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3CJG
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BU of 3cjg by Molmil
Crystal structure of VEGFR2 in complex with a 3,4,5-trimethoxy aniline containing pyrimidine
分子名称: N~4~-methyl-N~4~-(3-methyl-1H-indazol-6-yl)-N~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamine, SULFATE ION, Vascular endothelial growth factor receptor 2
著者Nolte, R.T.
登録日2008-03-12
公開日2008-10-07
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Discovery of 5-[[4-[(2,3-dimethyl-2H-indazol-6-yl)methylamino]-2-pyrimidinyl]amino]-2-methyl-benzenesulfonamide (Pazopanib), a novel and potent vascular endothelial growth factor receptor inhibitor.
J.Med.Chem., 51, 2008
3D0U
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BU of 3d0u by Molmil
Crystal Structure of Lysine Riboswitch Bound to Lysine
分子名称: IRIDIUM HEXAMMINE ION, LYSINE, Lysine Riboswitch RNA
著者Garst, A.D, Heroux, A, Rambo, R.P, Batey, R.T.
登録日2008-05-02
公開日2008-07-01
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structure of the lysine riboswitch regulatory mRNA element.
J.Biol.Chem., 283, 2008
3DDW
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BU of 3ddw by Molmil
Crystal structure of glycogen phosphorylase complexed with an anthranilimide based inhibitor GSK055
分子名称: (2S)-{[(3-{[(2-chloro-6-methylphenyl)carbamoyl]amino}naphthalen-2-yl)carbonyl]amino}(phenyl)ethanoic acid, (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ...
著者Nolte, R.T.
登録日2008-06-06
公開日2009-01-27
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Anthranilimide based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes. Part 3: X-ray crystallographic characterization, core and urea optimization and in vivo efficacy.
Bioorg.Med.Chem.Lett., 19, 2009
3DDS
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BU of 3dds by Molmil
Crystal structure of glycogen phosphorylase complexed with an anthranilimide based inhibitor GSK261
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CAFFEINE, ...
著者Nolte, R.T.
登録日2008-06-06
公開日2009-01-27
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Anthranilimide based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes. Part 3: X-ray crystallographic characterization, core and urea optimization and in vivo efficacy.
Bioorg.Med.Chem.Lett., 19, 2009
3DD1
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BU of 3dd1 by Molmil
Crystal structure of glycogen phophorylase complexed with an anthranilimide based inhibitor GSK254
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-cyclohexyl-N-[(3-{[(2,4,6-trimethylphenyl)carbamoyl]amino}naphthalen-2-yl)carbonyl]-D-alanine, ...
著者Nolte, R.T.
登録日2008-06-04
公開日2009-04-21
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.57 Å)
主引用文献Anthranilimide based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes. Part 3: X-ray crystallographic characterization, core and urea optimization and in vivo efficacy.
Bioorg.Med.Chem.Lett., 19, 2009
3DS7
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BU of 3ds7 by Molmil
Structure of an RNA-2'-deoxyguanosine complex
分子名称: 2'-DEOXY-GUANOSINE, 67-MER, ACETATE ION, ...
著者Edwards, A.L, Batey, R.T.
登録日2008-07-11
公開日2009-02-17
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献A structural basis for the recognition of 2'-deoxyguanosine by the purine riboswitch.
J.Mol.Biol., 385, 2009
3DNJ
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BU of 3dnj by Molmil
The structure of the Caulobacter crescentus ClpS protease adaptor protein in complex with a N-end rule peptide
分子名称: ATP-dependent Clp protease adapter protein clpS, MAGNESIUM ION, synthetic N-end rule peptide
著者Wang, K, Roman-Hernandez, G, Grant, R.A, Sauer, R.T, Baker, T.A.
登録日2008-07-02
公開日2008-11-18
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献The molecular basis of N-end rule recognition.
Mol.Cell, 32, 2008
3EQ2
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BU of 3eq2 by Molmil
Structure of Hexagonal Crystal form of Pseudomonas aeruginosa RssB
分子名称: Probable two-component response regulator
著者Levchenko, I, Grant, R.A, Sauer, R.T, Baker, T.A.
