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7V42
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BU of 7v42 by Molmil
Crystal structure of Class I P450 monooxygenase (P450tol) from Rhodococcus coprophilus TC-2 in complex with benzyl-alcohol.
分子名称: PHOSPHATE ION, PROTOPORPHYRIN IX CONTAINING FE, p450tol monooxygenase, ...
著者Zhang, L.L, Huang, J.W, Liu, W.D, Chen, C.C, Guo, R.T.
登録日2021-08-12
公開日2022-06-22
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Molecular Basis for a Toluene Monooxygenase to Govern Substrate Selectivity
Acs Catalysis, 12, 2022
8K2E
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BU of 8k2e by Molmil
Crystal structure of YTHDC1 and Y3 complex
分子名称: 2-chloranyl-6-(4-fluoranylphenoxy)benzoic acid, SULFATE ION, YTH domain-containing protein 1
著者Zhang, H.L, Yang, S.Y.
登録日2023-07-12
公開日2024-07-17
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献PocketFlow is a data-and-knowledge-driven structure-based molecular generative model
Nat. Mach. Intell., 6, 2024
7E0G
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BU of 7e0g by Molmil
Crystal structure of Lysine Specific Demethylase 1 (LSD1) with TAK-418, FAD-adduct
分子名称: GLYCEROL, IMIDAZOLE, Lysine-specific histone demethylase 1A, ...
著者Oki, H.
登録日2021-01-28
公開日2021-03-24
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献LSD1 enzyme inhibitor TAK-418 unlocks aberrant epigenetic machinery and improves autism symptoms in neurodevelopmental disorder models.
Sci Adv, 7, 2021
7XW8
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BU of 7xw8 by Molmil
Crystal structure of Lysine Specific Demethylase 1 (LSD1) with TAK-418 distomer, FAD-adduct
分子名称: GLYCEROL, Lysine-specific histone demethylase 1A, MAGNESIUM ION, ...
著者Oki, H.
登録日2022-05-26
公開日2022-10-12
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.28 Å)
主引用文献Design, synthesis, and structure-activity relationship of TAK-418 and its derivatives as a novel series of LSD1 inhibitors with lowered risk of hematological side effects.
Eur.J.Med.Chem., 239, 2022
1C8A
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BU of 1c8a by Molmil
NMR STRUCTURE OF INTRAMOLECULAR DIMER ANTIFREEZE PROTEIN RD3, 40 SA STRUCTURES
分子名称: PROTEIN (ANTIFREEZE PROTEIN TYPE III)
著者Miura, K, Tsuda, S.
登録日2000-05-04
公開日2001-02-28
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献NMR analysis of type III antifreeze protein intramolecular dimer. Structural basis for enhanced activity.
J.Biol.Chem., 276, 2001
1C89
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BU of 1c89 by Molmil
NMR STRUCTURE OF INTRAMOLECULAR DIMER ANTIFREEZE PROTEIN RD3, 40 SA STRUCTURES
分子名称: ANTIFREEZE PROTEIN TYPE III
著者Miura, K, Tsuda, S.
登録日2000-05-04
公開日2001-02-28
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献NMR analysis of type III antifreeze protein intramolecular dimer. Structural basis for enhanced activity.
J.Biol.Chem., 276, 2001
5AX6
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BU of 5ax6 by Molmil
The crystal structure of CofB, the minor pilin subunit of CFA/III from human enterotoxigenic Escherichia coli.
分子名称: ACETATE ION, CofB
著者Kawahara, K, Oki, K, Fukaksua, F, Maruno, T, Kobayashi, Y, Daisuke, M, Taniguchi, T, Honda, T, Iida, T, Nakamura, S, Ohkubo, T.
登録日2015-07-16
公開日2016-03-09
最終更新日2020-02-26
実験手法X-RAY DIFFRACTION (1.88 Å)
主引用文献Homo-trimeric Structure of the Type IVb Minor Pilin CofB Suggests Mechanism of CFA/III Pilus Assembly in Human Enterotoxigenic Escherichia coli
J.Mol.Biol., 428, 2016
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件を2024-09-04に公開中

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