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2GCZ
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BU of 2gcz by Molmil
Solution Structure of alpha-Conotoxin OmIA
分子名称: Alpha-conotoxin OmIA
著者Chi, S.-W, Kim, D.-H, Olivera, B.M, McIntosh, J.M, Han, K.-H.
登録日2006-03-15
公開日2006-07-25
最終更新日2020-06-24
実験手法SOLUTION NMR
主引用文献Solution conformation of a neuronal nicotinic acetylcholine receptor antagonist alpha-conotoxin OmIA that discriminates alpha3 vs. alpha6 nAChR subtypes
Biochem.Biophys.Res.Commun., 345, 2006
6EAS
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BU of 6eas by Molmil
Co-crystal of pseudokinase DRIK1 (drought responsive inactive kinase 1) bound to ENMD-2076
分子名称: 6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine, GLYCEROL, drought responsive inactive kinase 1
著者Aquino, B, Counago, R.M, Fala, A.M, Massirer, K.B, Elkins, J.M, Arruda, P, Structural Genomics Consortium (SGC)
登録日2018-08-03
公開日2018-08-22
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Co-crystal of pseudokinase DRIK1 with ENMD-2076
To be Published
2GAK
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BU of 2gak by Molmil
X-ray crystal structure of murine leukocyte-type Core 2 b1,6-N-acetylglucosaminyltransferase (C2GnT-L)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, beta-1,6-N-acetylglucosaminyltransferase
著者Pak, J.E, Rini, J.M.
登録日2006-03-09
公開日2006-07-11
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献X-ray Crystal Structure of Leukocyte Type Core 2 beta1,6-N-Acetylglucosaminyltransferase: Evidence for a covergence of metal ion independent glycosyltransferase mechanism.
J.Biol.Chem., 281, 2006
6EH0
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BU of 6eh0 by Molmil
Apo crystal structure of the Protein-Kinase A catalytic subunit from Criteculus
分子名称: cAMP-dependent protein kinase catalytic subunit alpha
著者Mueller, J.M, Heine, A, Klebe, G.
登録日2017-09-12
公開日2018-10-10
最終更新日2019-05-15
実験手法X-RAY DIFFRACTION (1.49 Å)
主引用文献Conceptional Design of Self-Assembling Bisubstrate-like Inhibitors of Protein Kinase A Resulting in a Boronic Acid Glutamate Linkage
Acs Omega, 2019
6EIM
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BU of 6eim by Molmil
Human STK10 bound to GW683134A
分子名称: 1,2-ETHANEDIOL, Serine/threonine-protein kinase 10, ~{N}-[5-[4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-1~{H}-benzimidazol-2-yl]furan-2-carboxamide
著者Sorrell, F.J, Berger, B.-T, Salah, E, von Delft, F, Bountra, C, Arrowsmith, C, Edwards, A.M, Knapp, S, Elkins, J.M.
登録日2017-09-19
公開日2017-11-01
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.43 Å)
主引用文献Human STK10 bound to GW683134
To Be Published
6ERW
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BU of 6erw by Molmil
Crystal Structure of the Protein-Kinase A catalytic subunit from Criteculus Griseus in complex with compounds RKp013 and Fasudil
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 5-(1,4-DIAZEPAN-1-SULFONYL)ISOQUINOLINE, UPF0418 protein FAM164A, ...
著者Mueller, J.M, Heine, A, Klebe, G.
登録日2017-10-19
公開日2018-10-31
最終更新日2019-05-15
実験手法X-RAY DIFFRACTION (1.89 Å)
主引用文献Conceptional Design of Self-Assembling Bisubstrate-like Inhibitors of Protein Kinase A Resulting in a Boronic Acid Glutamate Linkage
Acs Omega, 2019
6ESA
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BU of 6esa by Molmil
Crystal Structure of the Protein-Kinase A catalytic subunit from Criteculus Griseus in complex with compounds RKp120 and AMP
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, ADENOSINE MONOPHOSPHATE, beta-D-ribopyranose, ...
著者Mueller, J.M, Heine, A, Klebe, G.
登録日2017-10-19
公開日2018-10-31
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.307 Å)
主引用文献Conceptional Design of Self-Assembling Bisubstrate-like Inhibitors of Protein Kinase A Resulting in a Boronic Acid Glutamate Linkage
Acs Omega, 2019
7TFM
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BU of 7tfm by Molmil
Atomic Structure of the Leishmania spp. Hsp100 N-Domain
分子名称: ATP-dependent Clp protease subunit, heat shock protein 100 (HSP100), GLYCEROL
著者Mercado, J.M, Lee, S, Chang, C, Sung, N, Soong, L, Catic, A, Tsai, F.T.F.
登録日2022-01-06
公開日2022-02-16
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.055 Å)
主引用文献Atomic structure of the Leishmania spp. Hsp100 N-domain.
