8U16
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![BU of 8u16 by Molmil](/molmil-images/mine/8u16) | The ternary complex structure of DDB1-CRBN-SALL4(ZF1,2)-short bound to Pomalidomide | 分子名称: | 1,2-ETHANEDIOL, DNA damage-binding protein 1, Protein cereblon, ... | 著者 | Clifton, M.C, Ma, X, Ornelas, E. | 登録日 | 2023-08-30 | 公開日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Structural and biophysical comparisons of the pomalidomide- and CC-220-induced interactions of SALL4 with cereblon. Sci Rep, 13, 2023
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8U15
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![BU of 8u15 by Molmil](/molmil-images/mine/8u15) | The ternary complex structure of DDB1-CRBN-SALL4(ZF1,2)-short bound to CC-220 | 分子名称: | (3S)-3-[4-({4-[(morpholin-4-yl)methyl]phenyl}methoxy)-1-oxo-1,3-dihydro-2H-isoindol-2-yl]piperidine-2,6-dione, DDB1, Protein cereblon, ... | 著者 | Clifton, M.C, Ma, X, Ornelas, E. | 登録日 | 2023-08-30 | 公開日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.95 Å) | 主引用文献 | Structural and biophysical comparisons of the pomalidomide- and CC-220-induced interactions of SALL4 with cereblon. Sci Rep, 13, 2023
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6O5D
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![BU of 6o5d by Molmil](/molmil-images/mine/6o5d) | PYOCHELIN | 分子名称: | GLYCEROL, Neutrophil gelatinase-associated lipocalin, SULFATE ION | 著者 | Rupert, P.B, Strong, R.K, Clifton, M.C, Edwards, T.E, Seattle Structural Genomics Center for Infectious Disease (SSGCID) | 登録日 | 2019-03-01 | 公開日 | 2019-09-11 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Parsing the functional specificity of Siderocalin/Lipocalin 2/NGAL for siderophores and related small-molecule ligands. J Struct Biol X, 2, 2019
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3PEC
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![BU of 3pec by Molmil](/molmil-images/mine/3pec) | |
3PED
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![BU of 3ped by Molmil](/molmil-images/mine/3ped) | |
8EJB
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![BU of 8ejb by Molmil](/molmil-images/mine/8ejb) | |
8DEY
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![BU of 8dey by Molmil](/molmil-images/mine/8dey) | Ternary complex structure of Cereblon-DDB1 bound to IKZF2(ZF2,3) and the molecular glue DKY709 | 分子名称: | (3S)-3-[5-(1-benzylpiperidin-4-yl)-1-oxo-1,3-dihydro-2H-isoindol-2-yl]piperidine-2,6-dione, DNA damage-binding protein 1, Protein cereblon, ... | 著者 | Ma, X, Ornelas, E, Clifton, M.C. | 登録日 | 2022-06-21 | 公開日 | 2023-03-08 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.7 Å) | 主引用文献 | Discovery and characterization of a selective IKZF2 glue degrader for cancer immunotherapy. Cell Chem Biol, 30, 2023
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8U2E
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![BU of 8u2e by Molmil](/molmil-images/mine/8u2e) | Bruton's tyrosine kinase in complex with N-[(2R)-1-[(3R)-3-(methylcarbamoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(3-methylphenyl)-1-oxopropan-2-yl]-1H-indazole-5-carboxamide | 分子名称: | (2S)-6-fluoro-5-[(3S)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-2-(4-methylpiperazine-1-carbonyl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxamide, 1,2-ETHANEDIOL, CHLORIDE ION, ... | 著者 | Gajewski, S, Clifton, M.C. | 登録日 | 2023-09-05 | 公開日 | 2024-01-31 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Discovery and Preclinical Pharmacology of NX-2127, an Orally Bioavailable Degrader of Bruton's Tyrosine Kinase with Immunomodulatory Activity for the Treatment of Patients with B Cell Malignancies. J.Med.Chem., 67, 2024
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8U2D
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![BU of 8u2d by Molmil](/molmil-images/mine/8u2d) | Bruton's tyrosine kinase in complex with N-[(2R)-1-[(3R)-3-(methylcarbamoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(3-methylphenyl)-1-oxopropan-2-yl]-1H-indazole-5-carboxamide | 分子名称: | (3R)-2-[N-(1H-indazole-5-carbonyl)-3-methyl-D-phenylalanyl]-N-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxamide, 1,2-ETHANEDIOL, CHLORIDE ION, ... | 著者 | Gajewski, S, Clifton, M.C. | 登録日 | 2023-09-05 | 公開日 | 2024-01-31 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Discovery and Preclinical Pharmacology of NX-2127, an Orally Bioavailable Degrader of Bruton's Tyrosine Kinase with Immunomodulatory Activity for the Treatment of Patients with B Cell Malignancies. J.Med.Chem., 67, 2024
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7U8F
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![BU of 7u8f by Molmil](/molmil-images/mine/7u8f) | Ternary complex structure of Cereblon-DDB1 bound to IKZF2(ZF2) and the molecular glue DKY709 | 分子名称: | (3S)-3-[5-(1-benzylpiperidin-4-yl)-1-oxo-1,3-dihydro-2H-isoindol-2-yl]piperidine-2,6-dione, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, DNA damage-binding protein 1, ... | 著者 | Ma, X, Ornelas, E, Clifton, M.C. | 登録日 | 2022-03-08 | 公開日 | 2023-03-08 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.15 Å) | 主引用文献 | Discovery and characterization of a selective IKZF2 glue degrader for cancer immunotherapy. Cell Chem Biol, 30, 2023
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4QTP
