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8QRN
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BU of 8qrn by Molmil
mt-SSU in GTPBP8 knock-out cells, state 4
分子名称: 12S mitochondrial rRNA, 28S ribosomal protein S10, mitochondrial, ...
著者Valentin Gese, G, Cipullo, M, Rorbach, J, Hallberg, B.M.
登録日2023-10-09
公開日2024-06-26
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (2.98 Å)
主引用文献GTPBP8 plays a role in mitoribosome formation in human mitochondria.
Nat Commun, 15, 2024
8QU1
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BU of 8qu1 by Molmil
mt-LSU assembly intermediate in GTPBP8 knock-out cells, state 1
分子名称: 16S ribosomal RNA, 39S ribosomal protein L10, mitochondrial, ...
著者Valentin Gese, G, Cipullo, M, Rorbach, J, Hallberg, B.M.
登録日2023-10-13
公開日2024-06-26
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (2.74 Å)
主引用文献GTPBP8 plays a role in mitoribosome formation in human mitochondria.
Nat Commun, 15, 2024
8QRM
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BU of 8qrm by Molmil
mt-SSU assembly intermediate in GTPBP8 knock-out cells, state 3
分子名称: 12S mitochondrial rRNA, 28S ribosomal protein S10, mitochondrial, ...
著者Valentin Gese, G, Cipullo, M, Rorbach, J, Hallberg, B.M.
登録日2023-10-09
公開日2024-06-26
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (3.05 Å)
主引用文献GTPBP8 plays a role in mitoribosome formation in human mitochondria.
Nat Commun, 15, 2024
8QRK
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BU of 8qrk by Molmil
mt-SSU assembly intermediate in GTPBP8 knock-out cells, state 1
分子名称: 12S mitochondrial rRNA, 28S ribosomal protein S10, mitochondrial, ...
著者Valentin Gese, G, Cipullo, M, Rorbach, J, Hallberg, B.M.
登録日2023-10-09
公開日2024-06-26
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (6.69 Å)
主引用文献GTPBP8 plays a role in mitoribosome formation in human mitochondria.
Nat Commun, 15, 2024
8QRL
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BU of 8qrl by Molmil
mt-SSU assembly intermediate in GTPBP8 knock-out cells, state 2
分子名称: 12S mitochondrial rRNA, 12S rRNA N4-methylcytidine (m4C) methyltransferase, 28S ribosomal protein S10, ...
著者Valentin Gese, G, Cipullo, M, Rorbach, J, Hallberg, B.M.
登録日2023-10-09
公開日2024-06-26
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (3.34 Å)
主引用文献GTPBP8 plays a role in mitoribosome formation in human mitochondria.
Nat Commun, 15, 2024
8QU5
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BU of 8qu5 by Molmil
mt-LSU assembly intermediate in GTPBP8 knock-out cells, state 2
分子名称: 16S ribosomal RNA, 39S ribosomal protein L10, mitochondrial, ...
著者Valentin Gese, G, Cipullo, M, Rorbach, J, Hallberg, B.M.
登録日2023-10-13
公開日2024-06-26
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (2.42 Å)
主引用文献GTPBP8 plays a role in mitoribosome formation in human mitochondria.
Nat Commun, 15, 2024
1BFA
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BU of 1bfa by Molmil
RECOMBINANT BIFUNCTIONAL HAGEMAN FACTOR/AMYLASE INHIBITOR FROM MAIZE
分子名称: BIFUNCTIONAL AMYLASE/SERINE PROTEASE INHIBITOR
著者Behnke, C.A, Yee, V.C, Le Trong, I, Pedersen, L.C, Stenkamp, R.E, Kim, S.S, Reeck, G.R, Teller, D.C.
登録日1998-05-13
公開日1998-08-12
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural determinants of the bifunctional corn Hageman factor inhibitor: x-ray crystal structure at 1.95 A resolution.
Biochemistry, 37, 1998
2HWB
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BU of 2hwb by Molmil
A comparison of the anti-rhinoviral drug binding pocket in hrv14 and hrv1a
分子名称: 5-(3-(2,6-DICHLORO-4-(4,5-DIHYDRO-2-OXAZOLYL)PHENOXY)PROPYL)-3-METHYL ISOXAZOLE, HUMAN RHINOVIRUS 14 COAT PROTEIN (SUBUNIT VP1), HUMAN RHINOVIRUS 14 COAT PROTEIN (SUBUNIT VP2), ...
著者Kim, K.H, Rossmann, M.G.
登録日1994-01-25
公開日1994-11-01
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献A comparison of the anti-rhinoviral drug binding pocket in HRV14 and HRV1A.
J.Mol.Biol., 230, 1993
2HWC
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BU of 2hwc by Molmil
A COMPARISON OF THE ANTI-RHINOVIRAL DRUG BINDING POCKET IN HRV14 AND HRV1A
分子名称: 5-(5-(2,6-DICHLORO-4-(4,5-DIHYDRO-2-OXAZOLY)PHENOXY)PENTYL)-3-METHYL ISOXAZOLE, HUMAN RHINOVIRUS 14 COAT PROTEIN (SUBUNIT VP1), HUMAN RHINOVIRUS 14 COAT PROTEIN (SUBUNIT VP2), ...
