Loading
PDBj
メニューPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
2IZZ
DownloadVisualize
BU of 2izz by Molmil
Crystal structure of human pyrroline-5-carboxylate reductase
分子名称: 1,2-ETHANEDIOL, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, PYRROLINE-5-CARBOXYLATE REDUCTASE 1
著者Pike, A.C.W, Guo, K, Kavanagh, K, Pilka, E.S, Berridge, G, Colebrook, S, Bray, J, Salah, E, Savitsky, P, Papagrigoriou, E, Turnbull, A.P, von Delft, F, Arrowsmith, C, Edwards, A, Weigelt, J, Sundstrom, M, Oppermann, U.
登録日2006-07-31
公開日2006-08-01
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Crystal Structure of Human Pyrroline-5-Carboxylate Reductase
To be Published
2IXS
DownloadVisualize
BU of 2ixs by Molmil
Structure of SdaI restriction endonuclease
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, SDAI RESTRICTION ENDONUCLEASE, ...
著者Tamulaitiene, G, Jakubauskas, A, Urbanke, C, Huber, R, Grazulis, S, Siksnys, V.
登録日2006-07-11
公開日2006-09-14
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The Crystal Structure of the Rare-Cutting Restriction Enzyme Sdai Reveals Unexpected Domain Architecture
Structure, 14, 2006
2J6B
DownloadVisualize
BU of 2j6b by Molmil
crystal structure of AFV3-109, a highly conserved protein from crenarchaeal viruses
分子名称: AFV3-109
著者Keller, J, Leulliot, N, Cambillau, C, Campanacci, V, Porciero, S, Prangishvili, D, Cortez, D, Quevillon-Cheruel, S, Van Tilbeurgh, H.
登録日2006-09-27
公開日2007-02-20
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Crystal Structure of Afv3-109, a Highly Conserved Protein from Crenarchaeal Viruses.
Virol J., 4, 2007
8I7S
DownloadVisualize
BU of 8i7s by Molmil
The crystal structure of human abl1 kinase domain in complex with ABL1-B1
分子名称: 5-[3-(2-methoxy-5-oxidanyl-phenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]-N,N-dimethyl-pyridine-3-carboxamide, Tyrosine-protein kinase ABL1
著者Zhu, C, Zhang, Z.
登録日2023-02-02
公開日2024-10-09
実験手法X-RAY DIFFRACTION (1.94635463 Å)
主引用文献Rationally designed BCR-ABL kinase inhibitors for improved leukemia treatment via covalent and pro-/dual-drug targeting strategies.
J Adv Res, 2024
8I7Z
DownloadVisualize
BU of 8i7z by Molmil
The crystal structure of human abl1 kinase domain in complex with ABL1-B5
分子名称: 5-[3-(2-methoxy-5-oxidanyl-phenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]-N,N-dimethyl-pyridine-3-carboxamide, BETA-ALANINE, Tyrosine-protein kinase ABL1
著者Zhu, C, Zhang, Z.
登録日2023-02-02
公開日2024-10-23
実験手法X-RAY DIFFRACTION (2.25495815 Å)
主引用文献Rationally designed BCR-ABL kinase inhibitors for improved leukemia treatment via covalent and pro-/dual-drug targeting strategies.
J Adv Res, 2024
8I7T
DownloadVisualize
BU of 8i7t by Molmil
The crystal structure of human abl1 kinase domain in complex with ABL1-B4
分子名称: Tyrosine-protein kinase ABL1, [3-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-3-yl]-4-methoxy-phenyl] ethanesulfonate
著者Zhu, C, Zhang, Z.
登録日2023-02-02
公開日2024-10-23
実験手法X-RAY DIFFRACTION (2.80004954 Å)
主引用文献Rationally designed BCR-ABL kinase inhibitors for improved leukemia treatment via covalent and pro-/dual-drug targeting strategies.
J Adv Res, 2024
2J9P
DownloadVisualize
BU of 2j9p by Molmil
Crystal structure of the Bacillus subtilis PBP4a, and its complex with a peptidoglycan mimetic peptide.
分子名称: (2R)-2-AMINO-7-{[(1R)-1-CARBOXYETHYL]AMINO}-7-OXOHEPTANOIC ACID, D-ALANINE, D-alanyl-D-alanine carboxypeptidase DacC
著者Sauvage, E, Herman, R, Kerff, F, Duez, C, Charlier, P.
