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1CIZ
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BU of 1ciz by Molmil
X-RAY STRUCTURE OF HUMAN STROMELYSIN CATALYTIC DOMAIN COMPLEXES WITH NON-PEPTIDE INHIBITORS: IMPLICATION FOR INHIBITOR SELECTIVITY
分子名称: 3-(1H-INDOL-3-YL)-2-[4-(4-PHENYL-PIPERIDIN-1-YL)-BENZENESULFONYLAMINO]-PROPIONIC ACID, CALCIUM ION, PROTEIN (STROMELYSIN-1), ...
著者Pavlovsky, A.G, Williams, M.G, Ye, Q.-Z, Ortwine, D.F, Purchase II, C.F, White, A.D, Dhanaraj, V, Roth, B.D, Johnson, L.L, Hupe, D, Humblet, C, Blundell, T.L.
登録日1999-04-06
公開日1999-09-01
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.64 Å)
主引用文献X-ray structure of human stromelysin catalytic domain complexed with nonpeptide inhibitors: implications for inhibitor selectivity.
Protein Sci., 8, 1999
1CAQ
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BU of 1caq by Molmil
X-RAY STRUCTURE OF HUMAN STROMELYSIN CATALYTIC DOMAIN COMPLEXES WITH NON-PEPTIDE INHIBITORS: IMPLICATION FOR INHIBITOR SELECTIVITY
分子名称: 3-(1H-INDOL-3-YL)-2-[4-(4-PHENYL-PIPERIDIN-1-YL)-BENZENESULFONYLAMINO]-PROPIONIC ACID, CALCIUM ION, PROTEIN (STROMELYSIN-1), ...
著者Pavlovsky, A.G, Williams, M.G, Ye, Q.-Z, Ortwine, D.F, Purchase II, C.F, White, A.D, Dhanaraj, V, Roth, B.D, Johnson, L.L, Hupe, D, Humblet, C, Blundell, T.L.
登録日1999-02-23
公開日1999-07-07
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献X-ray structure of human stromelysin catalytic domain complexed with nonpeptide inhibitors: implications for inhibitor selectivity.
Protein Sci., 8, 1999
2P98
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BU of 2p98 by Molmil
E. coli methionine aminopeptidase monometalated with inhibitor YE7
分子名称: IMIDAZO[2,1-A]ISOQUINOLINE-2-CARBOHYDRAZIDE, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.
登録日2007-03-24
公開日2007-11-20
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Inhibition of Monometalated Methionine Aminopeptidase: Inhibitor Discovery and Crystallographic Analysis.
J.Med.Chem., 50, 2007
2Q94
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BU of 2q94 by Molmil
E. coli methionine aminopeptidase Mn-form with inhibitor A04
分子名称: 5-[2-(TRIFLUOROMETHOXY)PHENYL]-2-FUROIC ACID, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.-Z.
登録日2007-06-12
公開日2008-01-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.63 Å)
主引用文献Structural analysis of inhibition of E. coli methionine aminopeptidase: implication of loop flexibility in selective inhibition of bacterial enzymes.
Bmc Struct.Biol., 7, 2007
2Q92
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BU of 2q92 by Molmil
E. coli methionine aminopeptidase Mn-form with inhibitor B23
分子名称: 5-(2-NITROPHENYL)-2-FUROIC ACID, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.-Z.
登録日2007-06-12
公開日2008-01-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural analysis of inhibition of E. coli methionine aminopeptidase: implication of loop flexibility in selective inhibition of bacterial enzymes.
Bmc Struct.Biol., 7, 2007
2P9A
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BU of 2p9a by Molmil
E. coli methionine aminopeptidase dimetalated with inhibitor YE6
分子名称: 5-(2-chlorophenyl)furan-2-carbohydrazide, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.
登録日2007-03-24
公開日2007-11-20
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Inhibition of Monometalated Methionine Aminopeptidase: Inhibitor Discovery and Crystallographic Analysis.
J.Med.Chem., 50, 2007
2Q96
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BU of 2q96 by Molmil
E. coli methionine aminopeptidase Mn-form with inhibitor A18
分子名称: 5-(2-CHLOROBENZYL)-2-FUROIC ACID, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.-Z.
登録日2007-06-12
公開日2008-01-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural analysis of inhibition of E. coli methionine aminopeptidase: implication of loop flexibility in selective inhibition of bacterial enzymes.