著者Kim, K.H, Rossmann, M.G.
登録日1994-01-25
公開日1994-11-01
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献A comparison of the anti-rhinoviral drug binding pocket in HRV14 and HRV1A.
J.Mol.Biol., 230, 1993
2HWF
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BU of 2hwf by Molmil
A COMPARISON OF THE ANTI-RHINOVIRAL DRUG BINDING POCKET IN HRV14 AND HRV1A
分子名称: 3-METHOXY-6-[4-(3-METHYLPHENYL)-1-PIPERAZINYL]PYRIDAZINE, HUMAN RHINOVIRUS 1A COAT PROTEIN (SUBUNIT VP1), HUMAN RHINOVIRUS 1A COAT PROTEIN (SUBUNIT VP2), ...
著者Kim, K.H, Rossmann, M.G.
登録日1994-01-25
公開日1994-09-30
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献A comparison of the anti-rhinoviral drug binding pocket in HRV14 and HRV1A.
J.Mol.Biol., 230, 1993
2HWD
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BU of 2hwd by Molmil
A COMPARISON OF THE ANTI-RHINOVIRAL DRUG BINDING POCKET IN HRV14 AND HRV1A
分子名称: 5-(3-(2,6-DICHLORO-4-(4,5-DIHYDRO-2-OXAZOLYL)PHENOXY)PROPYL)-3-METHYL ISOXAZOLE, HUMAN RHINOVIRUS 1A COAT PROTEIN (SUBUNIT VP1), HUMAN RHINOVIRUS 1A COAT PROTEIN (SUBUNIT VP2), ...
著者Kim, K.H, Rossmann, M.G.
登録日1994-01-25
公開日1994-09-30
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献A comparison of the anti-rhinoviral drug binding pocket in HRV14 and HRV1A.
J.Mol.Biol., 230, 1993
2HWE
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BU of 2hwe by Molmil
A COMPARISON OF THE ANTI-RHINOVIRAL DRUG BINDING POCKET IN HRV14 AND HRV1A
分子名称: 5-(5-(2,6-DICHLORO-4-(4,5-DIHYDRO-2-OXAZOLY)PHENOXY)PENTYL)-3-METHYL ISOXAZOLE, HUMAN RHINOVIRUS 1A COAT PROTEIN (SUBUNIT VP1), HUMAN RHINOVIRUS 1A COAT PROTEIN (SUBUNIT VP2), ...
著者Kim, K.H, Rossmann, M.G.
登録日1994-01-25
公開日1994-09-30
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献A comparison of the anti-rhinoviral drug binding pocket in HRV14 and HRV1A.
J.Mol.Biol., 230, 1993
6LD2
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BU of 6ld2 by Molmil
Zika NS5 polymerase domain
分子名称: (1S,2S,4S,5R)-2,4-dimethoxy-5-thiophen-2-yl-cyclohexane-1-carboxylic acid, RNA-directed RNA polymerase NS5, ZINC ION
著者El Sahili, A, Lescar, J.
登録日2019-11-20
公開日2020-08-12
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Non-nucleoside Inhibitors of Zika Virus RNA-Dependent RNA Polymerase.
J.Virol., 94, 2020
6LD1
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BU of 6ld1 by Molmil
Zika NS5 polymerase domain
分子名称: 1,2-ETHANEDIOL, RNA-directed RNA polymerase NS5, ZINC ION
著者El Sahili, A, Lescar, J.
登録日2019-11-20
公開日2020-08-12
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Non-nucleoside Inhibitors of Zika Virus RNA-Dependent RNA Polymerase.
J.Virol., 94, 2020
6LD5
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BU of 6ld5 by Molmil
Zika NS5 polymerase domain
分子名称: 2,4-dimethoxy-5-thiophen-2-yl-benzoic acid, RNA-directed RNA polymerase NS5, ZINC ION, ...
著者El Sahili, A, Lescar, J.
登録日2019-11-20
公開日2020-08-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Non-nucleoside Inhibitors of Zika Virus RNA-Dependent RNA Polymerase.
J.Virol., 94, 2020
6LD4
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BU of 6ld4 by Molmil
Zika NS5 polymerase domain
分子名称: 2,4-dimethoxy-5-thiophen-2-yl-benzoic acid, 3-methoxybenzenesulfonamide, RNA-directed RNA polymerase NS5, ...
著者El Sahili, A, Lescar, J.
登録日2019-11-20
公開日2020-08-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Non-nucleoside Inhibitors of Zika Virus RNA-Dependent RNA Polymerase.
