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7FT1
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BU of 7ft1 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z2204875953
分子名称: (3P)-3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazole, 1,2-ETHANEDIOL, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.11 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT8
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BU of 7ft8 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with NCL-00024671
分子名称: 1,2-ETHANEDIOL, 2-(4-bromo-1H-pyrazol-1-yl)ethan-1-ol, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSN
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BU of 7fsn by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z254580486
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSL
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BU of 7fsl by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z730649594
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT0
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BU of 7ft0 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z56767614
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSX
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BU of 7fsx by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1328078283
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.91 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT5
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BU of 7ft5 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with POB0093
分子名称: 1,2-ETHANEDIOL, 4-(4-methoxyphenyl)oxane-4-carboxylic acid, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSO
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BU of 7fso by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z198195770
分子名称: 1,2-ETHANEDIOL, D-GLUTAMIC ACID, GLYCINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSQ
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BU of 7fsq by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1429867185
分子名称: 1,2-ETHANEDIOL, 4-methoxy-1H-indole, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSS
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BU of 7fss by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z839706072
分子名称: 1,2-ETHANEDIOL, 2-(4-bromanylpyrazol-1-yl)-~{N}-cyclopropyl-~{N}-methyl-ethanamide, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.11 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSZ
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BU of 7fsz by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z3006151474
分子名称: (5S)-5-(difluoromethoxy)pyridin-2(5H)-one, 1,2-ETHANEDIOL, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT4
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BU of 7ft4 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z48847594
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT3
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BU of 7ft3 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z291279160
分子名称: 1,2-ETHANEDIOL, 1-[2-(trifluoromethyloxy)phenyl]thiourea, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
5LBA
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BU of 5lba by Molmil
Crystal structure of human RECQL5 helicase in complex with DSPL fragment(1-cyclohexyl-3-(oxolan-2-ylmethyl)urea, SGC - Diamond XChem I04-1 fragment screening.
分子名称: 1-cyclohexyl-3-[[(2~{R})-oxolan-2-yl]methyl]urea, ADENOSINE-5'-DIPHOSPHATE, ATP-dependent DNA helicase Q5, ...
著者Newman, J.A, Aitkenhead, H, Talon, R, Savitsky, P, Krojer, T, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Gileadi, O, Structural Genomics Consortium (SGC)
登録日2016-06-15
公開日2016-07-06
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of human RECQL5 helicase in complex with 3D fragment (1-cyclohexyl-3-(oxolan-2-ylmethyl)urea)
To be published
5KKP
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BU of 5kkp by Molmil
Crystal Structure of Human Pseudouridylate Synthase 7
分子名称: 1,2-ETHANEDIOL, Pseudouridylate synthase 7, UNKNOWN ATOM OR ION
著者DONG, A, ZENG, H, WALKER, J.R, Bountra, C, Arrowsmith, C.H, Edwards, A.M, BROWN, P.J, WU, H, Structural Genomics Consortium (SGC)
登録日2016-06-22
公開日2016-08-17
実験手法X-RAY DIFFRACTION (2.26 Å)
主引用文献Crystal Structure of Human Pseudouridylate Synthase 7
to be published
4FUK
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BU of 4fuk by Molmil
Aminopeptidase from Trypanosoma brucei
分子名称: GLYCEROL, Methionine aminopeptidase, UNKNOWN ATOM OR ION, ...
著者El Bakkouri, M, Tempel, W, Osman, K.T, Loppnau, P, Graslund, S, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Hui, R, Lin, Y.H, Structural Genomics Consortium (SGC)
登録日2012-06-28
公開日2012-08-29
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Aminpeptidase from Trypanosoma brucei (CASP Target)
To be Published
3Q91
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BU of 3q91 by Molmil
Crystal Structure of Human Uridine Diphosphate Glucose Pyrophosphatase (NUDT14)
分子名称: Uridine diphosphate glucose pyrophosphatase
著者Tresaugues, L, Siponen, M.I, Arrowsmith, C.H, Berglund, H, Bountra, C, Collins, R, Edwards, A.M, Ekblad, T, Flodin, S, Flores, A, Graslund, S, Hammarstrom, M, Johansson, I, Karlberg, T, Kol, S, Kotenyova, T, Kouznetsova, E, Moche, M, Nyman, T, Persson, C, Schuler, H, Schutz, P, Thorsell, A.G, Van Der Berg, S, Wahlberg, E, Weigelt, J, Welin, M, Nordlund, P, Structural Genomics Consortium (SGC)