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![BU of 4qtp by Molmil](/molmil-images/mine/4qtp) | Crystal Structure of an Anti-sigma Factor Antagonist from Mycobacterium paratuberculosis | 分子名称: | 1,2-ETHANEDIOL, Anti-sigma factor antagonist, CITRIC ACID, ... | 著者 | Dranow, D.M, Clifton, M.C, Edwards, T.E, Lorimer, D, Seattle Structural Genomics Center for Infectious Disease, Seattle Structural Genomics Center for Infectious Disease (SSGCID) | 登録日 | 2014-07-08 | 公開日 | 2014-07-16 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal Structure of an Anti-sigma Factor Antagonist from Mycobacterium paratuberculosis TO BE PUBLISHED
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4K19
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![BU of 4k19 by Molmil](/molmil-images/mine/4k19) | The structure of Human Siderocalin bound to the bacterial siderophore fluvibactin | 分子名称: | (4S,5R)-N,N-bis{3-[(2,3-dihydroxybenzoyl)amino]propyl}-2-(2,3-dihydroxyphenyl)-5-methyl-4,5-dihydro-1,3-oxazole-4-carboxamide, CHLORIDE ION, FE (III) ION, ... | 著者 | Correnti, C, Clifton, M.C, Strong, R.K. | 登録日 | 2013-04-04 | 公開日 | 2013-07-31 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (2.74 Å) | 主引用文献 | Siderocalin Outwits the Coordination Chemistry of Vibriobactin, a Siderophore of Vibrio cholerae. Acs Chem.Biol., 8, 2013
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3HYJ
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![BU of 3hyj by Molmil](/molmil-images/mine/3hyj) | Crystal structure of the N-terminal LAGLIDADG domain of DUF199/WhiA | 分子名称: | CHLORIDE ION, GLYCEROL, Protein DUF199/WhiA, ... | 著者 | Kaiser, B.K, Clifton, M.C, Shen, B.W, Stoddard, B.L. | 登録日 | 2009-06-22 | 公開日 | 2009-09-01 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | The structure of a bacterial DUF199/WhiA protein: domestication of an invasive endonuclease. Structure, 17, 2009
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3HYI
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![BU of 3hyi by Molmil](/molmil-images/mine/3hyi) | Crystal structure of full-length DUF199/WhiA from Thermatoga maritima | 分子名称: | GLYCEROL, Protein DUF199/WhiA, SODIUM ION | 著者 | Kaiser, B.K, Clifton, M.C, Shen, B.W, Stoddard, B.L. | 登録日 | 2009-06-22 | 公開日 | 2009-09-01 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.34 Å) | 主引用文献 | The structure of a bacterial DUF199/WhiA protein: domestication of an invasive endonuclease Structure, 17, 2009
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3SAO
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![BU of 3sao by Molmil](/molmil-images/mine/3sao) | The Siderocalin Ex-FABP functions through dual ligand specificities | 分子名称: | (2R)-2-hydroxy-3-(phosphonooxy)propyl tetradecanoate, 2,3-DIHYDROXY-BENZOIC ACID, Extracellular fatty acid-binding protein, ... | 著者 | Correnti, C, Strong, R.K, Clifton, M.C. | 登録日 | 2011-06-03 | 公開日 | 2011-12-28 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Galline Ex-FABP Is an Antibacterial Siderocalin and a Lysophosphatidic Acid Sensor Functioning through Dual Ligand Specificities. Structure, 19, 2011
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3U0B
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![BU of 3u0b by Molmil](/molmil-images/mine/3u0b) | Crystal structure of an oxidoreductase from Mycobacterium smegmatis | 分子名称: | Oxidoreductase, short chain dehydrogenase/reductase family protein, SODIUM ION | 著者 | Arakaki, T.L, Staker, B.L, Clifton, M.C, Abendroth, J, Seattle Structural Genomics Center for Infectious Disease (SSGCID) | 登録日 | 2011-09-28 | 公開日 | 2011-10-05 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Increasing the structural coverage of tuberculosis drug targets. Tuberculosis (Edinb), 95, 2015
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3U0A
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![BU of 3u0a by Molmil](/molmil-images/mine/3u0a) | Crystal structure of an Acyl-CoA thioesterase II TesB2 from Mycobacterium marinum | 分子名称: | Acyl-CoA thioesterase II TesB2, GLYCEROL, SODIUM ION, ... | 著者 | Arakaki, T.L, Staker, B.L, Clifton, M.C, Sankaran, B, Seattle Structural Genomics Center for Infectious Disease (SSGCID) | 登録日 | 2011-09-28 | 公開日 | 2011-10-05 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Increasing the structural coverage of tuberculosis drug targets. Tuberculosis (Edinb), 95, 2015
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4TWG
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![BU of 4twg by Molmil](/molmil-images/mine/4twg) | |
5DWM
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![BU of 5dwm by Molmil](/molmil-images/mine/5dwm) | |
5DVW
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![BU of 5dvw by Molmil](/molmil-images/mine/5dvw) | |
3TZS
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![BU of 3tzs by Molmil](/molmil-images/mine/3tzs) | |
4QHQ
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![BU of 4qhq by Molmil](/molmil-images/mine/4qhq) | |
4KZK
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![BU of 4kzk by Molmil](/molmil-images/mine/4kzk) | |
4JPD
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![BU of 4jpd by Molmil](/molmil-images/mine/4jpd) | |
4JCP
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![BU of 4jcp by Molmil](/molmil-images/mine/4jcp) | |