登録日2006-11-15
公開日2007-07-03
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structure of the Bacillus subtilis penicillin-binding protein 4a, and its complex with a peptidoglycan mimetic peptide.
J. Mol. Biol., 371, 2007
2IKK
DownloadVisualize
BU of 2ikk by Molmil
Structural Genomics, the crystal structure of the C-terminal domain of Yurk from Bacillus subtilis subsp. subtilis str. 168
分子名称: Hypothetical transcriptional regulator yurK, SULFATE ION
著者Tan, K, Hatzos, C, Abdullah, J, Joachimiak, A, Midwest Center for Structural Genomics (MCSG)
登録日2006-10-02
公開日2006-10-31
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The crystal structure of the C-terminal domain of Yurk from Bacillus subtilis subsp. subtilis str. 168
To be Published
2IDK
DownloadVisualize
BU of 2idk by Molmil
Crystal Structure of Rat Glycine N-Methyltransferase Complexed With Folate
分子名称: 5-METHYL-5,6,7,8-TETRAHYDROFOLIC ACID, Glycine N-methyltransferase
著者Luka, Z, Pakhomova, S, Loukachevitch, L.V, Egli, M, Newcomer, M.E, Wagner, C.
登録日2006-09-15
公開日2006-12-19
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献5-methyltetrahydrofolate is bound in intersubunit areas of rat liver folate-binding protein glycine N-methyltransferase.
J.Biol.Chem., 282, 2007
8IQY
DownloadVisualize
BU of 8iqy by Molmil
Asterias forbesii ferritin mutant-P156H
分子名称: Ferritin
著者Zhao, G, Zhang, C, Zang, J, Zhang, T.
登録日2023-03-17
公開日2024-02-21
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Preparation and Unique Three-Dimensional Self-Assembly Property of Starfish Ferritin.
Foods, 12, 2023
8IQV
DownloadVisualize
BU of 8iqv by Molmil
Asterias forbesii ferritin
分子名称: Ferritin
著者Zhao, G, Zhang, C, Zang, J, Zhang, T.
登録日2023-03-17
公開日2024-02-21
実験手法X-RAY DIFFRACTION (1.91 Å)
主引用文献Preparation and Unique Three-Dimensional Self-Assembly Property of Starfish Ferritin.
Foods, 12, 2023
2IQI
DownloadVisualize
BU of 2iqi by Molmil
Crystal structure of protein XCC0632 from Xanthomonas campestris, Pfam DUF330
分子名称: Hypothetical protein XCC0632
著者Bonanno, J.B, Gilmore, J, Bain, K.T, Mckenzie, C, Pelletier, L, Wasserman, S, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2006-10-13
公開日2006-11-07
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structure of hypothetical protein XCC0632 from Xanthomonas campestris pv. campestris
To be Published
8IQW
DownloadVisualize
BU of 8iqw by Molmil
AfFer(Asterias forbesii ferritin) mutant-P156H
分子名称: Ferritin
著者Zhao, G, Zhang, C, Zang, J, Zhang, T.
登録日2023-03-17
公開日2024-02-21
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Preparation and Unique Three-Dimensional Self-Assembly Property of Starfish Ferritin.
Foods, 12, 2023
8IQZ
DownloadVisualize
BU of 8iqz by Molmil
Asterias forbesii ferritin mutant-P156F
分子名称: Ferritin
著者Zhao, G, Zhang, C, Zang, J, Zhang, T.
登録日2023-03-17
公開日2024-02-21
実験手法X-RAY DIFFRACTION (4.19 Å)
主引用文献Preparation and Unique Three-Dimensional Self-Assembly Property of Starfish Ferritin.
Foods, 12, 2023
8IY7
DownloadVisualize
BU of 8iy7 by Molmil
Cryo-EM structure of DIP-2I8I fibril polymorph1
分子名称: GLY-PHI-GLY-ASN-GLY-ASN-GLY-PHI-GLY
著者Li, D.N, Ma, Y.Y, Li, D, Dai, B, Liu, C.
