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6U7R
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BU of 6u7r by Molmil
NMR solution structure of SFTI1 based KLK7 protease inhibitor
分子名称: GLY-LYS-CYS-LEU-PHE-SER-ASN-PRO-PRO-ILE-CYS-PHE-PRO-ASN inhibitor
著者White, A.M, Harvey, P.J, Durek, T, Craik, D.J.
登録日2019-09-03
公開日2020-04-22
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Application and Structural Analysis of Triazole-Bridged Disulfide Mimetics in Cyclic Peptides.
Angew.Chem.Int.Ed.Engl., 59, 2020
6VY8
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BU of 6vy8 by Molmil
NMR solution structure of a triazole bridged trypsin inhibitor based on the framework of SFTI-1
分子名称: Trypsin inhibitor GLY-ARG-RVJ-THR-LYS-SER-ILE-PRO-PRO-ILE-2AG-PHE-PRO-ASP
著者White, A.M, Harvey, P.J, Durek, T, Craik, D.J.
登録日2020-02-25
公開日2020-07-01
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Application and Structural Analysis of Triazole-Bridged Disulfide Mimetics in Cyclic Peptides.
Angew.Chem.Int.Ed.Engl., 2020
6VXY
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BU of 6vxy by Molmil
Triazole bridged SFTI1 inhibitor in complex with beta-trypsin
分子名称: 1-methyl-1H-1,2,3-triazole, CALCIUM ION, Cationic trypsin, ...
著者White, A.M, King, G.J, Durek, T, Craik, D.J.
登録日2020-02-25
公開日2020-07-01
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.398 Å)
主引用文献Application and Structural Analysis of Triazole-Bridged Disulfide Mimetics in Cyclic Peptides.
Angew.Chem.Int.Ed.Engl., 2020
2MG9
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BU of 2mg9 by Molmil
Truncated EGF-A
分子名称: CALCIUM ION, Low-density lipoprotein receptor
著者Schroeder, C.I, Rosengren, K.
登録日2013-10-30
公開日2014-04-02
実験手法SOLUTION NMR
主引用文献Design and Synthesis of Truncated EGF-A Peptides that Restore LDL-R Recycling in the Presence of PCSK9 In Vitro.
Chem.Biol., 21, 2014
6BVH
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BU of 6bvh by Molmil
Trypsin complexed with a modified sunflower trypsin inhibitor, SFTI-TCTR(N12,N14)
分子名称: CALCIUM ION, Cationic trypsin, GLYCEROL, ...
著者Riley, B.T, Chen, X.
登録日2017-12-13
公開日2018-12-19
最終更新日2019-01-30
実験手法X-RAY DIFFRACTION (1.927 Å)
主引用文献Potent, multi-target serine protease inhibition achieved by a simplified beta-sheet motif.
PLoS ONE, 14, 2019
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件を2024-06-12に公開中

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