5R4X
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![BU of 5r4x by Molmil](/molmil-images/mine/5r4x) | XChem fragment screen -- CRYSTAL STRUCTURE OF THE BROMODOMAIN OF THE HUMAN ATAD2 in complex with N13413a | 分子名称: | 1,2-ETHANEDIOL, 4-acetyl-N-ethylpiperazine-1-carboxamide, ATPase family AAA domain-containing protein 2, ... | 著者 | Talon, R, Krojer, T, Fairhead, M, Sethi, R, Bradley, A.R, Aimon, A, Collins, P, Brandao-Neto, J, Douangamath, A, Wright, N, MacLean, E, Zhang, R, Dias, A, Brennan, P.E, Bountra, C, Arrowsmith, C.H, Edwards, A, von Delft, F. | 登録日 | 2020-02-28 | 公開日 | 2020-05-13 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | XChem fragment screen To Be Published
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5R4Y
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![BU of 5r4y by Molmil](/molmil-images/mine/5r4y) | XChem fragment screen -- CRYSTAL STRUCTURE OF THE BROMODOMAIN OF THE HUMAN ATAD2 in complex with N13612a | 分子名称: | 1,2-ETHANEDIOL, ATPase family AAA domain-containing protein 2, SULFATE ION, ... | 著者 | Talon, R, Krojer, T, Fairhead, M, Sethi, R, Bradley, A.R, Aimon, A, Collins, P, Brandao-Neto, J, Douangamath, A, Wright, N, MacLean, E, Zhang, R, Dias, A, Brennan, P.E, Bountra, C, Arrowsmith, C.H, Edwards, A, von Delft, F. | 登録日 | 2020-02-28 | 公開日 | 2020-05-13 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.84 Å) | 主引用文献 | XChem fragment screen To Be Published
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5R4G
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![BU of 5r4g by Molmil](/molmil-images/mine/5r4g) | PanDDA analysis group deposition -- CRYSTAL STRUCTURE OF THE BROMODOMAIN OF HUMAN NUCLEOSOME-REMODELING FACTOR SUBUNIT BPTF in complex with FMOPL000621a | 分子名称: | 4-(1,2,3-thiadiazol-4-yl)phenyl ethylcarbamate, DIMETHYL SULFOXIDE, Nucleosome-remodeling factor subunit BPTF | 著者 | Talon, R, Krojer, T, Fairhead, M, Sethi, R, Bradley, A.R, Aimon, A, Collins, P, Brandao-Neto, J, Douangamath, A, Wright, N, MacLean, E, Renjie, Z, Dias, A, Brennan, P.E, Bountra, C, Arrowsmith, C.H, Edwards, A, von Delft, F. | 登録日 | 2020-02-24 | 公開日 | 2020-04-01 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.25 Å) | 主引用文献 | PanDDA analysis group deposition To Be Published
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5ROB
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![BU of 5rob by Molmil](/molmil-images/mine/5rob) | PanDDA analysis group deposition of ground-state model of SARS-CoV-2 helicase | 分子名称: | Helicase, PHOSPHATE ION, ZINC ION | 著者 | Newman, J.A, Yosaatmadja, Y, Douangamath, A, Aimon, A, Powell, A.J, Dias, A, Fearon, D, Dunnett, L, Brandao-Neto, J, Krojer, T, Skyner, R, Gorrie-Stone, T, Thompson, W, von Delft, F, Arrowsmith, C.H, Edwards, A, Bountra, C, Gileadi, O. | 登録日 | 2020-09-22 | 公開日 | 2021-03-10 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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2HW5
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![BU of 2hw5 by Molmil](/molmil-images/mine/2hw5) | The crystal structure of human enoyl-coenzyme A (CoA) hydratase short chain 1, ECHS1 | 分子名称: | CROTONYL COENZYME A, Enoyl-CoA hydratase, MAGNESIUM ION | 著者 | Turnbull, A.P, Salah, E, Niesen, F, Debreczeni, J, Ugochukwu, E, Pike, A.C.W, Kavanagh, K, Gileadi, O, Gorrec, F, Umeano, C, von Delft, F, Weigelt, J, Edwards, A, Arrowsmith, C, Sundstrom, M, Oppermann, U, Structural Genomics Consortium (SGC) | 登録日 | 2006-07-31 | 公開日 | 2006-08-22 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | The crystal structure of human enoyl-coenzyme A (CoA) hydratase short chain 1, ECHS1 To be Published
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5RJP
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![BU of 5rjp by Molmil](/molmil-images/mine/5rjp) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00024672 | 分子名称: | 4-bromo-1-(2-hydroxyethyl)pyridin-2(1H)-one, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.242 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RK3
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![BU of 5rk3 by Molmil](/molmil-images/mine/5rk3) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1501469697 | 分子名称: | 3-amino-1,6-dimethylpyridin-2(1H)-one, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.31 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RKN
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![BU of 5rkn by Molmil](/molmil-images/mine/5rkn) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z373768900 | 分子名称: | N-(1-ethyl-1H-pyrazol-4-yl)cyclobutanecarboxamide, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.23 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RJW
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![BU of 5rjw by Molmil](/molmil-images/mine/5rjw) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z256709556 | 分子名称: | 3-methylthiophene-2-carboxylic acid, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.514 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RKB
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![BU of 5rkb by Molmil](/molmil-images/mine/5rkb) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z2004563941 | 分子名称: | (1S)-1-(1-cyclopentyl-1H-pyrazol-4-yl)ethan-1-ol, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.279 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RKR
