1A39
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![BU of 1a39 by Molmil](/molmil-images/mine/1a39) | HUMICOLA INSOLENS ENDOCELLULASE EGI S37W, P39W DOUBLE-MUTANT | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, ENDOGLUCANASE I | 著者 | Davies, G.J, Ducros, V, Lewis, R.J, Borchert, T.V, Schulein, M. | 登録日 | 1998-01-28 | 公開日 | 1999-03-02 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Oligosaccharide specificity of a family 7 endoglucanase: insertion of potential sugar-binding subsites. J.Biotechnol., 57, 1997
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1CNN
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![BU of 1cnn by Molmil](/molmil-images/mine/1cnn) | OMEGA-CONOTOXIN MVIIC FROM CONUS MAGUS | 分子名称: | OMEGA-CONOTOXIN MVIIC | 著者 | Nielsen, K.J, Adams, D, Thomas, L, Bond, T, Alewood, P.F, Craik, D.J, Lewis, R.J. | 登録日 | 1999-05-20 | 公開日 | 2000-05-31 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure-activity relationships of omega-conotoxins MVIIA, MVIIC and 14 loop splice hybrids at N and P/Q-type calcium channels. J.Mol.Biol., 289, 1999
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1A0M
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![BU of 1a0m by Molmil](/molmil-images/mine/1a0m) | 1.1 ANGSTROM CRYSTAL STRUCTURE OF A-CONOTOXIN [TYR15]-EPI | 分子名称: | ALPHA-CONOTOXIN [TYR15]-EPI | 著者 | Hu, S.-H, Loughnan, M, Miller, R, Weeks, C.M, Blessing, R.H, Alewood, P.F, Lewis, R.J, Martin, J.L. | 登録日 | 1997-12-03 | 公開日 | 1999-01-13 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.1 Å) | 主引用文献 | The 1.1 A resolution crystal structure of [Tyr15]EpI, a novel alpha-conotoxin from Conus episcopatus, solved by direct methods. Biochemistry, 37, 1998
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1E3A
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![BU of 1e3a by Molmil](/molmil-images/mine/1e3a) | A slow processing precursor penicillin acylase from Escherichia coli | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, CHLORIDE ION, ... | 著者 | Hewitt, L, Kasche, V, Lummer, K, Lewis, R.J, Murshudov, G.N, Verma, C.S, Dodson, G.G, Wilson, K.S. | 登録日 | 2000-06-07 | 公開日 | 2000-11-29 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure of a Slow Processing Precursor Penicillin Acylase from Escherichia Coli Reveals the Linker Peptide Blocking the Active-Site Cleft J.Mol.Biol., 302, 2000
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1AV3
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![BU of 1av3 by Molmil](/molmil-images/mine/1av3) | POTASSIUM CHANNEL BLOCKER KAPPA CONOTOXIN PVIIA FROM C. PURPURASCENS, NMR, 20 STRUCTURES | 分子名称: | Kappa-conotoxin PVIIA | 著者 | Scanlon, M.J, Naranjo, D, Thomas, L, Alewood, P.F, Lewis, R.J, Craik, D.J. | 登録日 | 1997-09-24 | 公開日 | 1998-10-14 | 最終更新日 | 2020-12-16 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure and proposed binding mechanism of a novel potassium channel toxin kappa-conotoxin PVIIA. Structure, 5, 1997
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1TTL
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![BU of 1ttl by Molmil](/molmil-images/mine/1ttl) | Omega-conotoxin GVIA, a N-type calcium channel blocker | 分子名称: | Omega-conotoxin GVIA | 著者 | Mould, J, Yasuda, T, Schroeder, C.I, Beedle, A.M, Doering, C.J, Zamponi, G.W, Adams, D.J, Lewis, R.J. | 登録日 | 2004-06-23 | 公開日 | 2004-07-13 | 最終更新日 | 2011-07-13 | 実験手法 | SOLUTION NMR | 主引用文献 | The alpha2delta auxiliary subunit reduces affinity of omega-conotoxins for recombinant N-type (Cav2.2) calcium channels J.Biol.Chem., 279, 2004
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1TR6