Proteins, 90, 2022
6WFV
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BU of 6wfv by Molmil
The crystal structure of a collagen galactosylhydroxylysyl glucosyltransferase from human
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, MAGNESIUM ION, MANGANESE (II) ION, ...
著者Guo, H.-F, Tsai, C.-L, Miller, M.D, Phillips Jr, G.N, Tainer, J.A, Kurie, J.M.
登録日2020-04-04
公開日2021-04-14
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The crystal structure of a collagen galactosylhydroxylysyl glucosyltransferase from human
To Be Published
6WJL
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BU of 6wjl by Molmil
Crystal structure of Glypican-2 core protein in complex with D3 Fab
分子名称: D3 Fab Heavy chain, D3 Fab Light Chain, Glypican-2, ...
著者Raman, S, Maris, J.M, Bosse, K.R, Julien, J.P.
登録日2020-04-14
公開日2021-04-21
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献A GPC2 antibody-drug conjugate is efficacious against neuroblastoma and small-cell lung cancer via binding a conformational epitope.
Cell Rep Med, 2, 2021
7B8W
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BU of 7b8w by Molmil
Structure of LIMK1 Kinase domain with allosteric inhibitor TH-470
分子名称: 1,2-ETHANEDIOL, 2-(2-methylpropanoylamino)-~{N}-[2-[(phenylmethyl)-[4-(phenylsulfamoyl)phenyl]carbonyl-amino]ethyl]-1,3-thiazole-5-carboxamide, LIM domain kinase 1
著者Lee, H, Yosaatmadja, Y, Burgess-Brown, N.A, von Delft, F, Arrowsmith, C.H, Edwards, A, Bountra, C, Elkins, J.M.
登録日2020-12-13
公開日2022-03-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of LIMK1 Kinase domain with allosteric inhibitor TH-470
To Be Published
7CW3
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BU of 7cw3 by Molmil
Cryo-EM structure of Chikungunya virus in complex with mAb CHK-263 IgG (subregion around icosahedral 2-fold vertex)
分子名称: Capsid protein, E1 glycoprotein, E2 glycoprotein, ...
著者Zhou, Q.F, Fox, J.M, Earnest, J.T, Ng, T.S, Kim, A.S, Fibriansah, G, Kostyuchenko, V.A, Shu, B, Diamond, M.S, Lok, S.M.
登録日2020-08-27
公開日2020-11-04
最終更新日2024-03-27
実験手法ELECTRON MICROSCOPY (9.4 Å)
主引用文献Structural basis of Chikungunya virus inhibition by monoclonal antibodies.
Proc.Natl.Acad.Sci.USA, 117, 2020
6XGR
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BU of 6xgr by Molmil
YSD1 major tail protein
分子名称: YSD1_22 major tail protein
著者Hardy, J.M, Dunstan, R, Venugopal, H, Lithgow, T.J, Coulibaly, F.J.
登録日2020-06-17
公開日2020-07-01
最終更新日2023-11-29
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献The architecture and stabilisation of flagellotropic tailed bacteriophages.
Nat Commun, 11, 2020
6X6K
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BU of 6x6k by Molmil
Cryo-EM Structure of the Helicobacter pylori dCag3 OMC
分子名称: Cag pathogenicity island protein, Cag pathogenicity island protein (Cag7), Type IV secretion system apparatus protein CagX
著者Sheedlo, M.J, Chung, J.M, Sawhney, N, Durie, C.L, Cover, T.L, Ohi, M.D, Lacy, D.B.
登録日2020-05-28
公開日2020-10-07
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Cryo-EM reveals species-specific components within the Helicobacter pylori Cag type IV secretion system core complex.
Elife, 9, 2020
6X9L
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BU of 6x9l by Molmil
Crystal Structure of Aldehyde Dehydrogenase C (AldC) mutant (C291A) from Pseudomonas syringae in complexed with NAD+ and Octanal
分子名称: Aldehyde dehydrogenase family protein, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, OCTANAL
著者Lee, S.G, Jez, J.M.
登録日2020-06-03
公開日2020-09-09
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.52 Å)
主引用文献The plant pathogen enzyme AldC is a long-chain aliphatic aldehyde dehydrogenase.
J.Biol.Chem., 295, 2020
7CN9
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BU of 7cn9 by Molmil
Cryo-EM structure of SARS-CoV-2 Spike ectodomain
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Ho, M, Chang, Y, Wang, C, Wu, Y, Huang, H, Chen, T, Lo, J.M, Chen, X, Ma, C.
登録日2020-07-30
公開日2020-08-26
最終更新日2021-03-10
実験手法ELECTRON MICROSCOPY (4.7 Å)
主引用文献A Carbohydrate-Binding Protein from the Edible Lablab Beans Effectively Blocks the Infections of Influenza Viruses and SARS-CoV-2.
Cell Rep, 32, 2020
6X66
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BU of 6x66 by Molmil
Legionella pneumophila dDot T4SS OMC
分子名称: DotC, DotD, Inner membrane lipoprotein YiaD, ...
