4K6F
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![BU of 4k6f by Molmil](/molmil-images/mine/4k6f) | |
4K6C
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![BU of 4k6c by Molmil](/molmil-images/mine/4k6c) | |
4OSE
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![BU of 4ose by Molmil](/molmil-images/mine/4ose) | |
4OTL
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![BU of 4otl by Molmil](/molmil-images/mine/4otl) | |
4MSO
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![BU of 4mso by Molmil](/molmil-images/mine/4mso) | |
4O5O
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![BU of 4o5o by Molmil](/molmil-images/mine/4o5o) | |
4O5H
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![BU of 4o5h by Molmil](/molmil-images/mine/4o5h) | |
4O5M
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![BU of 4o5m by Molmil](/molmil-images/mine/4o5m) | |
4OT8
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![BU of 4ot8 by Molmil](/molmil-images/mine/4ot8) | |
4N0W
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![BU of 4n0w by Molmil](/molmil-images/mine/4n0w) | |
4FUR
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![BU of 4fur by Molmil](/molmil-images/mine/4fur) | |
4DS3
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![BU of 4ds3 by Molmil](/molmil-images/mine/4ds3) | |
4F82
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![BU of 4f82 by Molmil](/molmil-images/mine/4f82) | |
4ECP
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![BU of 4ecp by Molmil](/molmil-images/mine/4ecp) | |
4EFZ
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![BU of 4efz by Molmil](/molmil-images/mine/4efz) | |
4GL8
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![BU of 4gl8 by Molmil](/molmil-images/mine/4gl8) | |
4HJH
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![BU of 4hjh by Molmil](/molmil-images/mine/4hjh) | |
4IJN
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![BU of 4ijn by Molmil](/molmil-images/mine/4ijn) | |
5UXW
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![BU of 5uxw by Molmil](/molmil-images/mine/5uxw) | |
3EK2
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![BU of 3ek2 by Molmil](/molmil-images/mine/3ek2) | |
3EJ2
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![BU of 3ej2 by Molmil](/molmil-images/mine/3ej2) | |
3EZO
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![BU of 3ezo by Molmil](/molmil-images/mine/3ezo) | |
7KP9
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![BU of 7kp9 by Molmil](/molmil-images/mine/7kp9) | asymmetric hTNF-alpha | 分子名称: | 1-{[2-(difluoromethoxy)phenyl]methyl}-2-methyl-6-[6-(piperazin-1-yl)pyridin-3-yl]-1H-benzimidazole, Tumor necrosis factor | 著者 | Arakaki, T.L, Abendroth, J, Fairman, J.W, Foley, A, Ceska, T. | 登録日 | 2020-11-10 | 公開日 | 2021-01-13 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Structural insights into the disruption of TNF-TNFR1 signalling by small molecules stabilising a distorted TNF. Nat Commun, 12, 2021
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4WMU
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![BU of 4wmu by Molmil](/molmil-images/mine/4wmu) | STRUCTURE OF MBP-MCL1 BOUND TO ligand 2 AT 1.55A | 分子名称: | 1,2-ETHANEDIOL, 6-chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1H-indole-2-carboxylic acid, FORMIC ACID, ... | 著者 | Clifton, M.C, Faiman, J.W. | 登録日 | 2014-10-09 | 公開日 | 2015-05-06 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | A Maltose-Binding Protein Fusion Construct Yields a Robust Crystallography Platform for MCL1. Plos One, 10, 2015
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7TI2
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![BU of 7ti2 by Molmil](/molmil-images/mine/7ti2) | Structure of KPC-2 bound to RPX-7063 at 1.75A | 分子名称: | 1,2-ETHANEDIOL, Carbapenem-hydrolyzing beta-lactamase KPC, {(3R,7S)-2-hydroxy-3-[2-(thiophen-2-yl)acetamido]-2,3,4,7-tetrahydro-1,2-oxaborepin-7-yl}acetic acid | 著者 | Clifton, M.C, Fairman, J.W, Edwards, T.E, Hecker, S.J. | 登録日 | 2022-01-12 | 公開日 | 2022-10-12 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Broad-spectrum cyclic boronate beta-lactamase inhibitors featuring an intramolecular prodrug for oral bioavailability. Bioorg.Med.Chem., 62, 2022
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