登録日2011-01-07
公開日2011-02-16
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal Structure of Human Uridine Diphosphate Glucose Pyrophosphatase (NUDT14)
To be Published
3Q90
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BU of 3q90 by Molmil
Crystal structure of the NTF2 domain of Ras GTPase-activating protein-binding protein 1
分子名称: Ras GTPase-activating protein-binding protein 1
著者Welin, M, Tresaugues, L, Arrowsmith, C.H, Berglund, H, Bountra, C, Collins, R, Edwards, A.M, Ekblad, T, Flodin, S, Flores, A, Graslund, S, Hammarstrom, M, Johansson, I, Karlberg, T, Kol, S, Kotenyova, T, Kouznetsova, E, Moche, M, Nyman, T, Persson, C, Schuler, H, Schutz, P, Siponen, M.I, Thorsell, A.G, Van Der Berg, S, Wahlberg, E, Weigelt, J, Nordlund, P, Structural Genomics Consortium (SGC)
登録日2011-01-07
公開日2011-02-16
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of the NTF2 domain of Ras GTPase-activating protein-binding protein 1
To be Published
4PXW
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BU of 4pxw by Molmil
Crystal structure of human DCAF1 WD40 repeats (Q1250L)
分子名称: Protein VPRBP, UNKNOWN ATOM OR ION
著者Xu, C, Tempel, W, He, H, Li, Y, Walker, J.R, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Min, J, Structural Genomics Consortium (SGC)
登録日2014-03-25
公開日2014-04-16
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献Crystal structure of human DCAF1 WD40 repeats (Q1250L)
TO BE PUBLISHED
4PY6
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BU of 4py6 by Molmil
Crystal Structure of bromodomain of PFA0510w from Plasmodium Falciparum
分子名称: 1,2-ETHANEDIOL, 4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide, Bromodomain protein, ...
著者Fonseca, M, Tallant, C, Hutchinson, A, Savitsky, P, Krojer, T, Filippakopoulos, P, Loppnau, P, Brennan, P.E, von Delft, F, Dong, A, Josling, G.A, Duffy, M.F, Arrowsmith, C.H, Bountra, C, Hui, R, Knapp, S, Wernimont, A.K, Structural Genomics Consortium (SGC)
登録日2014-03-26
公開日2014-04-30
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal Structure of bromodomain of PFA0510w from Plasmodium Falciparum
To be Published
4AW2
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BU of 4aw2 by Molmil
Crystal structure of CDC42 binding protein kinase alpha (MRCK alpha)
分子名称: 1,2-ETHANEDIOL, 5,11-dimethyl-1-oxo-2,6-dihydro-1h-pyrido[4,3-b]carbazol-9-yl benzoate, SERINE/THREONINE-PROTEIN KINASE MRCK ALPHA
著者Elkins, J.M, Muniz, J.R.C, Tan, I, Leung, T, Lafanechere, L, Prudent, R, Abdul Azeez, K, Szklarz, M, Phillips, C, Wang, J, von Delft, F, Bountra, C, Edwards, A, Knapp, S.
登録日2012-05-30
公開日2012-06-20
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Cdc42 Binding Protein Kinase Alpha (Mrck Alpha)
To be Published
3QWM
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BU of 3qwm by Molmil
Crystal Structure of GEP100, the plextrin homology domain of IQ motif and SEC7 domain-containing protein 1 isoform a
分子名称: IQ motif and SEC7 domain-containing protein 1
著者Filippakopoulos, P, Picaud, S, Felletar, I, Feller, S, Janning, M, Sabe, H, Krojer, T, Chaikuad, A, Allerston, C, von Delft, F, Bountra, C, Arrowsmith, C.H, Weigelt, J, Edwards, A, Knapp, S, Structural Genomics Consortium (SGC)
登録日2011-02-28
公開日2011-04-13
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.39 Å)
主引用文献Crystal Structure of GEP100, the plextrin homology domain of IQ motif and SEC7 domain-containing protein 1 isoform a
to be published
4GD4
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BU of 4gd4 by Molmil
Crystal Structure of JMJD2A Complexed with Inhibitor
分子名称: 2-(1H-pyrazol-3-yl)pyridine-4-carboxylic acid, CHLORIDE ION, Lysine-specific demethylase 4A, ...
著者King, O.N.F, Krojer, T, Arrowsmith, C.H, Edwards, A, Bountra, C, McDonough, M.A, Schofield, C.J, Structural Genomics Consortium (SGC)
登録日2012-07-31
公開日2012-08-15
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.33 Å)
主引用文献Crystal Structure of JMJD2A Complexed with Inhibitor
TO BE PUBLISHED
4QNS
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BU of 4qns by Molmil
Crystal structure of bromodomain from Plasmodium faciparum GCN5, PF3D7_0823300
分子名称: 1,2-ETHANEDIOL, ACETATE ION, Histone acetyltransferase GCN5, ...
著者Fonseca, M, Tallant, C, Knapp, S, Loppnau, P, von Delft, F, Wernimont, A.K, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Hui, R, Structural Genomics Consortium (SGC)
登録日2014-06-18
公開日2014-07-16
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.497 Å)
主引用文献Crystal structure of bromodomain from Plasmodium faciparum GCN5, PF3D7_0823300
TO BE PUBLISHED
4QQI
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BU of 4qqi by Molmil
Crystal structure of ANKRA2-RFX7 complex
分子名称: Ankyrin repeat family A protein 2, DNA-binding protein RFX7, SULFATE ION, ...
著者Xu, C, Tempel, W, Dong, A, Mackenzie, F, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Min, J, Structural Genomics Consortium (SGC)
登録日2014-06-27
公開日2014-09-03
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献Crystal structure of ANKRA2-RFX7 complex
To Be Published

222415

件を2024-07-10に公開中

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