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8K9O
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BU of 8k9o by Molmil
Crystal structure of Cyanobacteriochrome RcaE GAF domain in Pg state
分子名称: PHYCOCYANOBILIN, histidine kinase
著者Nagae, T, Hirose, Y, Mishima, M.
登録日2023-08-01
公開日2024-05-15
最終更新日2024-06-26
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Green/red light-sensing mechanism in the chromatic acclimation photosensor.
Sci Adv, 10, 2024
1EQ3
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BU of 1eq3 by Molmil
NMR STRUCTURE OF HUMAN PARVULIN HPAR14
分子名称: PEPTIDYL-PROLYL CIS/TRANS ISOMERASE (PPIASE)
著者Sekerina, E, Rahfeld, U.J, Muller, J, Fischer, G, Bayer, P.
登録日2000-04-02
公開日2001-04-04
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献NMR solution structure of hPar14 reveals similarity to the peptidyl prolyl cis/trans isomerase domain of the mitotic regulator hPin1 but indicates a different functionality of the protein.
J.Mol.Biol., 301, 2000
5LEV
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BU of 5lev by Molmil
Crystal structure of human UDP-N-acetylglucosamine-dolichyl-phosphate N-acetylglucosaminephosphotransferase (DPAGT1) (V264G mutant)
分子名称: UDP-N-acetylglucosamine--dolichyl-phosphate N-acetylglucosaminephosphotransferase, UNKNOWN LIGAND
著者Pike, A.C.W, Dong, Y.Y, Chu, A, Tessitore, A, Goubin, S, Dong, L, Mukhopadhyay, S, Mahajan, P, Chalk, R, Berridge, G, Wang, D, Kupinska, K, Belaya, K, Beeson, D, Burgess-Brown, N, Edwards, A.M, Arrowsmith, C.H, Bountra, C, Carpenter, E.P, Structural Genomics Consortium (SGC)
登録日2016-06-30
公開日2016-12-28
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structures of DPAGT1 Explain Glycosylation Disease Mechanisms and Advance TB Antibiotic Design.
Cell, 175, 2018
1WMZ
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BU of 1wmz by Molmil
Crystal Structure of C-type Lectin CEL-I complexed with N-acetyl-D-galactosamine
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-galactopyranose, CALCIUM ION, ...
著者Sugawara, H, Kusunoki, M, Kurisu, G, Fujimoto, T, Aoyagi, H, Hatakeyama, T.
登録日2004-07-22
公開日2004-09-07
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Characteristic Recognition of N-Acetylgalactosamine by an Invertebrate C-type Lectin, CEL-I, Revealed by X-ray Crystallographic Analysis
J.Biol.Chem., 279, 2004
1WMY
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BU of 1wmy by Molmil
Crystal Structure of C-type Lectin CEL-I from Cucumaria echinata
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, lectin CEL-I, ...
著者Sugawara, H, Kusunoki, M, Kurisu, G, Fujimoto, T, Aoyagi, H, Hatakeyama, T.
登録日2004-07-22
公開日2004-09-07
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Characteristic Recognition of N-Acetylgalactosamine by an Invertebrate C-type Lectin, CEL-I, Revealed by X-ray Crystallographic Analysis
J.Biol.Chem., 279, 2004
1GIJ
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BU of 1gij by Molmil
HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE CDK4 INHIBITOR
分子名称: 1-(5-OXO-2,3,5,9B-TETRAHYDRO-1H-PYRROLO[2,1-A]ISOINDOL-9-YL)-3-(5-PYRROLIDIN-2-YL-1H-PYRAZOL-3-YL)-UREA, CELL DIVISION PROTEIN KINASE 2
著者Ikuta, M, Nishimura, S.
登録日2001-02-06
公開日2002-02-06
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystallographic approach to identification of cyclin-dependent kinase 4 (CDK4)-specific inhibitors by using CDK4 mimic CDK2 protein.
