8J3T
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![BU of 8j3t by Molmil](/molmil-images/mine/8j3t) | Complex structure of human cytomegalovirus protease and a non-covalent small-molecule ligand | 分子名称: | (4R)-1-[1-[(S)-[1-cyclopentyl-3-(2-methylphenyl)pyrazol-4-yl]-(4-methylphenyl)methyl]-2-oxidanylidene-pyridin-3-yl]-3-methyl-2-oxidanylidene-N-(3-oxidanylidene-2-azabicyclo[2.2.2]octan-4-yl)imidazolidine-4-carboxamide, Assemblin | 著者 | Yoshida, S, Sako, Y, Nikaido, E, Ueda, T, Kozono, I, Ichihashi, Y, Nakahashi, A, Onishi, M, Yamatsu, Y, Kato, T, Nishikawa, J, Tachibana, Y. | 登録日 | 2023-04-18 | 公開日 | 2023-11-08 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Peptide-to-Small Molecule: Discovery of Non-Covalent, Active-Site Inhibitors of beta-Herpesvirus Proteases. Acs Med.Chem.Lett., 14, 2023
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8HH2
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![BU of 8hh2 by Molmil](/molmil-images/mine/8hh2) | F1 domain of FoF1-ATPase from Bacillus PS3,post-hyd,highATP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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8HHC
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![BU of 8hhc by Molmil](/molmil-images/mine/8hhc) | F1 domain of FoF1-ATPase from Bacillus PS3,post-hyd',lowATP | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ATP synthase subunit alpha, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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8HHB
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![BU of 8hhb by Molmil](/molmil-images/mine/8hhb) | F1 domain of FoF1-ATPase from Bacillus PS3,step waiting,lowATP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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8HHA
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![BU of 8hha by Molmil](/molmil-images/mine/8hha) | F1 domain of FoF1-ATPase from Bacillus PS3,120 degrees,lowATP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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8HH1
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![BU of 8hh1 by Molmil](/molmil-images/mine/8hh1) | FoF1-ATPase from Bacillus PS3, 81 degrees, highATP | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ATP synthase subunit alpha, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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8HH4
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![BU of 8hh4 by Molmil](/molmil-images/mine/8hh4) | F1 domain of FoF1-ATPase from Bacillus PS3,101 degrees, highATP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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8HH8
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![BU of 8hh8 by Molmil](/molmil-images/mine/8hh8) | F1 domain of FoF1-ATPase from Bacillus PS3,post-hyd,lowATP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-26 | 実験手法 | ELECTRON MICROSCOPY (2.8 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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8HH9
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![BU of 8hh9 by Molmil](/molmil-images/mine/8hh9) | F1 domain of FoF1-ATPase from Bacillus PS3, 90 degrees, low ATP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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8HH6
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![BU of 8hh6 by Molmil](/molmil-images/mine/8hh6) | F1 domain of FoF1-ATPase from Bacillus PS3,step waiting,highATP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-26 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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8HH3
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![BU of 8hh3 by Molmil](/molmil-images/mine/8hh3) | F1 domain of FoF1-ATPase from Bacillus PS3,90 degrees,highATP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-19 | 実験手法 | ELECTRON MICROSCOPY (4.3 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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8HH7
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![BU of 8hh7 by Molmil](/molmil-images/mine/8hh7) | F1 domain of FoF1-ATPase from Bacillus PS3, 81 degrees, lowATP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-26 | 実験手法 | ELECTRON MICROSCOPY (2.5 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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8HH5
