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4LRM
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BU of 4lrm by Molmil
EGFR D770_N771insNPG in complex with PD168393
分子名称: Epidermal growth factor receptor, N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide
著者Yun, C.H, Eck, M.J.
登録日2013-07-20
公開日2014-01-15
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.526 Å)
主引用文献Structural, Biochemical, and Clinical Characterization of Epidermal Growth Factor Receptor (EGFR) Exon 20 Insertion Mutations in Lung Cancer.
Sci Transl Med, 5, 2013
7E50
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BU of 7e50 by Molmil
Crystal structure of human microplasmin in complex with kazal-type inhibitor AaTI
分子名称: AAEL006007-PA, GLYCEROL, Plasminogen, ...
著者Varsha, A.W, Jobichen, C, Mok, Y.K.
登録日2021-02-16
公開日2022-02-16
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Crystal structure of Aedes aegypti trypsin inhibitor in complex with mu-plasmin reveals role for scaffold stability in Kazal-type serine protease inhibitor.
Protein Sci., 31, 2022
3U4R
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BU of 3u4r by Molmil
Novel HCV NS5B polymerase Inhibitors: Discovery of Indole C2 Acyl sulfonamides
分子名称: 1-[(2-aminopyridin-4-yl)methyl]-5-chloro-N-({3-[(methylsulfonyl)amino]phenyl}sulfonyl)-3-(2-oxo-1,2-dihydropyridin-3-yl)-1H-indole-2-carboxamide, RNA-directed RNA polymerase
著者Anilkumar, G.N, Selyutin, O, Rosenblum, S.B, Zeng, Q, Jiang, Y, Chan, T.-Y, Pu, H, Wang, L, Bennett, F, Chen, K.X, Lesburg, C.A, Duca, J.S, Gavalas, S, Huang, Y, Pinto, P, Sannagrahi, M, Velazquez, F, Venkataraman, S, Vilbubhan, B, Agrawal, S, Ferrari, E, Jiang, C.-K, Huang, H.-C, Shih, N.-Y, Njoroge, F.G, Kozlowski, J.A.
登録日2011-10-10
公開日2011-12-07
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献II. Novel HCV NS5B polymerase inhibitors: Discovery of indole C2 acyl sulfonamides.
Bioorg.Med.Chem.Lett., 22, 2012
7POZ
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BU of 7poz by Molmil
Crystal structure of Schistosoma mansoni HDAC8 with DMSO bound in the active site
分子名称: DIMETHYL SULFOXIDE, GLYCEROL, Histone deacetylase 8, ...
著者Saccoccia, F, Ruberti, G.
登録日2021-09-10
公開日2022-08-31
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structures of Schistosoma mansoni histone deacetylase 8 reveal a novel binding site for allosteric inhibitors.
J.Biol.Chem., 298, 2022
6DK9
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BU of 6dk9 by Molmil
Yeast Ddi2 Cyanamide Hydratase
分子名称: DNA damage-inducible protein, SULFATE ION, ZINC ION
著者Moore, S.A, Xiao, W, Li, J.
登録日2018-05-29
公開日2019-05-08
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structure of Ddi2, a highly inducible detoxifying metalloenzyme fromSaccharomyces cerevisiae.
J.Biol.Chem., 294, 2019
6DKA
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BU of 6dka by Molmil
Yeast Ddi2 Cyanamide Hydratase
分子名称: CYANAMIDE, DNA damage-inducible protein, SULFATE ION, ...
著者Moore, S.A, Xiao, W, Li, J.
登録日2018-05-29
公開日2019-05-08
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.901 Å)
主引用文献Structure of Ddi2, a highly inducible detoxifying metalloenzyme fromSaccharomyces cerevisiae.
J.Biol.Chem., 294, 2019
4KQM
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Crystal structure of yeast glycogen synthase E169Q mutant in complex with glucose and UDP
分子名称: 6-O-phosphono-alpha-D-glucopyranose, DI(HYDROXYETHYL)ETHER, Gsy2p, ...
著者Chikwana, V.M, Hurley, T.D.
登録日2013-05-15
公開日2013-12-11
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.77 Å)
主引用文献Structural basis for 2'-phosphate incorporation into glycogen by glycogen synthase.
Proc.Natl.Acad.Sci.USA, 110, 2013
4KQ2
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Glucose1,2cyclic phosphate bound activated state of Yeast Glycogen Synthase
分子名称: (2R,3aR,5R,6S,7S,7aR)-5-(hydroxymethyl)tetrahydro-3aH-[1,3,2]dioxaphospholo[4,5-b]pyran-2,6,7-triol 2-oxide, 6-O-phosphono-alpha-D-glucopyranose, BARIUM ION, ...
著者Chikwana, V.M, Hurley, T.D.
登録日2013-05-14
公開日2013-12-11
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Structural basis for 2'-phosphate incorporation into glycogen by glycogen synthase.
Proc.Natl.Acad.Sci.USA, 110, 2013
4KQ1
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BU of 4kq1 by Molmil
Crystal structure of yeast glycogen synthase in complex with uridine-5'-monophosphate
分子名称: 6-O-phosphono-alpha-D-glucopyranose, DI(HYDROXYETHYL)ETHER, Gsy2p, ...
著者Chikwana, V.M, Hurley, T.D.
登録日2013-05-14
公開日2013-12-11
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.66 Å)
主引用文献Structural basis for 2'-phosphate incorporation into glycogen by glycogen synthase.
Proc.Natl.Acad.Sci.USA, 110, 2013
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