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6SAZ
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BU of 6saz by Molmil
Cleaved human fetuin-b in complex with crayfish astacin
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Astacin, ...
著者Gomis-Ruth, F.X, Guevara, T, Cuppari, A, Korschgen, H, Schmitz, C, Kuske, M, Yiallouros, I, Floehr, J, Jahnen-Dechent, W, Stocker, W.
登録日2019-07-18
公開日2019-10-23
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献The C-terminal region of human plasma fetuin-B is dispensable for the raised-elephant-trunk mechanism of inhibition of astacin metallopeptidases.
Sci Rep, 9, 2019
3LG7
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BU of 3lg7 by Molmil
Crystal structure of HIV epitope-scaffold 4E10_S0_1EZ3A_002_C
分子名称: 4E10_S0_1EZ3A_002_C (T246), SULFATE ION
著者Holmes, M.A.
登録日2010-01-19
公開日2010-09-22
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Computational Design of Epitope-Scaffolds Allows Induction of Antibodies Specific for a Poorly Immunogenic HIV Vaccine Epitope.
Structure, 18, 2010
6HN1
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BU of 6hn1 by Molmil
Complex of Caprine Serum Albumin with diclofenac
分子名称: 2-[2,6-DICHLOROPHENYL)AMINO]BENZENEACETIC ACID, Albumin, CHLORIDE ION
著者Talaj, J.A, Bujacz, A, Bujacz, G.
登録日2018-09-13
公開日2019-10-09
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Structural Investigation of Diclofenac Binding to Ovine, Caprine, and Leporine Serum Albumins.
Int J Mol Sci, 24, 2023
6HSV
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BU of 6hsv by Molmil
Engineered higher-order assembly of Cholera Toxin B subunits via the addition of C-terminal parallel coiled-coiled domains
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, CHLORIDE ION, PHOSPHATE ION, ...
著者Pearson, A.R, Turnbull, W.B, Ross, J.F, Trinh, C.H, Webb, M.E.
登録日2018-10-01
公開日2019-03-20
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Directed Assembly of Homopentameric Cholera Toxin B-Subunit Proteins into Higher-Order Structures Using Coiled-Coil Appendages.
J.Am.Chem.Soc., 141, 2019
6HT9
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BU of 6ht9 by Molmil
Mouse fetuin-B in complex with crayfish astacin
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Astacin, ...
著者Gomis-Ruth, F.X, Goulas, T, Guevara, T, Cuppari, A.
登録日2018-10-03
公開日2019-03-13
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structure of mammalian plasma fetuin-B and its mechanism of selective metallopeptidase inhibition.
Iucrj, 6, 2019
6L4O
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BU of 6l4o by Molmil
Crystal structure of API5-FGF2 complex
分子名称: Apoptosis inhibitor 5, Fibroblast growth factor 2
著者Lee, B.I, Bong, S.M.
登録日2019-10-18
公開日2020-04-29
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Regulation of mRNA export through API5 and nuclear FGF2 interaction.
Nucleic Acids Res., 48, 2020
7UTG
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BU of 7utg by Molmil
2D9 nanobody to BCL11A-exZF23 fragment
分子名称: 2D9-V102G nanobody, SULFATE ION
著者Dassama, L.M.K, Zhai, L.
登録日2022-04-26
公開日2022-12-21
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献A Cell-Permeant Nanobody-Based Degrader That Induces Fetal Hemoglobin.
Acs Cent.Sci., 8, 2022
3U50
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BU of 3u50 by Molmil
Crystal Structure of the Tetrahymena telomerase processivity factor Teb1 OB-C
分子名称: Telomerase-associated protein 82, ZINC ION
著者Zeng, Z, Huang, J, Yang, Y, Lei, M.
登録日2011-10-10
公開日2011-12-14
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural basis for Tetrahymena telomerase processivity factor Teb1 binding to single-stranded telomeric-repeat DNA.
Proc.Natl.Acad.Sci.USA, 108, 2011
3U58
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BU of 3u58 by Molmil
Crystal Structure of the Tetrahymena telomerase processivity factor Teb1 AB
分子名称: DNA (5'-D(*GP*GP*GP*T)-3'), Tetrahymena Teb1 AB
著者Zeng, Z, Huang, J, Yang, Y, Lei, M.
登録日2011-10-11
公開日2011-12-28
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.613 Å)
主引用文献Structural basis for Tetrahymena telomerase processivity factor Teb1 binding to single-stranded telomeric-repeat DNA.
