro[5-oxapentacyclo[10.8.0.0^{2,9}.0^{4,8}.0^{13,18}]icos-18-ene-6,2'-oxane]-16-yl]oxyethyl]propane-1,3-diol, Bestrophin-2, ... | 著者 | Owji, A.P, Kittredge, A, Hendrickson, W.A, Tingting, Y. | 登録日 | 2022-05-27 | 公開日 | 2022-07-13 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (2.07 Å) | 主引用文献 | Structures and gating mechanisms of human bestrophin anion channels. Nat Commun, 13, 2022
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8D1O
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![BU of 8d1o by Molmil](/molmil-images/mine/8d1o) | hBest1_345 Ca2+-bound open state | 分子名称: | 1,2-DIMYRISTOYL-RAC-GLYCERO-3-PHOSPHOCHOLINE, Bestrophin-1, CALCIUM ION | 著者 | Owji, A.P, Kittredge, A, Hendrickson, W.A, Tingting, Y. | 登録日 | 2022-05-27 | 公開日 | 2022-07-13 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (2.44 Å) | 主引用文献 | Structures and gating mechanisms of human bestrophin anion channels. Nat Commun, 13, 2022
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8D1I
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![BU of 8d1i by Molmil](/molmil-images/mine/8d1i) | hBest1 1uM Ca2+ (Ca2+-bound) closed state | 分子名称: | 1,2-DIMYRISTOYL-RAC-GLYCERO-3-PHOSPHOCHOLINE, Bestrophin-1, CALCIUM ION | 著者 | Owji, A.P, Kittredge, A, Hendrickson, W.A, Tingting, Y. | 登録日 | 2022-05-27 | 公開日 | 2022-07-13 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (1.82 Å) | 主引用文献 | Structures and gating mechanisms of human bestrophin anion channels. Nat Commun, 13, 2022
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8D1K
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![BU of 8d1k by Molmil](/molmil-images/mine/8d1k) | hBest1 Ca2+-bound partially open neck state | 分子名称: | 1,2-DIMYRISTOYL-RAC-GLYCERO-3-PHOSPHOCHOLINE, Bestrophin-1, CALCIUM ION | 著者 | Owji, A.P, Kittredge, A, Hendrickson, W.A, Tingting, Y. | 登録日 | 2022-05-27 | 公開日 | 2022-07-13 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (2.28 Å) | 主引用文献 | Structures and gating mechanisms of human bestrophin anion channels. Nat Commun, 13, 2022
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8D1N
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![BU of 8d1n by Molmil](/molmil-images/mine/8d1n) | bBest2_345 Ca2+-bound open state | 分子名称: | 1,2-DIMYRISTOYL-RAC-GLYCERO-3-PHOSPHOCHOLINE, 2-[2-[(1~{S},2~{S},4~{S},5'~{R},6~{R},7~{S},8~{R},9~{S},12~{S},13~{R},16~{S})-5',7,9,13-tetramethylspiro[5-oxapentacyclo[10.8.0.0^{2,9}.0^{4,8}.0^{13,18}]icos-18-ene-6,2'-oxane]-16-yl]oxyethyl]propane-1,3-diol, Bestrophin, ... | 著者 | Owji, A.P, Kittredge, A, Hendrickson, W.A, Tingting, Y. | 登録日 | 2022-05-27 | 公開日 | 2022-07-13 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (1.93 Å) | 主引用文献 | Structures and gating mechanisms of human bestrophin anion channels. Nat Commun, 13, 2022
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