6P2B
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![BU of 6p2b by Molmil](/molmil-images/mine/6p2b) | Tethered PXR-LBD/SRC-1p bound to Garcinoic Acid | 分子名称: | (2Z,6E,10E)-13-[(2R)-6-hydroxy-2,8-dimethyl-3,4-dihydro-2H-1-benzopyran-2-yl]-2,6,10-trimethyltrideca-2,6,10-trienoic acid, DIMETHYL SULFOXIDE, Nuclear receptor subfamily 1 group I member 2 | 著者 | Walton, W.G, Pellock, S.J, Redinbo, M.R. | 登録日 | 2019-05-21 | 公開日 | 2020-04-01 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Garcinoic Acid Is a Natural and Selective Agonist of Pregnane X Receptor. J.Med.Chem., 63, 2020
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6ECA
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![BU of 6eca by Molmil](/molmil-images/mine/6eca) | Lactobacillus rhamnosus Beta-glucuronidase | 分子名称: | Beta-glucuronidase, CHLORIDE ION, GLYCEROL | 著者 | Biernat, K.A, Pellock, S.J, Bhatt, A.P, Bivins, M.M, Walton, W.G, Tran, B.N.T, Wei, L, Snider, M.C, Cesmat, A.P, Tripathy, A, Erie, D.A, Redinbo, M.R.R. | 登録日 | 2018-08-07 | 公開日 | 2019-02-13 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.853 Å) | 主引用文献 | Structure, function, and inhibition of drug reactivating human gut microbial beta-glucuronidases. Sci Rep, 9, 2019
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6AYI
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![BU of 6ayi by Molmil](/molmil-images/mine/6ayi) | Escherichia coli GusR | 分子名称: | 4-nitrophenyl beta-D-glucopyranosiduronic acid, HTH-type transcriptional regulator UidR | 著者 | Little, M.S, Pellock, S.J. | 登録日 | 2017-09-08 | 公開日 | 2017-12-20 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.09 Å) | 主引用文献 | Structural basis for the regulation of beta-glucuronidase expression by human gut Enterobacteriaceae. Proc. Natl. Acad. Sci. U.S.A., 115, 2018
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6AYH
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![BU of 6ayh by Molmil](/molmil-images/mine/6ayh) | Salmonella enterica GusR | 分子名称: | 4-nitrophenyl beta-D-glucopyranosiduronic acid, GLYCEROL, TetR family transcriptional regulator | 著者 | Little, M.S, Pellock, S.J. | 登録日 | 2017-09-08 | 公開日 | 2017-12-20 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structural basis for the regulation of beta-glucuronidase expression by human gut Enterobacteriaceae. Proc. Natl. Acad. Sci. U.S.A., 115, 2018
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5CZK
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![BU of 5czk by Molmil](/molmil-images/mine/5czk) | Structure of E. coli beta-glucuronidase bound with a novel, potent inhibitor 1-((6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl)-1-(2-hydroxyethyl)-3-(4-hydroxyphenyl)thiourea | 分子名称: | 1-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-(2-hydroxyethyl)-3-(4-hydroxyphenyl)thiourea, Beta-glucuronidase | 著者 | Roberts, A.R, Wallace, B.R, Redinbo, M.R. | 登録日 | 2015-07-31 | 公開日 | 2015-10-14 | 最終更新日 | 2019-12-04 | 実験手法 | X-RAY DIFFRACTION (2.39 Å) | 主引用文献 | Structure and Inhibition of Microbiome beta-Glucuronidases Essential to the Alleviation of Cancer Drug Toxicity. Chem.Biol., 22, 2015
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8U5A
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![BU of 8u5a by Molmil](/molmil-images/mine/8u5a) | Improving protein expression, stability, and function with ProteinMPNN | 分子名称: | Designed myoglobin, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Kalvet, I, Bera, A.K, Baker, D. | 登録日 | 2023-09-12 | 公開日 | 2024-01-17 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Improving Protein Expression, Stability, and Function with ProteinMPNN. J.Am.Chem.Soc., 146, 2024
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8SK7
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![BU of 8sk7 by Molmil](/molmil-images/mine/8sk7) | Cryo-EM structure of designed Influenza HA binder, HA_20, bound to Influenza HA (Strain: Iowa43) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, HA_20 minibinder (RFdiffusion-designed), ... | 著者 | Borst, A.J, Bennett, N.R. | 登録日 | 2023-04-18 | 公開日 | 2023-06-14 | 最終更新日 | 2023-09-13 | 実験手法 | ELECTRON MICROSCOPY (2.93 Å) | 主引用文献 | De novo design of protein structure and function with RFdiffusion. Nature, 620, 2023
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4JKL
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![BU of 4jkl by Molmil](/molmil-images/mine/4jkl) | |
4JKK
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![BU of 4jkk by Molmil](/molmil-images/mine/4jkk) | |
4JKM
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![BU of 4jkm by Molmil](/molmil-images/mine/4jkm) | |
7M5T
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![BU of 7m5t by Molmil](/molmil-images/mine/7m5t) | |
5UJ6
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![BU of 5uj6 by Molmil](/molmil-images/mine/5uj6) | |
6CXS
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![BU of 6cxs by Molmil](/molmil-images/mine/6cxs) | Crystal Structure of Clostridium perfringens beta-glucuronidase bound with a novel, potent inhibitor 4-(8-(piperazin-1-yl)-1,2,3,4-tetrahydro-[1,2,3]triazino[4',5':4,5]thieno[2,3-c]isoquinolin-5-yl)morpholine | 分子名称: | 4-(8-(piperazin-1-yl)-1,2,3,4-tetrahydro-[1,2,3]triazino[4',5':4,5]thieno[2,3-c]isoquinolin-5-yl)morpholine, Beta-glucuronidase, Maltose/maltodextrin-binding periplasmic protein | 著者 | Wallace, B.D, Redinbo, M.R. | 登録日 | 2018-04-04 | 公開日 | 2019-04-17 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Targeted inhibition of gut bacterial beta-glucuronidase activity enhances anticancer drug efficacy. Proc.Natl.Acad.Sci.USA, 2020
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6ED1
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![BU of 6ed1 by Molmil](/molmil-images/mine/6ed1) | Bacteroides dorei Beta-glucuronidase | 分子名称: | Glycosyl hydrolase family 2, sugar binding domain protein, SODIUM ION | 著者 | Biernat, K.A, Redinbo, M.R. | 登録日 | 2018-08-08 | 公開日 | 2019-02-13 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Structure, function, and inhibition of drug reactivating human gut microbial beta-glucuronidases. Sci Rep, 9, 2019
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6EC6
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![BU of 6ec6 by Molmil](/molmil-images/mine/6ec6) | |
6AZH
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![BU of 6azh by Molmil](/molmil-images/mine/6azh) | |