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![BU of 1tr6 by Molmil](/molmil-images/mine/1tr6) | NMR solution structure of omega-conotoxin [K10]GVIA, a cyclic cysteine knot peptide | 分子名称: | Omega-conotoxin GVIA | 著者 | Mould, J, Yasuda, T, Schroeder, C.I, Beedle, A.M, Doering, C.J, Zamponi, G.W, Adams, D.J, Lewis, R.J. | 登録日 | 2004-06-21 | 公開日 | 2004-07-13 | 最終更新日 | 2011-10-05 | 実験手法 | SOLUTION NMR | 主引用文献 | The alpha2delta auxiliary subunit reduces affinity of omega-conotoxins for recombinant N-type (Cav2.2) calcium channels J.Biol.Chem., 279, 2004
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1R9I
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![BU of 1r9i by Molmil](/molmil-images/mine/1r9i) | NMR Solution Structure of PIIIA toxin, NMR, 20 structures | 分子名称: | Mu-conotoxin PIIIA | 著者 | Nielsen, K.J, Watson, M, Adams, D.J, Hammarstrom, A.K, Gage, P.W, Hill, J.M, Craik, D.J, Thomas, L, Adams, D, Alewood, P.F, Lewis, R.J. | 登録日 | 2003-10-30 | 公開日 | 2003-11-18 | 最終更新日 | 2019-12-25 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of mu-conotoxin PIIIA, a preferential inhibitor of persistent tetrodotoxin-sensitive sodium channels J.Biol.Chem., 277, 2002
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1RMK
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![BU of 1rmk by Molmil](/molmil-images/mine/1rmk) | Solution structure of conotoxin MrVIB | 分子名称: | Mu-O-conotoxin MrVIB | 著者 | Daly, N.L, Ekberg, J.A, Thomas, L, Adams, D.J, Lewis, R.J, Craik, D.J. | 登録日 | 2003-11-28 | 公開日 | 2004-09-07 | 最終更新日 | 2022-03-02 | 実験手法 | SOLUTION NMR | 主引用文献 | Structures of muO-conotoxins from Conus marmoreus. Inhibitors of tetrodotoxin (TTX)-sensitive and TTX-resistant sodium channels in mammalian sensory neurons J.Biol.Chem., 279, 2004
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9BFL
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![BU of 9bfl by Molmil](/molmil-images/mine/9bfl) | |
7O0I
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![BU of 7o0i by Molmil](/molmil-images/mine/7o0i) | Vibrio vulnificus stressosome | 分子名称: | Anti-anti-sigma factor, RsbS, negative regulator of sigma-B | 著者 | Kaltwasser, S, Heinz, V, Madej, M.G, Pane-Farre, J, Ziegler, C. | 登録日 | 2021-03-26 | 公開日 | 2022-04-13 | 最終更新日 | 2023-11-01 | 実験手法 | ELECTRON MICROSCOPY (8.3 Å) | 主引用文献 | The Vibrio vulnificus stressosome is an oxygen-sensor involved in regulating iron metabolism Commun Biol, 2022
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8QHE
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![BU of 8qhe by Molmil](/molmil-images/mine/8qhe) | Crystal structure IR-09 | 分子名称: | 6-phosphogluconate dehydrogenase NADP-binding domain-containing protein, MAGNESIUM ION, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... | 著者 | Levy, C.W. | 登録日 | 2023-09-07 | 公開日 | 2023-10-11 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Biocatalysis in Drug Design: Engineered Reductive Aminases (RedAms) Are Used to Access Chiral Building Blocks with Multiple Stereocenters. J.Am.Chem.Soc., 145, 2023
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7Q5H
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![BU of 7q5h by Molmil](/molmil-images/mine/7q5h) | Keap1 compound complex | 分子名称: | (3S,5S,8R)-8-[[(2S)-1-ethanoylpyrrolidin-2-yl]carbonylamino]-N,N-dimethyl-3,7,11-tris(oxidanylidene)-10-oxa-3$l^{4}-thia-6-azabicyclo[10.4.0]hexadeca-1(16),12,14-triene-5-carboxamide, CHLORIDE ION, Kelch-like ECH-associated protein 1 | 著者 | Johansson, P. | 登録日 | 2021-11-03 | 公開日 | 2022-03-16 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.31 Å) | 主引用文献 | Importance of Binding Site Hydration and Flexibility Revealed When Optimizing a Macrocyclic Inhibitor of the Keap1-Nrf2 Protein-Protein Interaction. J.Med.Chem., 65, 2022
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7B3M