著者Durie, C.L, Sheedlo, M.J, Chung, J.M, Byrne, B.G, Su, M, Knight, T, Swanson, M.S, Lacy, D.B, Ohi, M.D.
登録日2020-05-27
公開日2020-10-28
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (4.2 Å)
主引用文献Structural analysis of the Legionella pneumophila Dot/Icm type IV secretion system core complex.
Elife, 9, 2020
6X6J
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BU of 6x6j by Molmil
Cryo-EM Structure of CagX and CagY within the Helicobacter pylori PR
分子名称: Cag pathogenicity island protein (Cag7), Cag pathogenicity island protein (Cag8)
著者Sheedlo, M.J, Chung, J.M, Sawhney, N, Durie, C.L, Cover, T.L, Ohi, M.D, Lacy, D.B.
登録日2020-05-28
公開日2020-09-30
最終更新日2021-04-14
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Cryo-EM reveals species-specific components within the Helicobacter pylori Cag type IV secretion system core complex.
Elife, 9, 2020
7CW0
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BU of 7cw0 by Molmil
Cryo-EM structure of Chikungunya virus in complex with mAb CHK-263 IgG
分子名称: Capsid protein, E1 glycoprotein, E2 glycoprotein, ...
著者Zhou, Q.F, Fox, J.M, Earnest, J.T, Ng, T.S, Kim, A.S, Fibriansah, G, Kostyuchenko, V.A, Shu, B, Diamond, M.S, Lok, S.M.
登録日2020-08-27
公開日2020-11-04
最終更新日2024-03-27
実験手法ELECTRON MICROSCOPY (5.9 Å)
主引用文献Structural basis of Chikungunya virus inhibition by monoclonal antibodies.
Proc.Natl.Acad.Sci.USA, 117, 2020
6X62
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Legionella pneumophila Dot T4SS OMC
分子名称: DotC, DotD, Inner membrane lipoprotein YiaD, ...
著者Durie, C.L, Sheedlo, M.J, Chung, J.M, Byrne, B.G, Su, M, Knight, T, Swanson, M.S, Lacy, D.B, Ohi, M.D.
登録日2020-05-27
公開日2020-09-30
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structural analysis of the Legionella pneumophila Dot/Icm type IV secretion system core complex.
Elife, 9, 2020
6XD3
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BU of 6xd3 by Molmil
Structure of the human CAK in complex with THZ1
分子名称: CDK-activating kinase assembly factor MAT1, Cyclin-H, Cyclin-dependent kinase 7, ...
著者Greber, B.J, Perez-Bertoldi, J.M, Lim, K, Iavarone, A.T, Toso, D.B, Nogales, E.
登録日2020-06-09
公開日2020-09-09
最終更新日2020-09-30
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献The cryoelectron microscopy structure of the human CDK-activating kinase.
Proc.Natl.Acad.Sci.USA, 117, 2020
6XGQ
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BU of 6xgq by Molmil
YSD1 bacteriophage capsid
分子名称: YSD1_16, YSD1_17
著者Hardy, J.M, Dunstan, R, Venugopal, H, Lithgow, T.J, Coulibaly, F.J.
登録日2020-06-17
公開日2020-07-01
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献The architecture and stabilisation of flagellotropic tailed bacteriophages.
Nat Commun, 11, 2020
6X65
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BU of 6x65 by Molmil
Legionella pneumophila Dot/Icm T4SS
分子名称: DotC, DotD, Inner membrane lipoprotein YiaD, ...
著者Durie, C.L, Sheedlo, M.J, Chung, J.M, Byrne, B.G, Su, M, Knight, T, Swanson, M.S, Lacy, D.B, Ohi, M.D.
登録日2020-05-27
公開日2020-10-07
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Structural analysis of the Legionella pneumophila Dot/Icm type IV secretion system core complex.
Elife, 9, 2020
6XPH
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BU of 6xph by Molmil
CutR dimer with domain swap
分子名称: Ethanolamine utilization protein EutS, GLYCEROL, POTASSIUM ION, ...
著者Ochoa, J.M, Sawaya, M.R, Nguyen, V.N, Duilio, C, Yeates, T.O, Nie, M.
登録日2020-07-08
公開日2020-07-22
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Symmetry breaking and structural polymorphism in a bacterial microcompartment shell protein for choline utilization.
Protein Sci., 29, 2020
6X64
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Legionella pneumophila Dot T4SS PR
分子名称: Type IV secretion system unknown protein fragment
著者Durie, C.L, Sheedlo, M.J, Chung, J.M, Byrne, B.G, Su, M, Knight, T, Swanson, M.S, Lacy, D.B, Ohi, M.D.
登録日2020-05-27
公開日2020-10-07
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Structural analysis of the Legionella pneumophila Dot/Icm type IV secretion system core complex.
Elife, 9, 2020

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