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![BU of 8hh5 by Molmil](/molmil-images/mine/8hh5) | F1 domain of FoF1-ATPase from Bacillus PS3,120 degrees,highATP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ATP synthase gamma chain, ... | 著者 | Nakano, A, Kishikawa, J, Mitsuoka, K, Yokoyama, K. | 登録日 | 2022-11-16 | 公開日 | 2023-07-26 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Rotation mechanism of ATP synthases driven by ATP hydrolysis To Be Published
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7EHZ
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![BU of 7ehz by Molmil](/molmil-images/mine/7ehz) | Structure of human NNMT in complex with macrocyclic peptide 2 | 分子名称: | Nicotinamide N-methyltransferase, macrocyclic peptide 2 | 著者 | Hayashi, K, Mikamiyama, H, Uehara, S, Yamamoto, S, Cary, D, Nishikawa, J, Ueda, T, Ozasa, H, Mihara, K, Yoshimura, N, Kawai, T, Ono, T, Yamamoto, S, Fumoto, M. | 登録日 | 2021-03-30 | 公開日 | 2021-12-15 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Macrocyclic Peptides as a Novel Class of NNMT Inhibitors: A SAR Study Aimed at Inhibitory Activity in the Cell. Acs Med.Chem.Lett., 12, 2021
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7EGU
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![BU of 7egu by Molmil](/molmil-images/mine/7egu) | Structure of human NNMT in complex with macrocyclic peptide X | 分子名称: | Nicotinamide N-methyltransferase, macrocyclic peptide X | 著者 | Hayashi, K, Mikamiyama, H, Uehara, S, Yamamoto, S, Cary, D, Nishikawa, J, Ueda, T, Ozasa, H, Mihara, K, Yoshimura, N, Kawai, T, Ono, T, Yamamoto, S, Fumoto, M. | 登録日 | 2021-03-26 | 公開日 | 2021-12-15 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Macrocyclic Peptides as a Novel Class of NNMT Inhibitors: A SAR Study Aimed at Inhibitory Activity in the Cell. Acs Med.Chem.Lett., 12, 2021
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7EI2
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![BU of 7ei2 by Molmil](/molmil-images/mine/7ei2) | Structure of human NNMT in complex with macrocyclic peptide 8 | 分子名称: | Nicotinamide N-methyltransferase, macrocyclic peptide 8 | 著者 | Hayashi, K, Mikamiyama, H, Uehara, S, Yamamoto, S, Cary, D, Nishikawa, J, Ueda, T, Ozasa, H, Mihara, K, Yoshimura, N, Kawai, T, Ono, T, Yamamoto, S, Fumoto, M. | 登録日 | 2021-03-30 | 公開日 | 2022-03-30 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | Macrocyclic Peptides as a Novel Class of NNMT Inhibitors: A SAR Study Aimed at Inhibitory Activity in the Cell. Acs Med.Chem.Lett., 12, 2021
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3WJ4
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![BU of 3wj4 by Molmil](/molmil-images/mine/3wj4) | Crystal structure of PPARgamma ligand binding domain in complex with tributyltin | 分子名称: | Peroxisome proliferator-activated receptor gamma, tributylstannanyl | 著者 | Harada, S, Hiromori, Y, Fukakusa, S, Kawahara, K, Nakamura, S, Noda, M, Uchiyama, S, Fukui, K, Nishikawa, J, Nagase, H, Kobayashi, Y, Ohkubo, T, Yoshida, T, Nakanishi, T. | 登録日 | 2013-10-04 | 公開日 | 2014-10-15 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Structural basis for PPARgamma transactivation by endocrine disrupting organotin compounds To be Published
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3WJ5
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![BU of 3wj5 by Molmil](/molmil-images/mine/3wj5) | Crystal structure of PPARgamma ligand binding domain in complex with triphenyltin | 分子名称: | Peroxisome proliferator-activated receptor gamma, triphenylstannanyl | 著者 | Harada, S, Hiromori, Y, Fukakusa, S, Kawahara, K, Nakamura, S, Noda, M, Uchiyama, S, Fukui, K, Nishikawa, J, Nagase, H, Kobayashi, Y, Ohkubo, T, Yoshida, T, Nakanishi, T. | 登録日 | 2013-10-04 | 公開日 | 2014-10-15 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | Structural basis for PPARgamma transactivation by endocrine disrupting organotin compounds To be Published
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7XK7
