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5FA5
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BU of 5fa5 by Molmil
Crystal Structure of PRMT5:MEP50 in complex with MTA and H4 peptide
分子名称: 5'-DEOXY-5'-METHYLTHIOADENOSINE, Histone H4, Methylosome protein 50, ...
著者Sprague, E.R, McNamara, J.T.
登録日2015-12-10
公開日2016-02-24
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.34 Å)
主引用文献Disordered methionine metabolism in MTAP/CDKN2A-deleted cancers leads to dependence on PRMT5.
Science, 351, 2016
5TQH
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BU of 5tqh by Molmil
IDH1 R132H mutant in complex with IDH889
分子名称: (4S)-3-[2-({(1S)-1-[5-(4-fluoro-3-methylphenyl)pyrimidin-2-yl]ethyl}amino)pyrimidin-4-yl]-4-(propan-2-yl)-1,3-oxazolidin-2-one, CITRATE ANION, Isocitrate dehydrogenase [NADP] cytoplasmic, ...
著者Xie, X, Kulathila, R.
登録日2016-10-24
公開日2017-01-25
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Optimization of 3-Pyrimidin-4-yl-oxazolidin-2-ones as Allosteric and Mutant Specific Inhibitors of IDH1.
ACS Med Chem Lett, 8, 2017
3GWJ
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BU of 3gwj by Molmil
Crystal structure of Antheraea pernyi arylphorin
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Arylphorin, FORMIC ACID, ...
著者Ryu, K.S, Lee, J.O, Kwon, T.H, Kim, S.
登録日2009-04-01
公開日2009-05-05
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.43 Å)
主引用文献The presence of monoglucosylated N196-glycan is important for the structural stability of storage protein, arylphorin
Biochem.J., 421, 2009
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件を2024-07-17に公開中

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