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![BU of 7b3m by Molmil](/molmil-images/mine/7b3m) | MEK1 in complex with compound 6 | 分子名称: | 1~{H}-indol-2-yl(pyridin-3-yl)methanone, Dual specificity mitogen-activated protein kinase kinase 1,Dual specificity mitogen-activated protein kinase kinase 1, MAGNESIUM ION, ... | 著者 | Kack, H, Oster, L. | 登録日 | 2020-12-01 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Fragment-Based Discovery of Novel Allosteric MEK1 Binders. Acs Med.Chem.Lett., 12, 2021
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7B7R
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![BU of 7b7r by Molmil](/molmil-images/mine/7b7r) | MEK1 in complex with compound 4 | 分子名称: | 2-[5-[ethyl(methyl)amino]imidazo[1,2-a]pyrimidin-7-yl]phenol, Dual specificity mitogen-activated protein kinase kinase 1,Dual specificity mitogen-activated protein kinase kinase 1, MAGNESIUM ION, ... | 著者 | Kack, H, Oster, L. | 登録日 | 2020-12-11 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Fragment-Based Discovery of Novel Allosteric MEK1 Binders. Acs Med.Chem.Lett., 12, 2021
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7B0U
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![BU of 7b0u by Molmil](/molmil-images/mine/7b0u) | Stressosome complex from Listeria innocua | 分子名称: | RsbR protein, RsbS protein | 著者 | Miksys, A, Fu, L, Madej, M.G, Ziegler, C. | 登録日 | 2020-11-22 | 公開日 | 2021-12-01 | 最終更新日 | 2022-07-20 | 実験手法 | ELECTRON MICROSCOPY (3.86 Å) | 主引用文献 | Molecular insights into intra-complex signal transmission during stressosome activation. Commun Biol, 5, 2022
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7B9L
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![BU of 7b9l by Molmil](/molmil-images/mine/7b9l) | MEK1 in complex with compound 23 | 分子名称: | Dual specificity mitogen-activated protein kinase kinase 1,Dual specificity mitogen-activated protein kinase kinase 1, GLYCEROL, MAGNESIUM ION, ... | 著者 | Kack, H, Oster, L. | 登録日 | 2020-12-14 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Fragment-Based Discovery of Novel Allosteric MEK1 Binders. Acs Med.Chem.Lett., 12, 2021
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7B94
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![BU of 7b94 by Molmil](/molmil-images/mine/7b94) | MEK1 in complex with compound 6 | 分子名称: | 2-(4-iodophenyl)-8~{H}-imidazo[1,2-c]pyrimidin-5-one, Dual specificity mitogen-activated protein kinase kinase 1,Dual specificity mitogen-activated protein kinase kinase 1, MAGNESIUM ION, ... | 著者 | Kack, H, Oster, L. | 登録日 | 2020-12-14 | 公開日 | 2021-03-03 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Fragment-Based Discovery of Novel Allosteric MEK1 Binders. Acs Med.Chem.Lett., 12, 2021
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5T90
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![BU of 5t90 by Molmil](/molmil-images/mine/5t90) | Structural mechanisms for alpha-conotoxin selectivity at the human alpha3beta4 nicotinic acetylcholine receptor | 分子名称: | Acetylcholine-binding protein, LsIA | 著者 | Abraham, N, Healy, M, Ragnarsson, L, Brust, A, Alewood, P, Lewis, R. | 登録日 | 2016-09-08 | 公開日 | 2017-04-12 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structural mechanisms for alpha-conotoxin activity at the human alpha 3 beta 4 nicotinic acetylcholine receptor. Sci Rep, 7, 2017
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6X8R
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![BU of 6x8r by Molmil](/molmil-images/mine/6x8r) | |
6KNO
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6KN3
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![BU of 6kn3 by Molmil](/molmil-images/mine/6kn3) | |
6KNP
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![BU of 6knp by Molmil](/molmil-images/mine/6knp) | |
6KN2
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![BU of 6kn2 by Molmil](/molmil-images/mine/6kn2) | |
6KMY
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![BU of 6kmy by Molmil](/molmil-images/mine/6kmy) | |