Proc.Natl.Acad.Sci.USA, 108, 2011
7W1I
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BU of 7w1i by Molmil
Crystal structure of carboxylesterase mutant from Thermobifida fusca with C8X and C9C
分子名称: 4-(2-hydroxyethyloxycarbonyl)benzoic acid, Carboxylesterase, bis(2-hydroxyethyl) benzene-1,4-dicarboxylate
著者Han, X, Gerlis, H, Li, Z, Gao, J, Wei, R, Liu, W.
登録日2021-11-19
公開日2022-11-23
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献Structural Insights into (Tere)phthalate-Ester Hydrolysis by a Carboxylesterase and Its Role in Promoting PET Depolymerization
Acs Catalysis, 12, 2022
7W1K
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BU of 7w1k by Molmil
Crystal structure of carboxylesterase from Thermobifida fusca
分子名称: Carboxylesterase
著者Han, X, Gerlis, H, Li, Z, Gao, J, Wei, R, Liu, W.
登録日2021-11-19
公開日2022-11-23
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.39 Å)
主引用文献Structural Insights into (Tere)phthalate-Ester Hydrolysis by a Carboxylesterase and Its Role in Promoting PET Depolymerization
Acs Catalysis, 12, 2022
7W1J
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BU of 7w1j by Molmil
Crystal structure of carboxylesterase from Thermobifida fusca with J1K
分子名称: 4-(2-hydroxyethylcarbamoyl)benzoic acid, Carboxylesterase
著者Han, X, Gerlis, H, Li, Z, Gao, J, Wei, R, Liu, W.
登録日2021-11-19
公開日2022-11-23
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献Structural Insights into (Tere)phthalate-Ester Hydrolysis by a Carboxylesterase and Its Role in Promoting PET Depolymerization
Acs Catalysis, 12, 2022
7W1L
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BU of 7w1l by Molmil
Crystal structure of carboxylesterase mutant from Thermobifida fusca with C8X
分子名称: Carboxylesterase, bis(2-hydroxyethyl) benzene-1,4-dicarboxylate
著者Han, X, Gerlis, H, Li, Z, Gao, J, Wei, R, Liu, W.
登録日2021-11-19
公開日2022-11-23
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.44 Å)
主引用文献Structural Insights into (Tere)phthalate-Ester Hydrolysis by a Carboxylesterase and Its Role in Promoting PET Depolymerization
Acs Catalysis, 12, 2022
5DOK
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BU of 5dok by Molmil
Crystal structure of Tetrahymena p45C
分子名称: MAGNESIUM ION, Telomerase associated protein p45
著者Wan, B, Tang, T, Wu, J, Lei, M.
登録日2015-09-11
公開日2015-11-25
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The Tetrahymena telomerase p75-p45-p19 subcomplex is a unique CST complex
Nat.Struct.Mol.Biol., 22, 2015
4FBS
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BU of 4fbs by Molmil
Structure of monomeric NT from Euprosthenops australis Major Ampullate Spidroin 1 (MaSp1)
分子名称: BROMIDE ION, Major ampullate spidroin 1
著者Askarieh, G, Hedhammar, M, Rising, A, Johansson, J, Knight, S.D.
登録日2012-05-23
公開日2012-08-01
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献pH-Dependent Dimerization of Spider Silk N-Terminal Domain Requires Relocation of a Wedged Tryptophan Side Chain
J.Mol.Biol., 2012
3PSU
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BU of 3psu by Molmil
HIV-1 protease in complex with an isobutyl decorated oligoamine (symmetric binding mode)
分子名称: CHLORIDE ION, N,N'-(iminodiethane-2,1-diyl)bis[4-amino-N-(2-methylpropyl)benzenesulfonamide], Protease
著者Lindemann, I, Heine, A, Klebe, G.
登録日2010-12-02
公開日2011-12-07
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献Multiple binding modes of a symmetric inhibitor in HIV-1 protease
To be Published
3U4V
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BU of 3u4v by Molmil
Crystal Structure of the Tetrahymena telomerase processivity factor Teb1 OB-A
分子名称: Telomerase-associated protein 82
著者Zeng, Z, Huang, J, Yang, Y, Lei, M.
登録日2011-10-10
公開日2011-12-28
最終更新日2012-05-23
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural basis for Tetrahymena telomerase processivity factor Teb1 binding to single-stranded telomeric-repeat DNA.