J.Virol., 94, 2020
6LD3
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BU of 6ld3 by Molmil
Zika NS5 polymerase domain
分子名称: 2,4-dimethoxy-5-thiophen-2-yl-benzoic acid, RNA-directed RNA polymerase NS5, ZINC ION, ...
著者El Sahili, A, Lescar, J.
登録日2019-11-20
公開日2020-08-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Non-nucleoside Inhibitors of Zika Virus RNA-Dependent RNA Polymerase.
J.Virol., 94, 2020
1S6P
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BU of 1s6p by Molmil
CRYSTAL STRUCTURE OF HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 REVERSE TRANSCRIPTASE (RT) IN COMPLEX WITH JANSSEN-R100943
分子名称: 1-(4-CYANO-PHENYL)-3-[2-(2,6-DICHLORO-PHENYL)-1-IMINO-ETHYL]-THIOUREA, MAGNESIUM ION, POL polyprotein [Contains: Reverse transcriptase]
著者Das, K, Arnold, E.
登録日2004-01-26
公開日2004-05-11
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Roles of Conformational and Positional Adaptability in Structure-Based Design of TMC125-R165335 (Etravirine) and Related Non-nucleoside Reverse Transcriptase Inhibitors That Are Highly Potent and Effective against Wild-Type and Drug-Resistant HIV-1 Variants
J.Med.Chem., 47, 2004
6N58
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BU of 6n58 by Molmil
Cryo-EM structure of Escherichia coli RNAP polymerase bound with TraR in conformation II
分子名称: CHAPSO, DNA-directed RNA polymerase subunit alpha, DNA-directed RNA polymerase subunit beta, ...
著者Chen, J, Chiu, C.E, Campbell, E.A, Darst, S.A.
登録日2018-11-21
公開日2020-02-26
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.78 Å)
主引用文献E. coliTraR allosterically regulates transcription initiation by altering RNA polymerase conformation.
Elife, 8, 2019
6N57
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BU of 6n57 by Molmil
Cryo-EM structure of Escherichia coli RNAP polymerase bound with TraR in conformation I
分子名称: CHAPSO, DNA-directed RNA polymerase subunit alpha, DNA-directed RNA polymerase subunit beta, ...
著者Chen, J, Chiu, C.E, Campbell, E.A, Darst, S.A.
登録日2018-11-21
公開日2020-02-26
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献E. coliTraR allosterically regulates transcription initiation by altering RNA polymerase conformation.
Elife, 8, 2019
5OOO
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BU of 5ooo by Molmil
Structure of the Rift Valley fever virus NSs protein core domain
分子名称: Non-structural protein NS-S
著者Barski, M.S, Potter, J.A, Schwarz-Linek, U.
登録日2017-08-08
公開日2017-08-16
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Rift Valley fever phlebovirus NSs protein core domain structure suggests molecular basis for nuclear filaments.
Elife, 6, 2017
4LV3
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BU of 4lv3 by Molmil
AmpC beta-lactamase in complex with (3,5-di-tert-butylphenyl) boronic acid
分子名称: (3,5-di-tert-butylphenyl)boronic acid, Beta-lactamase, PHOSPHATE ION
著者London, N, Eidam, O, Shoichet, B.K.
登録日2013-07-25
公開日2014-07-30
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献Covalent docking of large libraries for the discovery of chemical probes.
Nat.Chem.Biol., 10, 2014
4LV1
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BU of 4lv1 by Molmil
AmpC beta-lactamase in complex with [1-(3-chlorophenyl)-1H-pyrazol-4-yl] boronic acid
分子名称: Beta-lactamase, PHOSPHATE ION, [1-(3-chlorophenyl)-1H-pyrazol-4-yl]boronic acid
著者London, N, Eidam, O, Shoichet, B.K.
登録日2013-07-25
公開日2014-07-30
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.74 Å)
主引用文献Covalent docking of large libraries for the discovery of chemical probes.
Nat.Chem.Biol., 10, 2014
4M8T
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BU of 4m8t by Molmil
RSK2 T493M C-Terminal Kinase Domain in complex with 3-(3-(1H-pyrazol-4-yl)phenyl)-2-cyanoacrylamide
分子名称: (2E)-2-cyano-3-[3-(1H-pyrazol-4-yl)phenyl]prop-2-enamide, Ribosomal protein S6 kinase alpha-3, SODIUM ION
著者Miller, R.M, Taunton, J.
登録日2013-08-13
公開日2014-10-22
最終更新日2014-11-26
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Covalent docking of large libraries for the discovery of chemical probes.
Nat.Chem.Biol., 10, 2014
4LV0
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BU of 4lv0 by Molmil
AmpC beta-lactamase in complex with m-aminophenyl boronic acid
分子名称: Beta-lactamase, M-AMINOPHENYLBORONIC ACID, PHOSPHATE ION
著者London, N, Eidam, O, Shoichet, B.K.
登録日2013-07-25
公開日2014-07-30
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.652 Å)
主引用文献Covalent docking of large libraries for the discovery of chemical probes.
Nat.Chem.Biol., 10, 2014

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