5FH8
| Crystal structure of the fifth bromodomain of human PB1 in complex with compound 28 | 分子名称: | 1,2-ETHANEDIOL, 6-chloranyl-3-(2-ethylbutyl)-4~{H}-pyrrolo[1,2-a]quinazolin-5-one, DIMETHYL SULFOXIDE, ... | 著者 | Tallant, C, Sutherell, C.L, Siejka, P, Sorrell, F.J, Krojer, T, Picaud, S, Fedorov, O, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Brennan, P.E, Ley, S.V, Knapp, S. | 登録日 | 2015-12-21 | 公開日 | 2016-06-01 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Identification and Development of 2,3-Dihydropyrrolo[1,2-a]quinazolin-5(1H)-one Inhibitors Targeting Bromodomains within the Switch/Sucrose Nonfermenting Complex. J.Med.Chem., 59, 2016
|
|
6N3F
| Structure of HIV Tat-specific factor 1 U2AF Homology Motif bound to SF3b1 ULM5 | 分子名称: | DI(HYDROXYETHYL)ETHER, GLYCEROL, HIV Tat-specific factor 1, ... | 著者 | Leach, J.R, Jenkins, J.L, Kielkopf, C.L. | 登録日 | 2018-11-15 | 公開日 | 2019-01-02 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.099 Å) | 主引用文献 | The pre-mRNA splicing and transcription factor Tat-SF1 is a functional partner of the spliceosome SF3b1 subunit via a U2AF homology motif interface. J. Biol. Chem., 294, 2019
|
|
6N2O
| |
6N3E
| Structure of HIV Tat-specific factor 1 U2AF Homology Motif bound to U2AF ligand motif 4 | 分子名称: | FORMIC ACID, GLYCEROL, HIV Tat-specific factor 1, ... | 著者 | Loerch, S, Jenkins, J.L, Kielkopf, C.L. | 登録日 | 2018-11-15 | 公開日 | 2019-01-02 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.893 Å) | 主引用文献 | The pre-mRNA splicing and transcription factor Tat-SF1 is a functional partner of the spliceosome SF3b1 subunit via a U2AF homology motif interface. J. Biol. Chem., 294, 2019
|
|
6MWX
| CryoEM structure of Chimeric Eastern Equine Encephalitis Virus with Fab of EEEV-69 Antibody | 分子名称: | E1, E2, EEEV-69 antibody heavy chain, ... | 著者 | Hasan, S.S, Sun, C, Kim, A.S, Watanabe, Y, Chen, C.L, Klose, T, Buda, G, Crispin, M, Diamond, M.S, Klimstra, W.B, Rossmann, M.G. | 登録日 | 2018-10-30 | 公開日 | 2018-12-19 | 最終更新日 | 2024-10-16 | 実験手法 | ELECTRON MICROSCOPY (8.2 Å) | 主引用文献 | Cryo-EM Structures of Eastern Equine Encephalitis Virus Reveal Mechanisms of Virus Disassembly and Antibody Neutralization. Cell Rep, 25, 2018
|
|
5G2X
| Structure a of Group II Intron Complexed with its Reverse Transcriptase | 分子名称: | 5'-R(*CP*AP*CP*AP*UP*CP*CP*AP*UP*AP*AP*CP)-3', GROUP II INTRON, GROUP II INTRON-ENCODED PROTEIN LTRA | 著者 | Qu, G, Kaushal, P.S, Wang, J, Shigematsu, H, Piazza, C.L, Agrawal, R.K, Belfort, M, Wang, H.W. | 登録日 | 2016-04-16 | 公開日 | 2016-05-11 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Structure of a Group II Intron in Complex with its Reverse Transcriptase. Nat.Struct.Mol.Biol., 23, 2016
|
|
5FBK
| Crystal structure of the extracellular domain of human calcium sensing receptor | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, BICARBONATE ION, CHLORIDE ION, ... | 著者 | Zhang, T, Zhang, C, Miller, C.L, Zou, J, Moremen, K.W, Brown, E.M, Yang, J.J, Hu, J. | 登録日 | 2015-12-14 | 公開日 | 2016-06-22 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural basis for regulation of human calcium-sensing receptor by magnesium ions and an unexpected tryptophan derivative co-agonist. Sci Adv, 2, 2016
|
|
6N3D