Proc.Natl.Acad.Sci.USA, 108, 2011
3U4Z
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BU of 3u4z by Molmil
Crystal Structure of the Tetrahymena telomerase processivity factor Teb1 OB-B
分子名称: Telomerase-associated protein 82
著者Zeng, Z, Huang, J, Yang, Y, Lei, M.
登録日2011-10-10
公開日2011-12-14
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural basis for Tetrahymena telomerase processivity factor Teb1 binding to single-stranded telomeric-repeat DNA.
Proc.Natl.Acad.Sci.USA, 108, 2011
7UVF
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BU of 7uvf by Molmil
Crystal structure of ZED8 Fab complex with CD8 alpha
分子名称: CHLORIDE ION, GLYCEROL, Immunoglobulin heavy chain, ...
著者Yu, C, Davies, C, Koerber, J.T, Williams, S.
登録日2022-05-01
公開日2022-10-12
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Preclinical development of ZED8, an 89 Zr immuno-PET reagent for monitoring tumor CD8 status in patients undergoing cancer immunotherapy.
Eur J Nucl Med Mol Imaging, 50, 2023
1FHF
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BU of 1fhf by Molmil
THE STRUCTURE OF SOYBEAN PEROXIDASE
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CALCIUM ION, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Henriksen, A, Mirza, O, Indiana, C, Welinder, K, Teilum, K, Gajhede, M.
登録日2000-08-01
公開日2001-02-14
最終更新日2018-01-31
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of soybean seed coat peroxidase: a plant peroxidase with unusual stability and haem-apoprotein interactions.
Protein Sci., 10, 2001
4AS0
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BU of 4as0 by Molmil
Cyclometalated Phthalimides as Protein Kinase Inhibitors
分子名称: PHTALIMIDE-RUTHENIUM COMPLEX, SERINE/THREONINE-PROTEIN KINASE PIM-1
著者Blanck, S, Geisselbrecht, Y, Middel, S, Mietke, T, Harms, K, Essen, L.-O, Meggers, E.
登録日2012-04-27
公開日2012-10-03
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Bioactive Cyclometalated Phthalimides: Design, Synthesis and Kinase Inhibition.
Dalton Trans, 41, 2012
1E33
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BU of 1e33 by Molmil
Crystal structure of an Arylsulfatase A mutant P426L
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Arylsulfatase A, MAGNESIUM ION
著者von Buelow, R, Schmidt, B, Dierks, T, von Figura, K, Uson, I.
登録日2000-06-06
公開日2001-05-25
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Defective oligomerization of arylsulfatase a as a cause of its instability in lysosomes and metachromatic leukodystrophy.
J. Biol. Chem., 277, 2002
5U0M
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BU of 5u0m by Molmil
Fatty aldehyde dehydrogenase from Marinobacter aquaeolei VT8 and cofactor complex
分子名称: 1,2-ETHANEDIOL, CITRIC ACID, N-succinylglutamate 5-semialdehyde dehydrogenase, ...
著者Shi, K, Mulliner, K, Barney, B.M, Aihara, H.
登録日2016-11-24
公開日2017-04-26
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.075 Å)
主引用文献Five Fatty Aldehyde Dehydrogenase Enzymes from Marinobacter and Acinetobacter spp. and Structural Insights into the Aldehyde Binding Pocket.
Appl. Environ. Microbiol., 83, 2017
7SZQ
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BU of 7szq by Molmil
Human P300 complexed with an azaindazole inhibitor
分子名称: 1-[1-(4-chlorophenyl)cyclopentane-1-carbonyl]-N-1H-pyrazolo[4,3-b]pyridin-5-yl-D-prolinamide, Histone acetyltransferase p300
著者Shewchuk, L.M, Reid, R.A.
登録日2021-11-29
公開日2022-11-09
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Discovery of Proline-Based p300/CBP Inhibitors Using DNA-Encoded Library Technology in Combination with High-Throughput Screening.
J.Med.Chem., 65, 2022
7SSK
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BU of 7ssk by Molmil
Human P300 complexed with a glycine-based inhibitor
分子名称: 1,2-ETHANEDIOL, ACETATE ION, Histone acetyltransferase p300, ...
著者Shewchuk, L.M, Reid, R.A.
登録日2021-11-11
公開日2022-11-09
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.36 Å)
主引用文献Discovery of Proline-Based p300/CBP Inhibitors Using DNA-Encoded Library Technology in Combination with High-Throughput Screening.
J.Med.Chem., 65, 2022

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