J.Biol.Chem., 276, 2002
1GII
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BU of 1gii by Molmil
HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE CDK4 INHIBITOR
分子名称: 1-(5-OXO-2,3,5,9B-TETRAHYDRO-1H-PYRROLO[2,1-A]ISOINDOL-9-YL)-3-PYRIDIN-2-YL-UREA, CELL DIVISION PROTEIN KINASE 2
著者Ikuta, M, Nishimura, S.
登録日2001-02-06
公開日2002-02-06
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystallographic approach to identification of cyclin-dependent kinase 4 (CDK4)-specific inhibitors by using CDK4 mimic CDK2 protein.
J.Biol.Chem., 276, 2001
1GIH
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BU of 1gih by Molmil
HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE CDK4 INHIBITOR
分子名称: 1-(5-OXO-2,3,5,9B-TETRAHYDRO-1H-PYRROLO[2,1-A]ISOINDOL-9-YL)-3-PYRIDIN-2-YL-UREA, CELL DIVISION PROTEIN KINASE 2
著者Ikuta, M, Nishimura, S.
登録日2001-02-06
公開日2002-02-06
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystallographic approach to identification of cyclin-dependent kinase 4 (CDK4)-specific inhibitors by using CDK4 mimic CDK2 protein.
J.Biol.Chem., 276, 2001
3KRD
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BU of 3krd by Molmil
Crystal Structure of Mycobacterium Tuberculosis Proteasome in complex with Fellutamide B
分子名称: (3R)-3-HYDROXYDODECANOIC ACID, Fellutamide B, Proteasome subunit alpha, ...
著者Li, D, Li, H.
登録日2009-11-18
公開日2010-09-29
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Fellutamide B is a potent inhibitor of the Mycobacterium tuberculosis proteasome.
Arch.Biochem.Biophys., 501, 2010
2V1K
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BU of 2v1k by Molmil
Crystal structure of ferrous deoxymyoglobin at pH 6.8
分子名称: GLYCEROL, MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Hersleth, H.-P, Gorbitz, C.H, Andersson, K.K.
登録日2007-05-24
公開日2007-06-12
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Crystallographic and Spectroscopic Studies of Peroxide-Derived Myoglobin Compound II and Occurrence of Protonated Fe(Iv)-O
J.Biol.Chem., 282, 2007
2V1I
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BU of 2v1i by Molmil
Crystal structure of radiation-induced metmyoglobin - aqua ferrous myoglobin at pH 6.8
分子名称: GLYCEROL, MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Hersleth, H.-P, Gorbitz, C.H, Andersson, K.K.
登録日2007-05-24
公開日2007-06-12
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Crystallographic and Spectroscopic Studies of Peroxide-Derived Myoglobin Compound II and Occurrence of Protonated Fe(Iv)-O
J.Biol.Chem., 282, 2007
2V1E
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BU of 2v1e by Molmil
Crystal structure of radiation-induced myoglobin compound II - intermediate H at pH 6.8
分子名称: GLYCEROL, HYDROXIDE ION, MYOGLOBIN, ...
著者Hersleth, H.-P, Gorbitz, C.H, Andersson, K.K.
登録日2007-05-23
公開日2007-06-12
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Crystallographic and Spectroscopic Studies of Peroxide-Derived Myoglobin Compound II and Occurrence of Protonated Fe(Iv)-O
J.Biol.Chem., 282, 2007
2V1H
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BU of 2v1h by Molmil
Crystal structure of radiation-induced metmyoglobin - aqua ferrous myoglobin at pH 5.2
分子名称: GLYCEROL, MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Hersleth, H.-P, Gorbitz, C.H, Andersson, K.K.
登録日2007-05-24
公開日2007-06-12
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Crystallographic and Spectroscopic Studies of Peroxide-Derived Myoglobin Compound II and Occurrence of Protonated Fe(Iv)-O
J.Biol.Chem., 282, 2007
2V1G
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BU of 2v1g by Molmil
Crystal structure of radiation-induced myoglobin compound II - intermediate H at pH 5.2
分子名称: GLYCEROL, HYDROXIDE ION, MYOGLOBIN, ...
