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6TGU
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BU of 6tgu by Molmil
Crystal structure of human protein kinase CK2alpha'(CSNK2A2 gene product) in complex with the 2-aminothiazole-type inhibitor Cl-OH-3
分子名称: 1,2-ETHANEDIOL, 4-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxidanyl-benzoic acid, Casein kinase II subunit alpha'
著者Niefind, K, Lindenblatt, D, Jose, J, Applegate, V.M, Nickelsen, A.
登録日2019-11-18
公開日2020-07-08
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (0.833 Å)
主引用文献Structural and Mechanistic Basis of the Inhibitory Potency of Selected 2-Aminothiazole Compounds on Protein Kinase CK2.
J.Med.Chem., 63, 2020
8QCD
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BU of 8qcd by Molmil
STRUCTURE OF PROTEIN KINASE CK2 CATALYTIC SUBUNIT (ISOFORM CK2ALPHA'; CSNK2A2 GENE PRODUCT) IN COMPLEX WITH THE INHIBITOR 4,5,6,7-TETRABROMOBENZOTRIAZOLE
分子名称: 1,2-ETHANEDIOL, 4,5,6,7-TETRABROMOBENZOTRIAZOLE, Casein kinase II subunit alpha'
著者Werner, C, Niefind, K.
登録日2023-08-25
公開日2023-12-06
実験手法X-RAY DIFFRACTION (1.03 Å)
主引用文献Discovery and Exploration of Protein Kinase CK2 Binding Sites Using CK2alpha Cys336Ser as an Exquisite Crystallographic Tool
Kinases Phosphatases, 2023
8QCG
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BU of 8qcg by Molmil
STRUCTURE OF THE CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 (CK2ALPHA') IN COMPLEX WITH THE NON-HYDROLYZABLE ATP ANALOGUE AMPPNP
分子名称: Casein kinase II subunit alpha', MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
著者Werner, C, Lindenblatt, D, Niefind, K.
登録日2023-08-25
公開日2023-12-06
実験手法X-RAY DIFFRACTION (1.04 Å)
主引用文献Discovery and Exploration of Protein Kinase CK2 Binding Sites Using CK2alpha Cys336Ser as an Exquisite Crystallographic Tool
Kinases Phosphatases, 2023
8QBU
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BU of 8qbu by Molmil
STRUCTURE OF PROTEIN KINASE CK2 CATALYTIC SUBUNIT (ISOFORM CK2ALPHA'; CSNK2A2 GENE PRODUCT) IN COMPLEX WITH THE INHIBITOR CX-4945 AND THE ALPHA-D-POCKET LIGAND 3,4-DICHLORO PHENETHYLAMINE (DPA)
分子名称: 1,2-ETHANEDIOL, 2-(3,4-dichlorophenyl)ethanamine, 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid, ...
著者Werner, C, Niefind, K.
登録日2023-08-25
公開日2023-12-06
実験手法X-RAY DIFFRACTION (1.09 Å)
主引用文献Discovery and Exploration of Protein Kinase CK2 Binding Sites Using CK2alpha Cys336Ser as an Exquisite Crystallographic Tool
Kinases Phosphatases, 2023
8QF1
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BU of 8qf1 by Molmil
STRUCTURE OF THE CATALYTIC SUBUNIT OF PROTEIN KINASE CK2 (CK2ALPHA') IN COMPLEX WITH THE NON-HYDROLYZABLE GTP ANALOGUE GMPPNP
分子名称: Casein kinase II subunit alpha', MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER
著者Werner, C, Lindenblatt, D, Niefind, K.
登録日2023-09-01
公開日2023-12-06
実験手法X-RAY DIFFRACTION (1.32 Å)
主引用文献Discovery and Exploration of Protein Kinase CK2 Binding Sites Using CK2alpha Cys336Ser as an Exquisite Crystallographic Tool
Kinases Phosphatases, 2023
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件を2024-10-09に公開中

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