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8QCD

STRUCTURE OF PROTEIN KINASE CK2 CATALYTIC SUBUNIT (ISOFORM CK2ALPHA'; CSNK2A2 GENE PRODUCT) IN COMPLEX WITH THE INHIBITOR 4,5,6,7-TETRABROMOBENZOTRIAZOLE

Summary for 8QCD
Entry DOI10.2210/pdb8qcd/pdb
DescriptorCasein kinase II subunit alpha', 1,2-ETHANEDIOL, 4,5,6,7-TETRABROMOBENZOTRIAZOLE, ... (4 entities in total)
Functional Keywordsprotein kinase ck2 casein kinase 2 inhibitor tbb, transferase
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight43500.78
Authors
Werner, C.,Niefind, K. (deposition date: 2023-08-25, release date: 2023-12-06)
Primary citationWerner, C.,Lindenblatt, D.,Viht, K.,Uri, A.,Niefind, K.
Discovery and Exploration of Protein Kinase CK2 Binding Sites Using CK2alpha Cys336Ser as an Exquisite Crystallographic Tool
Kinases Phosphatases, 2023
Cited by
DOI: 10.3390/kinasesphosphatases1040018
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.03 Å)
Structure validation

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