登録日2023-04-04
公開日2024-04-10
実験手法ELECTRON MICROSCOPY (3.71 Å)
主引用文献Cryo-EM structure of DIP-2I8I fibril polymorph1
To Be Published
8IZZ
DownloadVisualize
BU of 8izz by Molmil
Cryo-EM structure of DIP-2I8I polymorph 2
分子名称: GLY-PHI-GLY-ASN-GLY-ASN-GLY-PHI-GLY
著者Li, D.N, Ma, Y.Y, Li, D, Dai, B, Liu, C.
登録日2023-04-09
公開日2024-04-10
実験手法ELECTRON MICROSCOPY (3.75 Å)
主引用文献Cryo-EM structure of DIP-2I8I fibril polymorph 2
To Be Published
2IVF
DownloadVisualize
BU of 2ivf by Molmil
Ethylbenzene dehydrogenase from Aromatoleum aromaticum
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-AMINO-5,6-DIMERCAPTO-7-METHYL-3,7,8A,9-TETRAHYDRO-8-OXA-1,3,9,10-TETRAAZA-ANTHRACEN-4-ONE GUANOSINE DINUCLEOTIDE, ACETATE ION, ...
著者Kloer, D.P, Hagel, C, Heider, J, Schulz, G.E.
登録日2006-06-13
公開日2006-09-14
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.88 Å)
主引用文献Crystal Structure of Ethylbenzene Dehydrogenase from Aromatoleum Aromaticum
Structure, 14, 2006
2J0G
DownloadVisualize
BU of 2j0g by Molmil
L-ficolin complexed to N-acetyl-mannosamine
分子名称: 2-acetamido-2-deoxy-alpha-D-mannopyranose, CALCIUM ION, FICOLIN-2, ...
著者Garlatti, V, Gaboriaud, C.
登録日2006-08-03
公開日2007-01-23
最終更新日2025-04-09
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Structural Insights Into the Innate Immune Recognition Specificities of L- and H-Ficolins.
Embo J., 26, 2007
2J86
DownloadVisualize
BU of 2j86 by Molmil
Structural analysis of the PP2C Family Phosphatase tPphA of Thermosynechococcus elongatus
分子名称: MAGNESIUM ION, PROTEIN SERINE-THREONINE PHOSPHATASE
著者Schlicker, C, Kloft, N, Forchhammer, K, Becker, S.
登録日2006-10-19
公開日2007-11-06
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.05 Å)
主引用文献Structural Analysis of the Pp2C Phosphatase Tppha from Thermosynechococcus Elongatus: A Flexible Flap Subdomain Controls Access to the Catalytic Site.
J.Mol.Biol., 376, 2008
8GCC
DownloadVisualize
BU of 8gcc by Molmil
T. cruzi topoisomerase II alpha bound to dsDNA and the covalent inhibitor CT1
分子名称: 2-{3-[(Z)-iminomethyl]-1H-1,2,4-triazol-1-yl}-1-{(3M)-3-[2-(trifluoromethyl)phenyl]-6H-pyrrolo[3,4-b]pyridin-6-yl}ethan-1-one, DNA (28-MER), DNA topoisomerase 2
著者Schenk, A, Deniston, C, Noeske, J.
登録日2023-03-01
公開日2023-07-12
最終更新日2024-11-06
実験手法ELECTRON MICROSCOPY (2.94 Å)
主引用文献Cyanotriazoles are selective topoisomerase II poisons that rapidly cure trypanosome infections.
Science, 380, 2023
2ID2
DownloadVisualize
BU of 2id2 by Molmil
GAPN T244S mutant X-ray structure at 2.5 A
分子名称: NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, NADP-dependent glyceraldehyde-3-phosphate dehydrogenase, SULFATE ION
著者Pailot, A, D'Ambrosio, K, Corbier, C, Talfournier, F, Branlant, G.
登録日2006-09-14
公開日2007-09-18
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Invariant Thr(244) is essential for the efficient acylation step of the non-phosphorylating glyceraldehyde-3-phosphate dehydrogenase from Streptococcus mutans.
Biochem.J., 400, 2006
2IZS
DownloadVisualize
BU of 2izs by Molmil
Structure of casein kinase gamma 3 in complex with inhibitor
分子名称: CASEIN KINASE I ISOFORM GAMMA-3, CHLORIDE ION, MAGNESIUM ION, ...
著者Bunkoczi, G, Salah, E, Rellos, P, Das, S, Fedorov, O, Savitsky, P, Debreczeni, J.E, Gileadi, O, Sundstrom, M, Edwards, A, Arrowsmith, C, Weigelt, J, von Delft, F, Knapp, S.