| Structure of HIV Tat-specific factor 1 U2AF Homology Motif (APO-State) | 分子名称: | CHLORIDE ION, DI(HYDROXYETHYL)ETHER, GLYCEROL, ... | 著者 | Loerch, S, Jenkins, J.L, Kielkopf, C.L. | 登録日 | 2018-11-15 | 公開日 | 2019-01-02 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.13 Å) | 主引用文献 | The pre-mRNA splicing and transcription factor Tat-SF1 is a functional partner of the spliceosome SF3b1 subunit via a U2AF homology motif interface. J. Biol. Chem., 294, 2019
|
|
1FNN
| CRYSTAL STRUCTURE OF CDC6P FROM PYROBACULUM AEROPHILUM | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, CELL DIVISION CONTROL PROTEIN 6, MAGNESIUM ION | 著者 | Liu, J, Smith, C.L, DeRyckere, D, DeAngelis, K, Martin, G.S, Berger, J.M. | 登録日 | 2000-08-22 | 公開日 | 2000-10-04 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure and function of Cdc6/Cdc18: implications for origin recognition and checkpoint control. Mol.Cell, 6, 2000
|
|
7WQA
| SARS-CoV-2 main protease in complex with Z-VAD-FMK | 分子名称: | 3C-like proteinase, Z-VAD(OMe)-FMK | 著者 | Wang, Y.C, Yang, C.S, Hou, M.H, Tsai, C.L, Chen, Y. | 登録日 | 2022-01-25 | 公開日 | 2023-03-22 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | SARS-CoV-2 main protease in complex with Z-VAD-FMK To Be Published
|
|
7WQ9
| Crystal structure of SARS-CoV-2 main protease in complex with Z-IETD-FMK | 分子名称: | 3C-like proteinase, Z-IETD-FMK | 著者 | Wang, Y.C, Yang, C.S, Hou, M.H, Tsai, C.L, Chen, Y. | 登録日 | 2022-01-25 | 公開日 | 2023-08-02 | 実験手法 | X-RAY DIFFRACTION (2.054 Å) | 主引用文献 | Crystal structure of SARS-CoV-2 main protease in complex with Z-IETD-FMK To Be Published
|
|
7WQ8
| Crystal structure of SARS-CoV-2 main protease in complex with Z-DEVD-FMK | 分子名称: | 3C-like proteinase, Z-DEVD-FMK | 著者 | Wang, Y.C, Yang, C.S, Hou, M.H, Tsai, C.L, Chen, Y. | 登録日 | 2022-01-24 | 公開日 | 2023-08-02 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal structure of SARS-CoV-2 main protease in complex with Z-DEVD-FMK To Be Published
|
|
7WQB
| SARS-CoV-2 main protease mutant (P168A) in complex with MG-132 | 分子名称: | 3C-like proteinase nsp5, MAGNESIUM ION, N-[(benzyloxy)carbonyl]-L-leucyl-N-[(2S)-1-hydroxy-4-methylpentan-2-yl]-L-leucinamide | 著者 | Wang, Y.C, Yang, C.S, Hou, M.H, Tsai, C.L, Chen, Y. | 登録日 | 2022-01-25 | 公開日 | 2023-08-02 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | SARS-CoV-2 main protease mutant (P168A) in complex with MG-132 To Be Published
|
|
7WQK
| wild-type SARS-CoV-2 main protease in complex with MG-132 | 分子名称: | 3C-like proteinase, MAGNESIUM ION, N-[(benzyloxy)carbonyl]-L-leucyl-N-[(2S)-1-hydroxy-4-methylpentan-2-yl]-L-leucinamide | 著者 | Wang, Y.C, Yang, C.S, Hou, M.H, Tsai, C.L, Chen, Y. | 登録日 | 2022-01-25 | 公開日 | 2023-08-02 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | wild-type SARS-CoV-2 main protease in complex with MG-132 To Be Published
|
|
6ND3
| |
5G2Y
| Structure a of Group II Intron Complexed with its Reverse Transcriptase | 分子名称: | GROUP II INTRON | 著者 | Qu, G, Kaushal, P.S, Wang, J, Shigematsu, H, Piazza, C.L, Agrawal, R.K, Belfort, M, Wang, H.W. | 登録日 | 2016-04-16 | 公開日 | 2016-05-04 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (4.5 Å) | 主引用文献 | Structure of a Group II Intron in Complex with its Reverse Transcriptase. Nat.Struct.Mol.Biol., 23, 2016