Bmc Struct.Biol., 7, 2007
2Q95
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BU of 2q95 by Molmil
E. coli methionine aminopeptidase Mn-form with inhibitor A05
分子名称: 5-(2-CHLORO-4-NITROPHENYL)-2-FUROIC ACID, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.-Z.
登録日2007-06-12
公開日2008-01-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural analysis of inhibition of E. coli methionine aminopeptidase: implication of loop flexibility in selective inhibition of bacterial enzymes.
Bmc Struct.Biol., 7, 2007
2Q93
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BU of 2q93 by Molmil
E. coli methionine aminopeptidase Mn-form with inhibitor B21
分子名称: 5-(2-METHOXYPHENYL)-2-FUROIC ACID, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.-Z.
登録日2007-06-12
公開日2008-01-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural analysis of inhibition of E. coli methionine aminopeptidase: implication of loop flexibility in selective inhibition of bacterial enzymes.
Bmc Struct.Biol., 7, 2007
2P99
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BU of 2p99 by Molmil
E. coli methionine aminopeptidase monometalated with inhibitor YE6
分子名称: 5-(2-chlorophenyl)furan-2-carbohydrazide, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Ye, Q.
登録日2007-03-24
公開日2007-11-20
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Inhibition of Monometalated Methionine Aminopeptidase: Inhibitor Discovery and Crystallographic Analysis.
J.Med.Chem., 50, 2007
2EVC
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BU of 2evc by Molmil
Crystal structure of E. Coli. methionine amino peptidase in complex with 5-(2-(trifluoromethyl)phenyl)furan-2-carboxylic acid
分子名称: 5-[2-(TRIFLUOROMETHYL)PHENYL]-2-FUROIC ACID, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Huang, W.-J.
登録日2005-10-31
公開日2006-03-28
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural analysis of metalloform-selective inhibition of methionine aminopeptidase.
Acta Crystallogr.,Sect.D, 62, 2006
2EVO
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BU of 2evo by Molmil
crystal structure of methionine amino peptidase in complex with N-cyclopentyl-N-(thiazol-2-yl)oxalamide
分子名称: COBALT (II) ION, Methionine aminopeptidase, N1-CYCLOPENTYL-N2-(THIAZOL-2-YL)OXALAMIDE
著者Huang, W.-J.
登録日2005-10-31
公開日2006-03-28
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural analysis of metalloform-selective inhibition of methionine aminopeptidase.
Acta Crystallogr.,Sect.D, 62, 2006
2EVM
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BU of 2evm by Molmil
crystal structure of methionine aminopeptidase in complex with 5-(2,5-dichlorophenyl)furan-2-carboxylic acid
分子名称: 5-(2,5-DICHLOROPHENYL)-2-FUROIC ACID, MANGANESE (II) ION, Methionine aminopeptidase, ...
著者Huang, W.-J.
登録日2005-10-31
公開日2006-03-28
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural analysis of metalloform-selective inhibition of methionine aminopeptidase.
Acta Crystallogr.,Sect.D, 62, 2006
1ZVX
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BU of 1zvx by Molmil
Crystal structure of the complex between MMP-8 and a phosphonate inhibitor (R-enantiomer)
分子名称: (1R)-1-{[(4'-METHOXY-1,1'-BIPHENYL-4-YL)SULFONYL]AMINO}-2-METHYLPROPYLPHOSPHONIC ACID, CALCIUM ION, Neutrophil collagenase, ...
著者Pochetti, G, Gavuzzo, E, Campestre, C, Agamennone, M, Tortorella, P, Consalvi, V, Gallina, C, Hiller, O, Tschesche, H, Tucker, P.A, Mazza, F.
登録日2005-06-03
公開日2006-05-16
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献Structural insight into the stereoselective inhibition of MMP-8 by enantiomeric sulfonamide phosphonates.
J.Med.Chem., 49, 2006
1ZS0
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BU of 1zs0 by Molmil
Crystal structure of the complex between MMP-8 and a phosphonate inhibitor (S-enantiomer)
分子名称: (1S)-1-{[(4'-METHOXY-1,1'-BIPHENYL-4-YL)SULFONYL]AMINO}-2-METHYLPROPYLPHOSPHONIC ACID, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
著者Pochetti, G, Gavuzzo, E, Campestre, C, Agamennone, M, Tortorella, P, Consalvi, V, Gallina, C, Hiller, O, Tschesche, H, Tucker, P.A, Mazza, F.
登録日2005-05-23
公開日2006-05-02
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Structural insight into the stereoselective inhibition of MMP-8 by enantiomeric sulfonamide phosphonates.
J.Med.Chem., 49, 2006
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