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![BU of 5rkr by Molmil](/molmil-images/mine/5rkr) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1432018343 | 分子名称: | (2S)-2-[(5-chloro-3-fluoropyridin-2-yl)amino]propan-1-ol, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.37 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RJO
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![BU of 5rjo by Molmil](/molmil-images/mine/5rjo) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00023827 | 分子名称: | 6-bromo-1,3-dihydro-2H-indol-2-one, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.22 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RK1
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![BU of 5rk1 by Molmil](/molmil-images/mine/5rk1) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1507502062 | 分子名称: | 6-methoxy-1,3,4,5-tetrahydro-2H-1-benzazepin-2-one, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.271 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RKI
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![BU of 5rki by Molmil](/molmil-images/mine/5rki) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z198194396 | 分子名称: | 4-(furan-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.268 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RJQ
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![BU of 5rjq by Molmil](/molmil-images/mine/5rjq) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00024665 | 分子名称: | 2-(4-bromanyl-2-methoxy-phenyl)ethanoic acid, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RK5
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![BU of 5rk5 by Molmil](/molmil-images/mine/5rk5) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z57478994 | 分子名称: | 5-(methoxymethyl)-1,3,4-thiadiazol-2-amine, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.243 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RKM
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![BU of 5rkm by Molmil](/molmil-images/mine/5rkm) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z2017168803 | 分子名称: | (2S)-2-[(3-fluoropyridin-2-yl)(methyl)amino]propan-1-ol, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.28 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RJI
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![BU of 5rji by Molmil](/molmil-images/mine/5rji) | PanDDA analysis group deposition of ground-state model of PHIP | 分子名称: | PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.24 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RJX
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![BU of 5rjx by Molmil](/molmil-images/mine/5rjx) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z285782452 | 分子名称: | N-methyl-2-(methylsulfonyl)aniline, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.291 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RKD
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![BU of 5rkd by Molmil](/molmil-images/mine/5rkd) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z2168282707 | 分子名称: | (6S)-1-methyl-4,5,6,7-tetrahydro-1H-benzotriazole-6-carboxylic acid, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.237 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RKU
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![BU of 5rku by Molmil](/molmil-images/mine/5rku) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z32367954 | 分子名称: | PH-interacting protein, ~{N}-cyclopropyl-1,3-benzodioxole-5-carboxamide | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RJK
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![BU of 5rjk by Molmil](/molmil-images/mine/5rjk) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00024661 | 分子名称: | 5-bromo-2-hydroxybenzonitrile, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.21 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RK0
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![BU of 5rk0 by Molmil](/molmil-images/mine/5rk0) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z30932204 | 分子名称: | N-[(4-sulfamoylphenyl)methyl]acetamide, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.24 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RKG
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![BU of 5rkg by Molmil](/molmil-images/mine/5rkg) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1124201124 | 分子名称: | PH-interacting protein, ethyl 1~{H}-pyrazole-4-carboxylate | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.282 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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5RKW
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![BU of 5rkw by Molmil](/molmil-images/mine/5rkw) | PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z27678561 | 分子名称: | N-(6-methoxy-1,3-benzothiazol-2-yl)cyclopropanecarboxamide, PH-interacting protein | 著者 | Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C. | 登録日 | 2020-06-02 | 公開日 | 2020-06-17 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.242 Å) | 主引用文献 | PanDDA analysis group deposition of ground-state model To Be Published
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