|
|
5FH7
| Crystal structure of the fifth bromodomain of human PB1 in complex with compound 18 | 分子名称: | 1,2-ETHANEDIOL, 6-chloranyl-3-[(dimethylamino)methyl]-4~{H}-pyrrolo[1,2-a]quinazolin-5-one, Protein polybromo-1 | 著者 | Tallant, C, Sutherell, C.L, Siejka, P, Sorrell, F.J, Krojer, T, Picaud, S, Fedorov, O, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Brennan, P.E, Ley, S.V, Knapp, S. | 登録日 | 2015-12-21 | 公開日 | 2016-06-01 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.47 Å) | 主引用文献 | Identification and Development of 2,3-Dihydropyrrolo[1,2-a]quinazolin-5(1H)-one Inhibitors Targeting Bromodomains within the Switch/Sucrose Nonfermenting Complex. J.Med.Chem., 59, 2016
|
|
5FAV
| E491Q mutant of choline TMA-lyase | 分子名称: | Choline trimethylamine-lyase, MALONATE ION, SODIUM ION | 著者 | Funk, M.A, Drennan, C.L. | 登録日 | 2015-12-12 | 公開日 | 2016-09-28 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Molecular Basis of C-N Bond Cleavage by the Glycyl Radical Enzyme Choline Trimethylamine-Lyase. Cell Chem Biol, 23, 2016
|
|
1ID3
| CRYSTAL STRUCTURE OF THE YEAST NUCLEOSOME CORE PARTICLE REVEALS FUNDAMENTAL DIFFERENCES IN INTER-NUCLEOSOME INTERACTIONS | 分子名称: | HISTONE H2A.1, HISTONE H2B.2, HISTONE H3, ... | 著者 | White, C.L, Suto, R.K, Luger, K. | 登録日 | 2001-04-03 | 公開日 | 2001-09-28 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structure of the yeast nucleosome core particle reveals fundamental changes in internucleosome interactions. EMBO J., 20, 2001
|
|
1G89
| |
1I7E
| C-Terminal Domain Of Mouse Brain Tubby Protein bound to Phosphatidylinositol 4,5-bis-phosphate | 分子名称: | L-ALPHA-GLYCEROPHOSPHO-D-MYO-INOSITOL-4,5-BIS-PHOSPHATE, TUBBY PROTEIN | 著者 | Santagata, S, Boggon, T.J, Baird, C.L, Shan, W.S, Shapiro, L. | 登録日 | 2001-03-08 | 公開日 | 2001-06-27 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | G-protein signaling through tubby proteins. Science, 292, 2001
|
|
1IW2
| X-ray structure of Human Complement Protein C8gamma at pH=7.O | 分子名称: | Complement Protein C8gamma | 著者 | Ortlund, E, Parker, C.L, Schreck, S.F, Ginell, S, Minor, W, Sodetz, J.M, Lebioda, L. | 登録日 | 2002-04-11 | 公開日 | 2002-06-12 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structure of human complement protein C8gamma at 1.2 A resolution reveals a lipocalin fold and a distinct ligand binding site. Biochemistry, 41, 2002
|
|
5T3W
| |
5T3T
| Ebola virus VP30 CTD bound to nucleoprotein | 分子名称: | Fusion protein of Nucleoprotein and Minor nucleoprotein VP30, SULFATE ION | 著者 | Kirchdoerfer, R.N, Moyer, C.L, Abelson, D.M, Saphire, E.O. | 登録日 | 2016-08-26 | 公開日 | 2016-09-28 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The Ebola Virus VP30-NP Interaction Is a Regulator of Viral RNA Synthesis. Plos Pathog., 12, 2016
|
|
5T7Z
| Monoclinic crystal form of the EpoB NRPS cyclization-docking bidomain from Sorangium cellulosum | 分子名称: | EpoB | 著者 | Dowling, D.P, Kung, Y, Croft, A.K, Taghizadeh, K, Kelly, W.L, Walsh, C.T, Drennan, C.L. | 登録日 | 2016-09-06 | 公開日 | 2016-11-09 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | Structural elements of an NRPS cyclization domain and its intermodule docking domain. Proc.Natl.Acad.Sci.USA, 113, 2016
|
|