登録日2008-09-30
公開日2009-10-20
最終更新日2017-10-25
実験手法X-RAY DIFFRACTION (3.401 Å)
主引用文献The structure of rssb, a clpx adaptor protein that regulates sigma S
To be Published
3EOD
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BU of 3eod by Molmil
Crystal structure of N-terminal domain of E. coli RssB
分子名称: Protein hnr
著者Levchenko, I, Grant, R.A, Sauer, R.T, Baker, T.A.
登録日2008-09-26
公開日2009-10-06
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献The structure of RssB, a ClpX adaptor protein that regulates sigma S
To be Published
3ES2
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BU of 3es2 by Molmil
Structure of the C-terminal phosphatase domain of P. aeruginonsa RssB
分子名称: Probable two-component response regulator
著者Levchenko, I, Grant, R.A, Sauer, R.T, Baker, T.A.
登録日2008-10-03
公開日2009-10-20
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献The structure of RSSB, a clpx adaptor protein that regulates sigma s
To be Published
3FO6
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BU of 3fo6 by Molmil
Crystal structure of guanine riboswitch bound to 6-O-methylguanine
分子名称: 6-O-methylguanine, ACETATE ION, COBALT HEXAMMINE(III), ...
著者Gilbert, S.D, Reyes, F.E, Batey, R.T.
登録日2008-12-28
公開日2009-06-23
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Adaptive ligand binding by the purine riboswitch in the recognition of Guanine and adenine analogs.
Structure, 17, 2009
3F7A
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BU of 3f7a by Molmil
Structure of Orthorhombic crystal form of Pseudomonas aeruginosa RssB
分子名称: Probable two-component response regulator
著者levchenko, I, Grant, R.A, Sauer, R.T, Baker, T.A.
登録日2008-11-07
公開日2009-11-24
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (4.308 Å)
主引用文献The structure of RSSB, a CLPX adaptor protein that regulates sigma S
To be Published
3FO4
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BU of 3fo4 by Molmil
Crystal structure of guanine riboswitch C74U mutant bound to 6-chloroguanine
分子名称: 6-chloroguanine, ACETATE ION, COBALT HEXAMMINE(III), ...
著者Gilbert, S.D, Batey, R.T.
登録日2008-12-27
公開日2009-06-23
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Adaptive ligand binding by the purine riboswitch in the recognition of Guanine and adenine analogs.
Structure, 17, 2009
3F79
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BU of 3f79 by Molmil
Structure of pseudo-centered cell crystal form of the C-terminal phosphatase domain of P. aeruginosa RssB
分子名称: MAGNESIUM ION, Probable two-component response regulator
著者Levchenko, I, Grant, R.A, Sauer, R.T, Baker, T.A.
登録日2008-11-07
公開日2009-11-24
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The structure of RSSB, a CLPX adaptor protein that regulates sigma S
To be Published
3GCO
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BU of 3gco by Molmil
Crystal structure of DegS H198P/D320A mutant modified by DFP in complex with DNRDGNVYQF OMP peptide
分子名称: DNRDGNVYQF peptide, Protease degS
著者Sohn, J, Grant, R.A, Sauer, R.T.
登録日2009-02-22
公開日2009-03-31
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (2.798 Å)
主引用文献OMP peptides activate the DegS stress-sensor protease by a relief of inhibition mechanism.
Structure, 17, 2009
3GDS
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BU of 3gds by Molmil
Crystal structure of DegS H198P/D320A mutant modified by DFP in complex with DNRDGNVYYF peptide
分子名称: DNRDGNVYYF peptide, Protease degS
著者Sohn, J, Grant, R.A, Sauer, R.T.
登録日2009-02-24
公開日2009-03-31
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献OMP peptides activate the DegS stress-sensor protease by a relief of inhibition mechanism.
Structure, 17, 2009
3G4M
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BU of 3g4m by Molmil
Crystal structure of guanine riboswitch bound to 2-aminopurine
分子名称: 9H-purin-2-amine, ACETATE ION, COBALT HEXAMMINE(III), ...
著者Gilbert, S.D, Batey, R.T.