著者Hersleth, H.-P, Dalhus, B, Gorbitz, C.H, Andersson, K.K.
登録日2007-05-24
公開日2007-06-12
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Crystallographic and Spectroscopic Studies of Peroxide-Derived Myoglobin Compound II and Occurrence of Protonated Fe(Iv)-O
J.Biol.Chem., 282, 2007
2V1J
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BU of 2v1j by Molmil
Crystal structure of radiation-induced metmyoglobin - aqua ferrous myoglobin at pH 8.7
分子名称: GLYCEROL, MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Hersleth, H.-P, Gorbitz, C.H, Andersson, K.K.
登録日2007-05-24
公開日2007-06-12
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Crystallographic and Spectroscopic Studies of Peroxide-Derived Myoglobin Compound II and Occurrence of Protonated Fe(Iv)-O
J.Biol.Chem., 282, 2007
2V1F
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BU of 2v1f by Molmil
Crystal structure of radiation-induced myoglobin compound II - intermediate H at pH 8.7
分子名称: GLYCEROL, HYDROXIDE ION, MYOGLOBIN, ...
著者Hersleth, H.-P, Gorbitz, C.H, Andersson, K.K.
登録日2007-05-24
公開日2007-06-12
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Crystallographic and Spectroscopic Studies of Peroxide-Derived Myoglobin Compound II and Occurrence of Protonated Fe(Iv)-O
J.Biol.Chem., 282, 2007
6KD5
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BU of 6kd5 by Molmil
Crystal structure of the extracellular domain of MSPL/TMPRSS13 in complex with dec-RVKR-cmk inhibitor
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, DECANOYL-ARG-VAL-LYS-ARG-CHLOROMETHYLKETONE INHIBITOR, ...
著者Ohno, A, Maita, N, Okumura, Y, Nikawa, T.
登録日2019-06-30
公開日2020-06-24
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Crystal structure of inhibitor-bound human MSPL that can activate high pathogenic avian influenza.
Life Sci Alliance, 4, 2021
6EQL
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BU of 6eql by Molmil
Crystal Structure of Human Glycogenin-1 (GYG1) Tyr195pIPhe mutant complexed with manganese and UDP
分子名称: 1,2-ETHANEDIOL, Glycogenin-1, MANGANESE (II) ION, ...
著者Bailey, H.J, Kopec, J, Bilyard, M.K, Bezerra, G.A, Seo Lee, S, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Davis, B.G, Yue, W.W.
登録日2017-10-13
公開日2017-12-20
最終更新日2018-11-14
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献Palladium-mediated enzyme activation suggests multiphase initiation of glycogenesis.
Nature, 563, 2018
6EQJ
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BU of 6eqj by Molmil
Crystal Structure of Human Glycogenin-1 (GYG1) Tyr195pIPhe mutant, apo form
分子名称: 1,2-ETHANEDIOL, Glycogenin-1
著者Bailey, H.J, Kopec, J, Bilyard, M.K, Bezerra, G.A, Seo Lee, S, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Davis, B.G, Yue, W.W.
登録日2017-10-13
公開日2017-12-20
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Palladium-mediated enzyme activation suggests multiphase initiation of glycogenesis.
Nature, 563, 2018
6FWZ
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BU of 6fwz by Molmil
Crystal structure of human UDP-N-acetylglucosamine-dolichyl-phosphate N-acetylglucosaminephosphotransferase (DPAGT1) (V264G mutant) in complex with UDP-GlcNAc
分子名称: (2S)-3-{[{[(2S)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-2-[(6E)-HEXADEC-6-ENOYLOXY]PROPYL (8E)-OCTADEC-8-ENOATE, MAGNESIUM ION, UDP-N-acetylglucosamine--dolichyl-phosphate N-acetylglucosaminephosphotransferase, ...