登録日2006-07-26
公開日2006-08-01
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Inhibitor Binding by Casein Kinases
To be Published
7B83
DownloadVisualize
BU of 7b83 by Molmil
Structure of SARS-CoV-2 Main Protease bound to pyrithione zinc
分子名称: 3C-like proteinase, 9-oxa-7-thia-1-azonia-8$l^{2}-zincabicyclo[4.3.0]nona-1,3,5-triene, CHLORIDE ION, ...
著者Guenther, S, Reinke, P, Oberthuer, D, Yefanov, O, Gelisio, L, Ginn, H, Lieske, J, Domaracky, M, Brehm, W, Rahmani Mashour, A, White, T.A, Knoska, J, Pena Esperanza, G, Koua, F, Tolstikova, A, Groessler, M, Fischer, P, Hennicke, V, Fleckenstein, H, Trost, F, Galchenkova, M, Gevorkov, Y, Li, C, Awel, S, Paulraj, L.X, Ullah, N, Falke, S, Alves Franca, B, Schwinzer, M, Brognaro, H, Werner, N, Perbandt, M, Tidow, H, Seychell, B, Beck, T, Meier, S, Doyle, J.J, Giseler, H, Melo, D, Dunkel, I, Lane, T.J, Peck, A, Saouane, S, Hakanpaeae, J, Meyer, J, Noei, H, Gribbon, P, Ellinger, B, Kuzikov, M, Wolf, M, Zhang, L, Ehrt, C, Pletzer-Zelgert, J, Wollenhaupt, J, Feiler, C, Weiss, M, Schulz, E.C, Mehrabi, P, Norton-Baker, B, Schmidt, C, Lorenzen, K, Schubert, R, Han, H, Chari, A, Fernandez Garcia, Y, Turk, D, Hilgenfeld, R, Rarey, M, Zaliani, A, Chapman, H.N, Pearson, A, Betzel, C, Meents, A.
登録日2020-12-12
公開日2021-01-13
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献X-ray screening identifies active site and allosteric inhibitors of SARS-CoV-2 main protease.
Science, 372, 2021
6Q0Q
DownloadVisualize
BU of 6q0q by Molmil
Crystal structure of Human galectin-3 CRD in complex with Methyl 3-O-(1-{3-O-[1-(b-D-galactopyranosyl)-1,2,3-triazol-4-yl]-methyl-b-D-galactopyranosyl}-1,2,3-triazol-4-yl)-methyl-b-D-galactopyranoside
分子名称: (2~{R},3~{R},4~{S},5~{R},6~{R})-2-(hydroxymethyl)-6-[4-[[(2~{R},3~{S},4~{S},5~{R},6~{R})-2-(hydroxymethyl)-6-[4-[[(2~{R},3~{S},4~{S},5~{R},6~{R})-2-(hydroxymethyl)-6-methoxy-3,5-bis(oxidanyl)oxan-4-yl]oxymethyl]-1,2,3-triazol-1-yl]-3,5-bis(oxidanyl)oxan-4-yl]oxymethyl]-1,2,3-triazol-1-yl]oxane-3,4,5-triol, CHLORIDE ION, Galectin-3
著者Kishor, C, Blanchard, H.
登録日2019-08-02
公開日2020-04-29
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.98601174 Å)
主引用文献Linear triazole-linked pseudo oligogalactosides as scaffolds for galectin inhibitor development.
Chem.Biol.Drug Des., 96, 2020
6Q17
DownloadVisualize
BU of 6q17 by Molmil
Crystal structure of Human galectin-3 CRD in complex with Methyl 3-O-[1-(b-D-galactopyranosyl)-1,2,3-triazol-4-yl]-methyl-b-D-galactopyranoside
分子名称: CHLORIDE ION, Galectin-3, methyl 3-O-[(1-beta-D-galactopyranosyl-1H-1,2,3-triazol-4-yl)methyl]-beta-D-galactopyranoside
著者Kishor, C, Blanchard, H.
登録日2019-08-02
公開日2020-04-29
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献Linear triazole-linked pseudo oligogalactosides as scaffolds for galectin inhibitor development.
Chem.Biol.Drug Des., 96, 2020

238582

件を2025-07-09に公開中

PDB statisticsPDBj update infoContact PDBjnumon