登録日2009-02-04
公開日2009-06-23
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Adaptive ligand binding by the purine riboswitch in the recognition of Guanine and adenine analogs.
Structure, 17, 2009
3GCN
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BU of 3gcn by Molmil
Crystal structure of DegS H198P/D320A mutant modified by DFP in complex with OMP peptide (YQF)
分子名称: Protease degS, YQF peptide
著者Sohn, J, Sauer, R.T, Grant, R.A.
登録日2009-02-22
公開日2009-03-31
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (3.002 Å)
主引用文献Mechanisms of allosteric activation of the DegS protease by OMP-peptide binding and protein-substrate binding
To be Published
3GDU
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BU of 3gdu by Molmil
Crystal structure of DegS H198P/D320A mutant modified by DFP and in complex with YRF peptide
分子名称: DegS protease, YRF peptide
著者Sohn, J, Grant, R.A, Sauer, R.T.
登録日2009-02-24
公開日2009-03-31
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献OMP peptides activate the DegS stress-sensor protease by a relief of inhibition mechanism.
Structure, 17, 2009
3G1B
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BU of 3g1b by Molmil
The structure of the M53A mutant of Caulobacter crescentus clpS protease adaptor protein in complex with WLFVQRDSKE peptide
分子名称: 10-residue peptide, ATP-dependent Clp protease adapter protein clpS, MAGNESIUM ION
著者Baker, T.A, Roman-Hernandez, G, Sauer, R.T, Grant, R.A.
登録日2009-01-29
公開日2009-04-28
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.448 Å)
主引用文献Molecular basis of substrate selection by the N-end rule adaptor protein ClpS.
Proc.Natl.Acad.Sci.USA, 106, 2009
3GDV
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BU of 3gdv by Molmil
Crystal structure of DegS H198P/D320A mutant modified by DFP and in complex with YQF peptide
分子名称: DegS protease, YQF peptide
著者Sohn, J, Grant, R.A, Sauer, R.T.
登録日2009-02-24
公開日2009-03-31
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (2.489 Å)
主引用文献OMP peptides activate the DegS stress-sensor protease by a relief of inhibition mechanism.
Structure, 17, 2009
3GES
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BU of 3ges by Molmil
Crystal structure of the guanine riboswitch C74U mutant bound to 6-O-methylguanine
分子名称: 6-O-methylguanine, ACETATE ION, COBALT HEXAMMINE(III), ...
著者Gilbert, S.D, Batey, R.T.
登録日2009-02-26
公開日2009-06-23
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Adaptive ligand binding by the purine riboswitch in the recognition of Guanine and adenine analogs
Structure, 17, 2009
3G19
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BU of 3g19 by Molmil
The structure of the Caulobacter crescentus clpS protease adaptor protein in complex with LLL tripeptide
分子名称: ATP-dependent Clp protease adapter protein clpS, LLL tripeptide
著者Baker, T.A, Roman-Hernandez, G, Sauer, R.T, Grant, R.A.
登録日2009-01-29
公開日2009-04-28
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.849 Å)
主引用文献Molecular basis of substrate selection by the N-end rule adaptor protein ClpS.
Proc.Natl.Acad.Sci.USA, 106, 2009
3GER
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BU of 3ger by Molmil
Guanine riboswitch bound to 6-chloroguanine
分子名称: 6-chloroguanine, ACETATE ION, COBALT HEXAMMINE(III), ...
著者Gilbert, S.D, Batey, R.T.
登録日2009-02-25
公開日2009-06-23
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Adaptive ligand binding by the purine riboswitch in the recognition of Guanine and adenine analogs
Structure, 17, 2009
3G3P
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BU of 3g3p by Molmil
The structure of the M53A Mutant of the Caulobacter crescentus CLPS in complex with a peptide containing an amino-terminal norleucine residue
分子名称: ATP-dependent Clp protease adapter protein clpS, MAGNESIUM ION, Peptide (NLE)LFVQRDSKE
著者Baker, T.A, Roman-Hernandez, G, Sauer, R.T, Grant, R.A.
登録日2009-02-02
公開日2010-03-09
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (1.478 Å)
主引用文献Structure of Caulobacter crescentus ClpS in complex with various peptides
To be Published

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