3WUU
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4NJ3
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3S4Q
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![BU of 3s4q by Molmil](/molmil-images/mine/3s4q) | P38 alpha kinase complexed with a pyrazolo-triazine based inhibitor | 分子名称: | 3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-N-cyclopropyl-4-methylbenzamide, Mitogen-activated protein kinase 14 | 著者 | Sack, J.S. | 登録日 | 2011-05-20 | 公開日 | 2012-02-01 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.27 Å) | 主引用文献 | Discovery of pyrrolo[2,1-f][1,2,4]triazine C6-ketones as potent, orally active p38α MAP kinase inhibitors. Bioorg.Med.Chem.Lett., 21, 2011
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4JDI
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7LYG
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7LYF
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2M8J
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![BU of 2m8j by Molmil](/molmil-images/mine/2m8j) | Structure of Pin1 WW domain phospho-mimic S16E | 分子名称: | Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | 著者 | Luh, L.M, Kirchner, D.K, Loehr, F, Haensel, R, Doetsch, V. | 登録日 | 2013-05-22 | 公開日 | 2014-04-09 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Molecular crowding drives active Pin1 into nonspecific complexes with endogenous proteins prior to substrate recognition. J.Am.Chem.Soc., 135, 2013
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7MEL
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![BU of 7mel by Molmil](/molmil-images/mine/7mel) | Sco GlgEI-V279S in complex with 4-alpha-glucoside of validamine | 分子名称: | (1R,2R,3S,4S,6R)-4-amino-2,3-dihydroxy-6-(hydroxymethyl)cyclohexyl alpha-D-glucopyranoside, 1,2-ETHANEDIOL, Alpha-1,4-glucan:maltose-1-phosphate maltosyltransferase 1, ... | 著者 | Jayasinghe, T.D, Ronning, D.R. | 登録日 | 2021-04-06 | 公開日 | 2021-07-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Stereoselective synthesis of a 4-alpha-glucoside of valienamine and its X-ray structure in complex with Streptomyces coelicolor GlgE1-V279S. Sci Rep, 11, 2021
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4KIQ
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4KS8
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![BU of 4ks8 by Molmil](/molmil-images/mine/4ks8) | PAK6 kinase domain in complex with sunitinib | 分子名称: | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carbo xamide, Serine/threonine-protein kinase PAK 6 | 著者 | Gao, J, Boggon, T.J. | 登録日 | 2013-05-17 | 公開日 | 2013-09-11 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Substrate and Inhibitor Specificity of the Type II p21-Activated Kinase, PAK6. Plos One, 8, 2013
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4KS7
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7Z7P
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7Z7O
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7Z7Q
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4KIP
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4GH4
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![BU of 4gh4 by Molmil](/molmil-images/mine/4gh4) | Crystal Structure of Foot and Mouth Disease Virus A22 Serotype | 分子名称: | capsid protein VP1, capsid protein VP2, capsid protein VP3, ... | 著者 | Kotecha, A, Jinshan, R, Curry, S, Fry, E, Stuart, D. | 登録日 | 2012-08-07 | 公開日 | 2013-02-20 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Perturbations in the surface structure of A22 Iraq foot-and-mouth disease virus accompanying coupled changes in host cell specificity and antigenicity. Structure, 4, 1996
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2M8I
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![BU of 2m8i by Molmil](/molmil-images/mine/2m8i) | Structure of Pin1 WW domain | 分子名称: | Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | 著者 | Luh, L.M, Kirchner, D.K, Loehr, F, Haensel, R, Doetsch, V. | 登録日 | 2013-05-22 | 公開日 | 2014-04-09 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Molecular crowding drives active Pin1 into nonspecific complexes with endogenous proteins prior to substrate recognition. J.Am.Chem.Soc., 135, 2013
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7MGY
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![BU of 7mgy by Molmil](/molmil-images/mine/7mgy) | Sco GlgEI-V279S in complex with 4-alpha-glucoside of valienamine | 分子名称: | (1R,4S,5S,6R)-4-amino-5,6-dihydroxy-2-(hydroxymethyl)cyclohex-2-en-1-yl alpha-D-glucopyranoside, Alpha-1,4-glucan:maltose-1-phosphate maltosyltransferase 1, DI(HYDROXYETHYL)ETHER, ... | 著者 | Jayasinghe, T.D, Ronning, D.R. | 登録日 | 2021-04-13 | 公開日 | 2021-07-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | Stereoselective synthesis of a 4-⍺-glucoside of valienamine and its X-ray structure in complex with Streptomyces coelicolor GlgE1-V279S. Sci Rep, 11, 2021
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4JDK
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4JDH
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4KIN
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2EWL
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![BU of 2ewl by Molmil](/molmil-images/mine/2ewl) | |
2F8B
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4JDJ
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1YYF
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![BU of 1yyf by Molmil](/molmil-images/mine/1yyf) | Correction of X-ray Intensities from an HslV-HslU co-crystal containing lattice translocation defects | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ATP-dependent hsl protease ATP-binding subunit hslU, ATP-dependent protease hslV | 著者 | Wang, J, Rho, S.H, Park, H.H, Eom, S.H. | 登録日 | 2005-02-24 | 公開日 | 2005-07-12 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (4.16 Å) | 主引用文献 | Correction of X-ray intensities from an HslV-HslU co-crystal containing lattice-translocation defects. Acta Crystallogr.,Sect.D, 61, 2005
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