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![BU of 7xk7 by Molmil](/molmil-images/mine/7xk7) | Cryo-EM structure of Na+-pumping NADH-ubiquinone oxidoreductase from Vibrio cholerae, with korormicin | 分子名称: | 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, CALCIUM ION, DODECYL-BETA-D-MALTOSIDE, ... | 著者 | Kishikawa, J, Ishikawa, M, Masuya, T, Murai, M, Barquera, B, Miyoshi, H. | 登録日 | 2022-04-19 | 公開日 | 2022-07-20 | 最終更新日 | 2022-08-10 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Cryo-EM structures of Na + -pumping NADH-ubiquinone oxidoreductase from Vibrio cholerae. Nat Commun, 13, 2022
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7XK4
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![BU of 7xk4 by Molmil](/molmil-images/mine/7xk4) | Cryo-EM structure of Na+-pumping NADH-ubiquinone oxidoreductase from Vibrio cholerae, state 2 | 分子名称: | 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, CALCIUM ION, DODECYL-BETA-D-MALTOSIDE, ... | 著者 | Kishikawa, J, Ishikawa, M, Masuya, T, Murai, M, Barquera, B, Miyoshi, H. | 登録日 | 2022-04-19 | 公開日 | 2022-07-20 | 最終更新日 | 2022-08-10 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Cryo-EM structures of Na + -pumping NADH-ubiquinone oxidoreductase from Vibrio cholerae. Nat Commun, 13, 2022
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7XK5
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![BU of 7xk5 by Molmil](/molmil-images/mine/7xk5) | Cryo-EM structure of Na+-pumping NADH-ubiquinone oxidoreductase from Vibrio cholerae, state 3 | 分子名称: | 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, CALCIUM ION, DODECYL-BETA-D-MALTOSIDE, ... | 著者 | Kishikawa, J, Ishikawa, M, Masuya, T, Murai, M, Barquera, B, Miyoshi, H. | 登録日 | 2022-04-19 | 公開日 | 2022-07-20 | 最終更新日 | 2022-08-10 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Cryo-EM structures of Na + -pumping NADH-ubiquinone oxidoreductase from Vibrio cholerae. Nat Commun, 13, 2022
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7XK6
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![BU of 7xk6 by Molmil](/molmil-images/mine/7xk6) | Cryo-EM structure of Na+-pumping NADH-ubiquinone oxidoreductase from Vibrio cholerae, with aurachin D-42 | 分子名称: | 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, Aurachin D, CALCIUM ION, ... | 著者 | Kishikawa, J, Ishikawa, M, Masuya, T, Murai, M, Barquera, B, Miyoshi, H. | 登録日 | 2022-04-19 | 公開日 | 2022-07-20 | 最終更新日 | 2022-08-10 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Cryo-EM structures of Na + -pumping NADH-ubiquinone oxidoreductase from Vibrio cholerae. Nat Commun, 13, 2022
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7XK3
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![BU of 7xk3 by Molmil](/molmil-images/mine/7xk3) | Cryo-EM structure of Na+-pumping NADH-ubiquinone oxidoreductase from Vibrio cholerae, state 1 | 分子名称: | 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, CALCIUM ION, DODECYL-BETA-D-MALTOSIDE, ... | 著者 | Kishikawa, J, Ishikawa, M, Masuya, T, Murai, M, Barquera, B, Miyoshi, H. | 登録日 | 2022-04-19 | 公開日 | 2022-07-20 | 最終更新日 | 2022-08-10 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Cryo-EM structures of Na + -pumping NADH-ubiquinone oxidoreductase from Vibrio cholerae. Nat Commun, 13, 2022
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8JJE
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![BU of 8jje by Molmil](/molmil-images/mine/8jje) | RBD of SARS-CoV2 spike protein with ACE2 decoy | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Angiotensin-converting enzyme 2, ... | 著者 | Kishikawa, J, Hirose, M, Kato, T, Okamoto, T. | 登録日 | 2023-05-30 | 公開日 | 2023-12-27 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | An inhaled ACE2 decoy confers protection against SARS-CoV-2 infection in preclinical models. Sci Transl Med, 15, 2023
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6LY8
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![BU of 6ly8 by Molmil](/molmil-images/mine/6ly8) | V/A-ATPase from Thermus thermophilus, the soluble domain, including V1, d, two EG stalks, and N-terminal domain of a-subunit. | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, V-type ATP synthase alpha chain, V-type ATP synthase beta chain, ... | 著者 | Kishikawa, J, Nakanishi, A, Furuta, A, Kato, T, Namba, K, Tamakoshi, M, Mitsuoka, K, Yokoyama, K. | 登録日 | 2020-02-13 | 公開日 | 2020-09-09 | 最終更新日 | 2020-09-30 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Mechanical inhibition of isolated V o from V/A-ATPase for proton conductance. Elife, 9, 2020
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