著者Pike, A.C.W, Dong, Y.Y, Chu, A, Tessitore, A, Goubin, S, Dong, L, Mukhopadhyay, S, Mahajan, P, Chalk, R, Berridge, G, Wang, D, Kupinska, K, Belaya, K, Beeson, D, Burgess-Brown, N, Edwards, A.M, Arrowsmith, C.H, Bountra, C, Carpenter, E.P, Structural Genomics Consortium (SGC)
登録日2018-03-07
公開日2018-07-25
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structures of DPAGT1 Explain Glycosylation Disease Mechanisms and Advance TB Antibiotic Design.
Cell, 175, 2018
6FM9
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BU of 6fm9 by Molmil
Crystal structure of human UDP-N-acetylglucosamine-dolichyl-phosphate N-acetylglucosaminephosphotransferase (DPAGT1)
分子名称: (2S)-3-{[{[(2S)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-2-[(6E)-HEXADEC-6-ENOYLOXY]PROPYL (8E)-OCTADEC-8-ENOATE, UDP-N-acetylglucosamine--dolichyl-phosphate N-acetylglucosaminephosphotransferase
著者Pike, A.C.W, Dong, Y.Y, Chu, A, Tessitore, A, Goubin, S, Dong, L, Mukhopadhyay, S, Mahajan, P, Chalk, R, Berridge, G, Wang, D, Kupinska, K, Belaya, K, Beeson, D, Burgess-Brown, N, Edwards, A.M, Arrowsmith, C.H, Bountra, C, Carpenter, E.P, Structural Genomics Consortium (SGC)
登録日2018-01-30
公開日2018-02-28
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3.6 Å)
主引用文献Structures of DPAGT1 Explain Glycosylation Disease Mechanisms and Advance TB Antibiotic Design.
Cell, 175, 2018
3HFA
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BU of 3hfa by Molmil
Crystal Structure of Mycobacterium Tuberculosis Proteasome open-gate mutant
分子名称: DIMETHYLFORMAMIDE, Proteasome (Alpha subunit) PrcA, Proteasome (Beta subunit) PrcB
著者Li, D, Li, H.
登録日2009-05-11
公開日2009-09-15
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.504 Å)
主引用文献Inhibitors selective for mycobacterial versus human proteasomes.
Nature, 461, 2009
3H6I
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BU of 3h6i by Molmil
Crystal Structure of Mycobacterium Tuberculosis Proteasome Modified by inhibitor GL1
分子名称: DIMETHYLFORMAMIDE, Proteasome (Alpha subunit) PrcA, Proteasome (Beta subunit) PrcB
著者Li, D, Li, H, Lin, G.
登録日2009-04-23
公開日2009-09-15
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.43 Å)
主引用文献Inhibitors selective for mycobacterial versus human proteasomes.
Nature, 461, 2009
3H6F
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BU of 3h6f by Molmil
Crystal Structure of Mycobacterium Tuberculosis Proteasome Modified by inhibitor HT1171
分子名称: DIMETHYLFORMAMIDE, Proteasome (Alpha subunit) PrcA, Proteasome (Beta subunit) PrcB
著者Li, D, Li, H, Lin, G.
登録日2009-04-23
公開日2009-09-15
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Inhibitors selective for mycobacterial versus human proteasomes.
Nature, 461, 2009
3HF9
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BU of 3hf9 by Molmil
Crystal Structure of Mycobacterium Tuberculosis Proteasome open-gate mutant modified by inhibitor GL1
分子名称: Proteasome (Alpha subunit) PrcA, Proteasome (Beta subunit) PrcB
著者Li, D, Li, H.
登録日2009-05-11
公開日2009-09-15
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.878 Å)
主引用文献Inhibitors selective for mycobacterial versus human proteasomes.
Nature, 461, 2009

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